NO20025091D0 - Oksazolidinonderivater med antibiotisk aktivitet - Google Patents
Oksazolidinonderivater med antibiotisk aktivitetInfo
- Publication number
- NO20025091D0 NO20025091D0 NO20025091A NO20025091A NO20025091D0 NO 20025091 D0 NO20025091 D0 NO 20025091D0 NO 20025091 A NO20025091 A NO 20025091A NO 20025091 A NO20025091 A NO 20025091A NO 20025091 D0 NO20025091 D0 NO 20025091D0
- Authority
- NO
- Norway
- Prior art keywords
- sup
- alkyl
- optionally substituted
- atom
- het
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/10—Spiro-condensed systems
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0009803.8A GB0009803D0 (en) | 2000-04-25 | 2000-04-25 | Chemical compounds |
PCT/GB2001/001815 WO2001081350A1 (en) | 2000-04-25 | 2001-04-23 | Oxazolidinone derivatives with antibiotic activity |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20025091D0 true NO20025091D0 (no) | 2002-10-23 |
NO20025091L NO20025091L (no) | 2002-12-09 |
NO328549B1 NO328549B1 (no) | 2010-03-15 |
Family
ID=9890314
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20025091A NO328549B1 (no) | 2000-04-25 | 2002-10-23 | Oksazolidinonderivater med antibiotisk aktivitet |
Country Status (29)
Country | Link |
---|---|
US (1) | US7141583B2 (no) |
EP (1) | EP1286998B2 (no) |
JP (1) | JP2003531211A (no) |
KR (1) | KR100858771B1 (no) |
CN (1) | CN1277829C (no) |
AT (1) | ATE268778T1 (no) |
AU (1) | AU781784B2 (no) |
BR (1) | BR0110240A (no) |
CA (1) | CA2405349C (no) |
CZ (1) | CZ20023527A3 (no) |
DE (1) | DE60103754T3 (no) |
DK (1) | DK1286998T4 (no) |
EE (1) | EE200200598A (no) |
ES (1) | ES2220759T5 (no) |
GB (1) | GB0009803D0 (no) |
HK (1) | HK1053114A1 (no) |
HU (1) | HUP0300416A2 (no) |
IL (2) | IL152284A0 (no) |
IS (1) | IS6583A (no) |
MX (1) | MXPA02010453A (no) |
NO (1) | NO328549B1 (no) |
NZ (1) | NZ521765A (no) |
PL (1) | PL358326A1 (no) |
PT (1) | PT1286998E (no) |
RU (1) | RU2002131455A (no) |
SI (1) | SI1286998T2 (no) |
TR (1) | TR200402261T4 (no) |
WO (1) | WO2001081350A1 (no) |
ZA (1) | ZA200208187B (no) |
Families Citing this family (54)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0113299D0 (en) * | 2001-06-01 | 2001-07-25 | Astrazeneca Ab | Chemical process & intermediates |
MXPA04002303A (es) | 2001-09-11 | 2004-06-29 | Astrazeneca Ab | Oxazolidinona y/o isoxazolina como agentes antibacterianos. |
WO2003035073A1 (en) | 2001-10-25 | 2003-05-01 | Astrazeneca Ab | Isoxazoline derivatives useful as antimicrobials |
KR100445437B1 (ko) * | 2002-02-08 | 2004-08-21 | 한국과학기술연구원 | 네오마이신-옥사졸리디논 헤테로 이합체, 그의 제조방법및 그의 용도 |
US7141588B2 (en) | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
US7199143B2 (en) | 2002-02-28 | 2007-04-03 | Astrazeneca Ab | Chemical compounds |
CA2477344A1 (en) * | 2002-02-28 | 2003-09-04 | Astrazeneca Ab | 3-cyclyl-5-(nitrogen-containing 5-membered ring) methyl-oxazolidinone derivatives and their use as antibacterial agents |
AU2003259159A1 (en) | 2002-08-12 | 2004-02-25 | Pharmacia & Upjohn Company Llc | N-aryl-2-oxazolidinones and their derivatives |
TW200420573A (en) * | 2002-09-26 | 2004-10-16 | Rib X Pharmaceuticals Inc | Bifunctional heterocyclic compounds and methods of making and using same |
US6875784B2 (en) | 2002-10-09 | 2005-04-05 | Pharmacia & Upjohn Company | Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives |
DE60309504T2 (de) | 2002-11-21 | 2007-05-16 | Pharmacia & Upjohn Co. Llc, Kalamazoo | N-(4-(piperazin-1-yl)-phenyl-2-oxazolidinon-5-carbosäureamid-derivate und verwandte verbindungen als antibakterielle mittel |
EP1581524A2 (en) * | 2002-11-28 | 2005-10-05 | AstraZeneca AB | Oxazolidinones as antibacterial agents |
GB0227701D0 (en) * | 2002-11-28 | 2003-01-08 | Astrazeneca Ab | Chemical compounds |
GB0229522D0 (en) * | 2002-12-19 | 2003-01-22 | Astrazeneca Ab | Chemical compounds |
