SK51197A3 - Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitiors - Google Patents

Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitiors Download PDF

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Publication number
SK51197A3
SK51197A3 SK511-97A SK51197A SK51197A3 SK 51197 A3 SK51197 A3 SK 51197A3 SK 51197 A SK51197 A SK 51197A SK 51197 A3 SK51197 A3 SK 51197A3
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Slovakia
Prior art keywords
carbon atoms
group
phenyl
aryl
moiety contains
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SK511-97A
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English (en)
Slovak (sk)
Inventor
Harold C E Kluender
Guenter Hans H H Benz
David R Brittelli
William H Bullock
Kerry J Combs
Brian R Dixon
Stephan Schneider
Jill E Wood
Michael C Vanzandt
Donald J Wolanin
Scott M Wilhelm
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Bayer Ag
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Publication of SK51197A3 publication Critical patent/SK51197A3/sk

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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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SK511-97A 1994-11-15 1995-11-09 Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitiors SK51197A3 (en)

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