IS4480A - Útskiptar 4-biarylbutyric- eða 5-biarylpentanoic-sýrur og afleiður þeirra sem hindra virkni bandvefsmálmpróteasa - Google Patents

Útskiptar 4-biarylbutyric- eða 5-biarylpentanoic-sýrur og afleiður þeirra sem hindra virkni bandvefsmálmpróteasa

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Publication number
IS4480A
IS4480A IS4480A IS4480A IS4480A IS 4480 A IS4480 A IS 4480A IS 4480 A IS4480 A IS 4480A IS 4480 A IS4480 A IS 4480A IS 4480 A IS4480 A IS 4480A
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IS
Iceland
Prior art keywords
biarylbutyric
inhibit
derivatives
activity
replaced
Prior art date
Application number
IS4480A
Other languages
English (en)
Inventor
C. E. Kluender Harold
H. H. H. Benz Guenter
R. Brittelli David
H. Bullock William
J. Combs Kerry
R. Dixon Brian
Schneider Stephan
E. Wood Jill
C. Vanzandt Michael
J. Wolanin Donald
M. Wilhelm Scott
Original Assignee
Bayer Corporation
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Publication date
Application filed by Bayer Corporation filed Critical Bayer Corporation
Publication of IS4480A publication Critical patent/IS4480A/is

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    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
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    • A61K31/19—Carboxylic acids, e.g. valproic acid
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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IS4480A 1994-11-15 1997-05-12 Útskiptar 4-biarylbutyric- eða 5-biarylpentanoic-sýrur og afleiður þeirra sem hindra virkni bandvefsmálmpróteasa IS4480A (is)

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US5861428A (en) 1999-01-19
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MA26357A1 (fr) 2004-11-01
BR9509686A (pt) 1997-09-30
JPH10509146A (ja) 1998-09-08
NZ297174A (en) 2001-04-27
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CZ147797A3 (cs) 1998-02-18
DZ1943A1 (fr) 2002-02-17
US5859047A (en) 1999-01-12
US5789434A (en) 1998-08-04
US5886024A (en) 1999-03-23
EE03435B1 (et) 2001-06-15
US5861427A (en) 1999-01-19
ZA959647B (en) 1997-08-14
DE69527798T2 (de) 2003-01-02
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CA2201863A1 (en) 1996-05-23
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ATE222230T1 (de) 2002-08-15
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