US20090298179A1
(en)
*
|
2003-04-29 |
2009-12-03 |
Connie Erickson-Miller |
Methods For Treating Degenerative Diseases/Injuries
|
US20090143453A1
(en)
*
|
2003-04-29 |
2009-06-04 |
Connie Erickson-Miller |
Methods for treating degenerative diseases/injuries
|
JP4895807B2
(ja)
*
|
2003-04-29 |
2012-03-14 |
グラクソスミスクライン・リミテッド・ライアビリティ・カンパニー |
変性疾患/損傷の治療方法
|
US20090048318A1
(en)
*
|
2003-04-29 |
2009-02-19 |
Connie Erickson-Miller |
Methods for treating degenerative diseases/injuries
|
US8354427B2
(en)
*
|
2004-06-24 |
2013-01-15 |
Vertex Pharmaceutical Incorporated |
Modulators of ATP-binding cassette transporters
|
US7625890B2
(en)
*
|
2005-11-10 |
2009-12-01 |
Smithkline Beecham Corp. |
Substituted imidazo[4,5-c]pyridine compounds as Akt inhibitors
|
MY159449A
(en)
*
|
2005-12-13 |
2017-01-13 |
Incyte Holdings Corp |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as janus kinase inhibitors
|
CA2634787C
(en)
*
|
2005-12-23 |
2014-10-21 |
Smithkline Beecham Corporation |
Azaindole inhibitors of aurora kinases
|
EP1998777A1
(en)
*
|
2006-03-20 |
2008-12-10 |
F. Hoffmann-La Roche AG |
Methods of inhibiting btk and syk protein kinases
|
CL2007003244A1
(es)
|
2006-11-16 |
2008-04-04 |
Millennium Pharm Inc |
Compuestos derivados de pirimido[5,4-d][2]benzazepina; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento del cancer.
|
UY30892A1
(es)
|
2007-02-07 |
2008-09-02 |
Smithkline Beckman Corp |
Inhibidores de la actividad akt
|
TR201903488T4
(tr)
|
2007-06-13 |
2019-04-22 |
Incyte Holdings Corp |
Janus kinaz inhibitörü (r)-3-(4-(7h-pirolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)-3-siklopentilpropannitril tuzlarının kullanımı.
|
AR070127A1
(es)
*
|
2008-01-11 |
2010-03-17 |
Novartis Ag |
Pirrolo - pirimidinas y pirrolo -piridinas
|
CN102014627B
(zh)
|
2008-04-30 |
2014-10-29 |
国家卫生研究院 |
作为极光激酶抑制剂的稠合双环嘧啶化合物
|
CL2009001884A1
(es)
*
|
2008-10-02 |
2010-05-14 |
Incyte Holdings Corp |
Uso de 3-ciclopentil-3-[4-(7h-pirrolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)propanonitrilo, inhibidor de janus quinasa, y uso de una composición que lo comprende para el tratamiento del ojo seco.
|
EP2344484B1
(en)
*
|
2008-10-17 |
2016-06-08 |
Akaal Pharma Pty Ltd |
S1p receptors modulators and use thereof
|
EP2344446A4
(en)
|
2008-10-17 |
2012-04-04 |
Akaal Pharma Pty Ltd |
S1P RECEPTOR MODULATORS
|
DE102008052943A1
(de)
|
2008-10-23 |
2010-04-29 |
Merck Patent Gmbh |
Azaindolderivate
|
EP2198710A1
(de)
|
2008-12-19 |
2010-06-23 |
Bayer CropScience AG |
Verwendung von 5-Pyridin-4yl-(1,3)Thiazole zur Bekämpfung phytopathogener Pilze
|
MX2011006725A
(es)
*
|
2008-12-22 |
2011-09-15 |
Millennium Pharm Inc |
Combinacion de inhibidores de aurora cinasa y anticuerpos anti-cd20.
