TWI343920B - 2 - (pyridin -2- ylamino)- pyrido [2,3-d] pyrimidin -7-ones - Google Patents

2 - (pyridin -2- ylamino)- pyrido [2,3-d] pyrimidin -7-ones Download PDF

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Publication number
TWI343920B
TWI343920B TW092101242A TW92101242A TWI343920B TW I343920 B TWI343920 B TW I343920B TW 092101242 A TW092101242 A TW 092101242A TW 92101242 A TW92101242 A TW 92101242A TW I343920 B TWI343920 B TW I343920B
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Taiwan
Prior art keywords
ylamino
cyclopentyl
pyrido
pyrimidin
methyl
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TW092101242A
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English (en)
Chinese (zh)
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TW200302224A (en
Inventor
Robert Barvian Mark
John Booth Richard
Quin John Iii
Thomas Repine Joseph
James Sheehan Derek
Laurence Toogood Peter
Norman Vanderwel Scott
Zhou Hairong
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Warner Lambert Co
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Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of TW200302224A publication Critical patent/TW200302224A/zh
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/675—Phosphorus compounds having nitrogen as a ring hetero atom, e.g. pyridoxal phosphate
    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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TW092101242A 2002-01-22 2003-01-21 2 - (pyridin -2- ylamino)- pyrido [2,3-d] pyrimidin -7-ones TWI343920B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US35087702P 2002-01-22 2002-01-22

Publications (2)

Publication Number Publication Date
TW200302224A TW200302224A (en) 2003-08-01
TWI343920B true TWI343920B (en) 2011-06-21

Family

ID=27613435

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TW092101242A TWI343920B (en) 2002-01-22 2003-01-21 2 - (pyridin -2- ylamino)- pyrido [2,3-d] pyrimidin -7-ones

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US (4) US6936612B2 (enExample)
EP (1) EP1470124B1 (enExample)
JP (1) JP4291696B2 (enExample)
KR (2) KR20060111716A (enExample)
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CR (1) CR20120129A (enExample)
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TW (1) TWI343920B (enExample)
UA (1) UA79444C2 (enExample)
UY (1) UY27617A1 (enExample)
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KR20090052385A (ko) 2006-09-08 2009-05-25 화이자 프로덕츠 인크. 2-（피리딘-2-일아미노）-피리도［2,3-ｄ］피리미딘-7-온의합성

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