SI2486029T1 - Postopki za pripravo z glukopiranozilom substituiranih benzil-benzenskih derivatov - Google Patents

Postopki za pripravo z glukopiranozilom substituiranih benzil-benzenskih derivatov

Info

Publication number
SI2486029T1
SI2486029T1 SI201031009T SI201031009T SI2486029T1 SI 2486029 T1 SI2486029 T1 SI 2486029T1 SI 201031009 T SI201031009 T SI 201031009T SI 201031009 T SI201031009 T SI 201031009T SI 2486029 T1 SI2486029 T1 SI 2486029T1
Authority
SI
Slovenia
Prior art keywords
glucopyranosyl
preparing
processes
substituted benzyl
benzene derivatives
Prior art date
Application number
SI201031009T
Other languages
English (en)
Inventor
Dirk Weber
Tobias Fiedler
Christian Filser
Rainer Hamm
Simone Orlich
Matthias Post
Svenja Renner
Xiao-Jun Wang
Thomas Wirth
Original Assignee
Boehringer Ingelheim International Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim International Gmbh filed Critical Boehringer Ingelheim International Gmbh
Publication of SI2486029T1 publication Critical patent/SI2486029T1/sl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C07D309/12—Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives
    • C07H1/06—Separation; Purification
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals
SI201031009T 2009-09-30 2010-09-24 Postopki za pripravo z glukopiranozilom substituiranih benzil-benzenskih derivatov SI2486029T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US24714409P 2009-09-30 2009-09-30
EP10762899.2A EP2486029B1 (en) 2009-09-30 2010-09-24 Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives
PCT/EP2010/064120 WO2011039108A2 (en) 2009-09-30 2010-09-24 Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives

Publications (1)

Publication Number Publication Date
SI2486029T1 true SI2486029T1 (sl) 2015-10-30

Family

ID=43736212

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201031009T SI2486029T1 (sl) 2009-09-30 2010-09-24 Postopki za pripravo z glukopiranozilom substituiranih benzil-benzenskih derivatov

Country Status (24)

Country Link
US (2) US9024010B2 (sl)
EP (1) EP2486029B1 (sl)
JP (1) JP5758900B2 (sl)
KR (1) KR101813025B1 (sl)
CN (1) CN102574829B (sl)
AR (1) AR078193A1 (sl)
AU (1) AU2010303124B2 (sl)
BR (1) BR112012007085B8 (sl)
CA (1) CA2775962C (sl)
CL (1) CL2012000581A1 (sl)
DK (1) DK2486029T3 (sl)
EA (1) EA022032B1 (sl)
ES (1) ES2546762T3 (sl)
HR (1) HRP20150945T1 (sl)
HU (1) HUE026133T2 (sl)
IL (1) IL218101A0 (sl)
IN (1) IN2012DN02751A (sl)
MX (1) MX2012003048A (sl)
NZ (1) NZ598366A (sl)
PL (1) PL2486029T3 (sl)
PT (1) PT2486029E (sl)
SI (1) SI2486029T1 (sl)
TW (1) TWI465458B (sl)
WO (1) WO2011039108A2 (sl)

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BR112012007085A2 (pt) 2015-09-15
US20150218200A1 (en) 2015-08-06
AU2010303124B2 (en) 2014-01-23
MX2012003048A (es) 2012-05-08
TW201127848A (en) 2011-08-16

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