|
MY161598A
(en)
*
|
2009-01-30 |
2017-04-28 |
Glaxosmithkline Llc |
Crystalline n-{ (1s)-2-amino-1-[(3-fluorophenyl)methyl]ethyl} -5-chloro-4-(4-chloro-1-methyl-1h-pyrazol-5-yl)-2-thiophenecarboxamide hydrochloride
|
JO3635B1
(ar)
|
2009-05-18 |
2020-08-27 |
Millennium Pharm Inc |
مركبات صيدلانية صلبة وطرق لانتاجها
|
WO2010135650A1
(en)
|
2009-05-22 |
2010-11-25 |
Incyte Corporation |
N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS
|
AR076920A1
(es)
|
2009-05-22 |
2011-07-20 |
Incyte Corp |
3-(4-(7h-pirrolo(2,3-d)pirimidin-4-il)-1h-pirazol-1-il)octano-o heptano--nitrilo como inhibidores de jak
|
JO3434B1
(ar)
*
|
2009-07-31 |
2019-10-20 |
Millennium Pharm Inc |
مركبات صيدلانية لمعالجة السرطان وامراض واضطرابات اخري
|
EA201290073A1
(ru)
|
2009-08-24 |
2013-01-30 |
Эсэпиен Фармасьютикалз, Инк. |
Соединения мочевины, содержащие 5,6-бициклический гетероарил, как ингибиторы киназ
|
AR078012A1
(es)
*
|
2009-09-01 |
2011-10-05 |
Incyte Corp |
Derivados heterociclicos de las pirazol-4-il- pirrolo (2,3-d) pirimidinas como inhibidores de la quinasa janus
|
EP2308866A1
(de)
*
|
2009-10-09 |
2011-04-13 |
Bayer CropScience AG |
Phenylpyri(mi)dinylpyrazole und ihre Verwendung als Fungizide
|
CA2777108A1
(en)
|
2009-10-09 |
2011-04-14 |
Zafgen Corporation |
Sulphone compounds and methods of making and using same
|
US8653064B2
(en)
|
2010-02-19 |
2014-02-18 |
Millennium Pharmaceuticals, Inc. |
Crystalline forms of sodium 4-{[9-chloro-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-D][2]benzazepin-2-yl]amino}-2-methoxybenzoate
|
PT3050882T
(pt)
*
|
2010-03-10 |
2018-04-16 |
Incyte Holdings Corp |
Derivados de piperidin-4-ilazetidina como inibidores de jak1
|
CN103154246B
(zh)
|
2010-05-14 |
2015-11-25 |
达那-法伯癌症研究所 |
用于治疗白血病的组合物和方法
|
JP6022442B2
(ja)
|
2010-05-14 |
2016-11-09 |
ダナ−ファーバー キャンサー インスティテュート, インコーポレイテッド |
男性用避妊組成物および使用方法
|
PT2571503E
(pt)
|
2010-05-14 |
2015-04-29 |
Dana Farber Cancer Inst Inc |
Composições e a sua utilização no tratamento de neoplasia, doença inflamatória e outros distúrbios
|
EP2574168B9
(en)
|
2010-05-21 |
2016-10-05 |
Incyte Holdings Corporation |
Topical formulation for a jak inhibitor
|
BR112013001613A2
(pt)
|
2010-07-22 |
2016-05-24 |
Zafgen Inc |
compostos tricíclicos e métodos para fazer e usar os mesmos.
|
CA2818545C
(en)
|
2010-11-19 |
2019-04-16 |
Incyte Corporation |
Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors
|
AU2011329734B2
(en)
|
2010-11-19 |
2015-05-28 |
Incyte Holdings Corporation |
Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as JAK inhibitors
|
JP6058557B2
(ja)
|
2011-01-26 |
2017-01-11 |
ザフゲン,インコーポレイテッド |
テトラゾール化合物ならびにその作製方法および使用方法
|
EA025526B1
(ru)
|
2011-05-06 |
2017-01-30 |
Зафджен Инк. |
Частично насыщенные трициклические соединения и способы их получения и применения
|
KR20140053013A
(ko)
|
2011-05-06 |
2014-05-07 |
자프겐 인크. |
삼환식 설폰아마이드 화합물 그리고 그의 제조방법 및 그를 이용하는 방법
|
AU2012253760B2
(en)
|
2011-05-06 |
2016-02-04 |
Zafgen, Inc. |
Tricyclic pyrazole sulfonamide compounds and methods of making and using same
|
ES2560611T3
(es)
|
2011-06-20 |
2016-02-22 |
Incyte Holdings Corporation |
Derivados de fenil de azetidinilo, carboxamida de piridilo o pirazinilo como inhibidores de JAK