US7012088B2 (en) | 2003-02-24 | 2006-03-14 | Pharmacia & Upjohn Company | Indolone oxazolidinones and derivatives thereof |
GB0304723D0 (en) * | 2003-03-01 | 2003-04-02 | Astrazeneca Ab | Chemical compounds |
GB0306358D0 (en) * | 2003-03-20 | 2003-04-23 | Astrazeneca Ab | Chemical compounds |
GB0306357D0 (en) | 2003-03-20 | 2003-04-23 | Astrazeneca Ab | Chemical compounds |
EP1615916A1 (en) | 2003-04-09 | 2006-01-18 | Pharmacia & Upjohn Company LLC | Antimicrobial 3.1.0 bicyclohexylphenyl-oxazolidinone derivatives and analogues |
SI1656370T1 (sl) * | 2003-06-03 | 2012-12-31 | Rib-X Pharmaceuticals, Inc. | Biarilne heterociklične spojine in postopki za njihovo izdelavo in uporabo |
US8324398B2 (en) | 2003-06-03 | 2012-12-04 | Rib-X Pharmaceuticals, Inc. | Process for the synthesis of biaryl oxazolidinones |
AR045690A1 (es) * | 2003-06-03 | 2005-11-09 | Rib X Pharmaceuticals Inc | Compuestos biaril heterociclicos y metodos para preparar y utilizar los mismos |
EP1646629B1 (en) | 2003-07-02 | 2010-06-23 | Merck Sharp & Dohme Corp. | Cyclopropyl group substituted oxazolidinone antibiotics and derivatives thereof |
CA2529294A1 (en) * | 2003-07-02 | 2005-01-20 | Merck & Co., Inc. | Oxazolidinone antibiotics and derivatives thereof |
JP2007500707A (ja) * | 2003-07-29 | 2007-01-18 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | ビアリールヘテロ環状のアミン、アミドおよび硫黄−含有化合物、並びに該化合物の製造方法および使用方法 |
JP2007503426A (ja) * | 2003-08-25 | 2007-02-22 | ワーナー−ランバート カンパニー リミティド ライアビリティー カンパニー | 新規な抗微生物性アリールオキサゾリジノン化合物 |
US7687627B2 (en) * | 2003-09-08 | 2010-03-30 | Wockhardt Limited | Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy |
US7304050B2 (en) | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
WO2005042523A1 (en) * | 2003-11-03 | 2005-05-12 | Il-Dong Pharm. Co., Ltd. | A novel oxazolidinone derivative and manufacturing process thereof |
WO2005061468A1 (en) | 2003-12-17 | 2005-07-07 | Rib-X Pharmaceuticals, Inc. | Halogenated biaryl heterocyclic compounds and methods of making and using the same |
KR100854211B1 (ko) * | 2003-12-18 | 2008-08-26 | 동아제약주식회사 | 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물 |
EP1723159B1 (en) | 2004-02-27 | 2019-06-12 | Melinta Therapeutics, Inc. | Macrocyclic compounds and methods of making and using the same |
CA2566963A1 (en) * | 2004-05-25 | 2005-12-08 | Astrazeneca Ab | 3-[4-{6-substituted alkanoyl pyridin-3-yl}-3-phenyl]-5-(1h-1,2,3-triazol-1-ylmethyl)-1,3-oxazolidin-2-ones as antibacterial agents |
WO2005116023A1 (en) * | 2004-05-25 | 2005-12-08 | Astrazeneca Ab | 3- {4- (pyridin-3-yl) phenyl} -5- (1h-1, 2, 3-triazol-1-ylmethyl) -1, 3-oxazolidin-2-ones as antibacterial agents |
CN100360525C (zh) * | 2004-09-16 | 2008-01-09 | 中国科学院上海药物研究所 | 一类新的噁唑烷酮衍生物、其制备方法和用途 |
KR100629327B1 (ko) | 2004-10-20 | 2006-09-29 | 한국과학기술연구원 | 신규 트리아졸릴메틸옥사졸리디논 유도체 |
JP5534497B2 (ja) | 2005-06-08 | 2014-07-02 | メリンタ セラピューティクス,インコーポレイテッド | トリアゾール類の合成方法 |
JP5395432B2 (ja) | 2005-08-24 | 2014-01-22 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | トリアゾール化合物ならびにこれを作製する方法および使用する方法 |
EP1934237A2 (en) | 2005-08-24 | 2008-06-25 | Rib-X Pharmaceuticals, Inc. | Triazole compounds and methods of making and using the same |
EP2004640A1 (en) * | 2006-02-08 | 2008-12-24 | Pfizer Products Inc. | Oxazolidinones containing oxindoles as antibacterial agents |
CN100406455C (zh) * | 2006-02-20 | 2008-07-30 | 中国科学院上海药物研究所 | 含三氮唑基的噁唑烷酮类化合物及其制备方法和用途 |
TW200815428A (en) * | 2006-08-15 | 2008-04-01 | Wyeth Corp | Oxazolidone derivatives as PR modulators |
WO2008021338A2 (en) * | 2006-08-15 | 2008-02-21 | Wyeth | Tricyclic oxazolidone derivatives useful as pr modulators |
US8575337B2 (en) | 2008-06-24 | 2013-11-05 | Research Foundation Itsuu Laboratory | Oxazolidinone derivative having fused ring |
EP2757104B1 (en) * | 2008-10-10 | 2019-08-14 | Merck Sharp & Dohme Corp. | Compounds used in the synthesis of oxazolidinones |
