PL2486029T3 - Sposoby otrzymywania podstawionych glukopiranozylem pochodnych benzylo-benzenowych - Google Patents

Sposoby otrzymywania podstawionych glukopiranozylem pochodnych benzylo-benzenowych

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Publication number
PL2486029T3
PL2486029T3 PL10762899T PL10762899T PL2486029T3 PL 2486029 T3 PL2486029 T3 PL 2486029T3 PL 10762899 T PL10762899 T PL 10762899T PL 10762899 T PL10762899 T PL 10762899T PL 2486029 T3 PL2486029 T3 PL 2486029T3
Authority
PL
Poland
Prior art keywords
glucopyranosyl
preparing
processes
substituted benzyl
benzene derivatives
Prior art date
Application number
PL10762899T
Other languages
English (en)
Polish (pl)
Inventor
Dirk Weber
Tobias Fiedler
Christian Filser
Rainer Hamm
Simone Orlich
Matthias Post
Svenja Renner
Xiao-Jun Wang
Thomas Wirth
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of PL2486029T3 publication Critical patent/PL2486029T3/pl

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10Oxygen atoms
    • C07D309/12Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26Acyclic or carbocyclic radicals, substituted by hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • C07H1/06Separation; Purification
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04Carbocyclic radicals

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Molecular Biology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Packaging Of Annular Or Rod-Shaped Articles, Wearing Apparel, Cassettes, Or The Like (AREA)
  • Wrapping Of Specific Fragile Articles (AREA)
PL10762899T 2009-09-30 2010-09-24 Sposoby otrzymywania podstawionych glukopiranozylem pochodnych benzylo-benzenowych PL2486029T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24714409P 2009-09-30 2009-09-30
EP10762899.2A EP2486029B1 (en) 2009-09-30 2010-09-24 Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives
PCT/EP2010/064120 WO2011039108A2 (en) 2009-09-30 2010-09-24 Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives

Publications (1)

Publication Number Publication Date
PL2486029T3 true PL2486029T3 (pl) 2015-11-30

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ID=43736212

Family Applications (1)

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PL10762899T PL2486029T3 (pl) 2009-09-30 2010-09-24 Sposoby otrzymywania podstawionych glukopiranozylem pochodnych benzylo-benzenowych

Country Status (25)

Country Link
US (2) US9024010B2 (en0)
EP (1) EP2486029B1 (en0)
JP (1) JP5758900B2 (en0)
KR (1) KR101813025B1 (en0)
CN (1) CN102574829B (en0)
AR (1) AR078193A1 (en0)
AU (1) AU2010303124B2 (en0)
BR (1) BR112012007085B8 (en0)
CA (1) CA2775962C (en0)
CL (1) CL2012000581A1 (en0)
DK (1) DK2486029T3 (en0)
EA (1) EA022032B1 (en0)
ES (1) ES2546762T3 (en0)
HR (1) HRP20150945T1 (en0)
HU (1) HUE026133T2 (en0)
IL (1) IL218101A0 (en0)
IN (1) IN2012DN02751A (en0)
MX (1) MX2012003048A (en0)
NZ (1) NZ598366A (en0)
PH (1) PH12012500634A1 (en0)
PL (1) PL2486029T3 (en0)
PT (1) PT2486029E (en0)
SI (1) SI2486029T1 (en0)
TW (1) TWI465458B (en0)
WO (1) WO2011039108A2 (en0)

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ES2546762T3 (es) 2015-09-28
BR112012007085A2 (pt) 2015-09-15
AU2010303124A1 (en) 2012-03-15
JP5758900B2 (ja) 2015-08-05
CA2775962C (en) 2017-09-05
CL2012000581A1 (es) 2012-08-03
NZ598366A (en) 2014-03-28
PT2486029E (pt) 2015-10-14
WO2011039108A2 (en) 2011-04-07
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BR112012007085B1 (pt) 2020-10-13
EA201200537A1 (ru) 2012-11-30
CA2775962A1 (en) 2011-04-07
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AR078193A1 (es) 2011-10-19
EP2486029A2 (en) 2012-08-15
SI2486029T1 (sl) 2015-10-30
CN102574829B (zh) 2015-07-01
US9024010B2 (en) 2015-05-05
AU2010303124B2 (en) 2014-01-23
KR20120081592A (ko) 2012-07-19
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US9873714B2 (en) 2018-01-23
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TWI465458B (zh) 2014-12-21
BR112012007085B8 (pt) 2021-05-25

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