|
TW201313721A
(zh)
|
2011-08-18 |
2013-04-01 |
Incyte Corp |
作為jak抑制劑之環己基氮雜環丁烷衍生物
|
UA111854C2
(uk)
|
2011-09-07 |
2016-06-24 |
Інсайт Холдінгс Корпорейшн |
Способи і проміжні сполуки для отримання інгібіторів jak
|
AU2013209723B2
(en)
|
2012-01-18 |
2016-11-24 |
Zafgen, Inc. |
Tricyclic sulfonamide compounds and methods of making and using same
|
CA2861381A1
(en)
|
2012-01-18 |
2013-07-25 |
Zafgen, Inc. |
Tricyclic sulfone compounds and methods of making and using same
|
US20130303519A1
(en)
|
2012-03-20 |
2013-11-14 |
Millennium Pharmaceuticals, Inc. |
Methods of treating cancer using aurora kinase inhibitors
|
TW201406761A
(zh)
|
2012-05-18 |
2014-02-16 |
Incyte Corp |
做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
|
JP6189948B2
(ja)
|
2012-06-29 |
2017-08-30 |
ファイザー・インク |
LRRK2阻害薬としての新規な4−(置換アミノ)−7H−ピロロ[2,3−d]ピリミジン
|
CN103664936A
(zh)
*
|
2012-09-17 |
2014-03-26 |
杨育新 |
一类治疗创伤性脑损伤疾病的化合物及其用途
|
CN103800345A
(zh)
*
|
2012-11-02 |
2014-05-21 |
常辉 |
一类治疗精神分裂症的化合物及其用途
|
CN104918615B
(zh)
|
2012-11-05 |
2018-10-12 |
扎夫根股份有限公司 |
治疗肝病的方法
|
BR112015010225A2
(pt)
|
2012-11-05 |
2017-07-11 |
Zafgen Inc |
compostos tricíclicos e seus métodos de produção e utilização
|
EP2925737B1
(en)
|
2012-11-05 |
2017-06-14 |
Zafgen, Inc. |
Tricyclic compounds for use in the treatment and/or control of obesity
|
BR112015010663B1
(pt)
|
2012-11-15 |
2022-12-06 |
Incyte Holdings Corporation |
Formas de dosagem oral de liberação sustentada, e uso de ruxolitinib ou de sal farmaceuticamente aceitável do mesmo
|
AR094929A1
(es)
|
2013-02-28 |
2015-09-09 |
Bristol Myers Squibb Co |
Derivados de fenilpirazol como inhibidores potentes de rock1 y rock2
|
WO2014134391A1
(en)
|
2013-02-28 |
2014-09-04 |
Bristol-Myers Squibb Company |
Phenylpyrazole derivatives as potent rock1 and rock2 inhibitors
|
UA121532C2
(uk)
|
2013-03-06 |
2020-06-10 |
Інсайт Холдінгс Корпорейшн |
Способи і проміжні сполуки при отриманні інгібітора jak
|
JP2016514113A
(ja)
|
2013-03-14 |
2016-05-19 |
アッヴィ・インコーポレイテッド |
ピロロ[2,3−b]ピリジンcdk9キナーゼ阻害剤
|
TW201444836A
(zh)
*
|
2013-03-14 |
2014-12-01 |
Abbvie Inc |
吡咯并[2,3-b]吡啶cdk9激酶抑制劑
|
CN105209042B
(zh)
|
2013-03-22 |
2019-03-08 |
米伦纽姆医药公司 |
催化性mtorc 1/2抑制剂与选择性极光a激酶抑制剂的组合
|
RU2016105108A
(ru)
|
2013-07-25 |
2017-08-30 |
Дана-Фарбер Кэнсер Инститьют, Инк. |
Ингибиторы факторов транскрипции и их применение
|
EP3721873A1
(en)
|
2013-08-07 |
2020-10-14 |
Incyte Corporation |
Sustained release dosage forms for a jak1 inhibitor
|
WO2015070020A2
(en)
|
2013-11-08 |
2015-05-14 |
Dana-Farber Cancer Institute, Inc. |
Combination therapy for cancer using bromodomain and extra-terminal (bet) protein inhibitors
|
US9695171B2
(en)
|
2013-12-17 |
2017-07-04 |
Pfizer Inc. |
3,4-disubstituted-1 H-pyrrolo[2,3-b]pyridines and 4,5-disubstituted-7H-pyrrolo[2,3-c]pyridazines as LRRK2 inhibitors
|
KR20160115953A
(ko)
|
2014-01-31 |
2016-10-06 |
다나-파버 캔서 인스티튜트 인크. |
디아미노피리미딘 벤젠술폰 유도체 및 그의 용도
|
JP2017504651A
(ja)
|
2014-01-31 |
2017-02-09 |
ダナ−ファーバー キャンサー インスティテュート, インコーポレイテッド |
ジアゼパン誘導体の使用
|
MX2016011160A
(es)
|
2014-02-28 |
2017-04-27 |
Tensha Therapeutics Inc |
Tratamiento de afecciones asociadas con la hiperinsulinemia.
