SG178454A1 - Heterocyclic compounds and uses thereof - Google Patents

Heterocyclic compounds and uses thereof Download PDF

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Publication number
SG178454A1
SG178454A1 SG2012010849A SG2012010849A SG178454A1 SG 178454 A1 SG178454 A1 SG 178454A1 SG 2012010849 A SG2012010849 A SG 2012010849A SG 2012010849 A SG2012010849 A SG 2012010849A SG 178454 A1 SG178454 A1 SG 178454A1
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SG
Singapore
Prior art keywords
alkyl
compound
heteroaryl
aryl
taken together
Prior art date
Application number
SG2012010849A
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English (en)
Inventor
Pingda Ren
Yi Liu
Liansheng Li
Katrina Chan
Troy Edward Wilson
Simon Fraser Campbell
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Intellikine Inc
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43607312&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG178454(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Intellikine Inc filed Critical Intellikine Inc
Publication of SG178454A1 publication Critical patent/SG178454A1/en

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/423—Oxazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
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    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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