|
US9498467B2
(en)
|
2014-05-30 |
2016-11-22 |
Incyte Corporation |
Treatment of chronic neutrophilic leukemia (CNL) and atypical chronic myeloid leukemia (aCML) by inhibitors of JAK1
|
JP2017525759A
(ja)
|
2014-08-08 |
2017-09-07 |
ダナ−ファーバー キャンサー インスティテュート, インコーポレイテッド |
ジヒドロプテリジノン誘導体およびその使用
|
BR112017002369A2
(pt)
|
2014-08-08 |
2017-12-05 |
Dana Farber Cancer Inst Inc |
derivados de diazepana e usos dos mesmos
|
EP3212654B1
(en)
|
2014-10-27 |
2020-04-08 |
Tensha Therapeutics, Inc. |
Bromodomain inhibitors
|
EA037112B1
(ru)
*
|
2015-03-02 |
2021-02-08 |
Ригель Фармасьютикалс, Инк. |
Ингибиторы tgf-
|
EP3307728A4
(en)
|
2015-06-12 |
2019-07-17 |
Dana Farber Cancer Institute, Inc. |
ASSOCIATION THERAPY USING TRANSCRIPTION INHIBITORS AND KINASE INHIBITORS
|
JP2018524292A
(ja)
|
2015-07-21 |
2018-08-30 |
ミレニアム ファーマシューティカルズ, インコーポレイテッドMillennium Pharmaceuticals, Inc. |
オーロラキナーゼインヒビターと化学療法剤の投与
|
JP2018526421A
(ja)
|
2015-09-11 |
2018-09-13 |
ダナ−ファーバー キャンサー インスティテュート, インコーポレイテッド |
シアノチエノトリアゾロジアゼピンおよびこれらの使用
|
SG10202007099TA
(en)
|
2015-09-11 |
2020-08-28 |
Dana Farber Cancer Inst Inc |
Acetamide thienotriazoldiazepines and uses thereof
|
RU2722149C1
(ru)
|
2015-09-14 |
2020-05-27 |
Пфайзер Инк. |
Новые производные имидазо[4,5-c] хинолинов и имидазо[4,5-c][1,5] нафтиридинов в качестве ингибиторов LRRK2
|
EP3380100A4
(en)
|
2015-11-25 |
2019-10-02 |
Dana-Farber Cancer Institute, Inc. |
BIVALENT BROMODOMAIN INHIBITORS AND USES THEREOF
|
US10596161B2
(en)
|
2017-12-08 |
2020-03-24 |
Incyte Corporation |
Low dose combination therapy for treatment of myeloproliferative neoplasms
|
EA202091830A1
(ru)
|
2018-01-30 |
2020-12-29 |
Инсайт Корпорейшн |
Способы и промежуточные соединения для получения ингибитора jak
|
MA52219A
(fr)
|
2018-03-30 |
2021-02-17 |
Incyte Corp |
Traitement de l'hidradénite suppurée à l'aide d'inhibiteurs de jak
|
WO2020223456A1
(en)
*
|
2019-05-01 |
2020-11-05 |
Nemucore Medical Innovations, Inc. |
Degradation of aurora kinase (aurk) by conjugation of aurk inhibitors with e3 ligase ligand
|
CN114008046B
(zh)
*
|
2019-06-27 |
2023-08-18 |
南京明德新药研发有限公司 |
作为cdk9抑制剂的氮杂吲哚连吡唑类化合物
|
US11833155B2
(en)
|
2020-06-03 |
2023-12-05 |
Incyte Corporation |
Combination therapy for treatment of myeloproliferative neoplasms
|
CN112225723B
(zh)
*
|
2020-12-16 |
2021-03-30 |
北京华氏开元医药科技有限公司 |
一种吲哚类衍生物、制备方法及应用
|
CN116685588A
(zh)
*
|
2020-12-25 |
2023-09-01 |
南京明德新药研发有限公司 |
吡啶并吡咯类化合物的晶型、制备方法及其应用
|
CN115572294B
(zh)
*
|
2022-11-13 |
2023-11-21 |
药康众拓(江苏)医药科技有限公司 |
一种氘代氮杂吲哚联吡唑类化合物、药物组合物和用途
|