ES2734724T3 (es) | 2009-02-03 | 2019-12-11 | Merck Sharp & Dohme | Forma cristalina de dihidrogenofosfato de (R)-3-(4-(2-(2-metiltetrazol-5-il)piridin-5-il)-3-fluorofenil)-5-hidroximetiloxazolidin-2-ona |
US8580767B2 (en) * | 2009-05-28 | 2013-11-12 | Trius Therapeutics, Inc. | Oxazolidinone containing dimer compounds, compositions and methods to make and use |
CN101792437B (zh) * | 2010-03-10 | 2012-01-25 | 天津药物研究院 | 一类三氮唑的衍生物、其制备方法和用途 |
US9464062B2 (en) | 2012-11-28 | 2016-10-11 | Temple University—Of the Commonwealth System of Higher Education | Disubstituted oxazolidin-2-ones 5-hydroxytryptamine receptor 2B activity modulators |
CA2986349A1 (en) * | 2015-07-22 | 2017-01-26 | Anavex Life Sciences Corp. | Crystal forms of tetrahydro-n,n-dimethyl-2,2-diphenyl-3-furanmethanamine hydrochloride, processes of making such forms, and their pharmaceutical compositions |
EP3914587A4 (en) * | 2019-01-18 | 2022-11-23 | Merck Sharp & Dohme LLC | OXAZOLIDINONE COMPOUNDS AND USES THEREOF AS ANTIBACTERIAL AGENTS |
WO2020234636A1 (en) * | 2019-05-17 | 2020-11-26 | Cadila Healthcare Limited | Novel compounds for the treatment of mammalian infections |
CN111560014A (zh) * | 2020-05-13 | 2020-08-21 | 河南科技大学第一附属医院 | 一种杀菌消毒所用噁唑链接三唑类药物分子及其制备方法和应用 |
Family Cites Families (93)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2338268A1 (fr) | 1976-01-16 | 1977-08-12 | Nativelle Spa | Nouveaux derives d'oxazolidinone, preparation et application a la synthese d'aryloxypropanolamines |
FR2356422A1 (fr) * | 1976-03-01 | 1978-01-27 | Delalande Sa | Nouveaux hydroxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application en therapeutique |
FR2458547B2 (fr) | 1978-06-09 | 1986-05-16 | Delalande Sa | Nouvelles n-aryle azolones, leur procede de preparation et leur application en therapeutique |
US4348393A (en) * | 1978-06-09 | 1982-09-07 | Delalande S.A. | N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones |
CH647772A5 (fr) * | 1979-05-07 | 1985-02-15 | Delalande Sa | Derives de la 5h-furanone-2 et de la 3h-dihydro-furanone-2, leurs procedes de preparation, et medicament les contenant. |
US4340606A (en) * | 1980-10-23 | 1982-07-20 | E. I. Du Pont De Nemours And Company | 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents |
FR2500450A1 (fr) * | 1981-02-25 | 1982-08-27 | Delalande Sa | Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique |
ES533097A0 (es) | 1983-06-07 | 1985-08-01 | Du Pont | Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno. |
US4705799A (en) * | 1983-06-07 | 1987-11-10 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents |
CA1260948A (en) | 1984-12-05 | 1989-09-26 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents |
US5272167A (en) * | 1986-12-10 | 1993-12-21 | Schering Corporation | Pharmaceutically active compounds |
US5750532A (en) * | 1986-12-10 | 1998-05-12 | Schering Corporation | Pharmaceutically active compounds |
US4851423A (en) * | 1986-12-10 | 1989-07-25 | Schering Corporation | Pharmaceutically active compounds |
US4942183A (en) * | 1987-10-16 | 1990-07-17 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents |
US4977173A (en) * | 1987-10-21 | 1990-12-11 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents |
US4948801A (en) * | 1988-07-29 | 1990-08-14 | E. I. Du Pont De Nemours And Company | Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents |
US5225565A (en) * | 1988-09-15 | 1993-07-06 | The Upjohn Company | Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones |
US5164510A (en) * | 1988-09-15 | 1992-11-17 | The Upjohn Company | 5'Indolinyl-5β-amidomethyloxazolidin-2-ones |
US5182403A (en) * | 1988-09-15 | 1993-01-26 | The Upjohn Company | Substituted 3(5'indazolyl) oxazolidin-2-ones |
DE68929303T2 (de) | 1988-09-15 | 2002-05-02 | Upjohn Co | 3-(Stickstoff substituierte)phenyl-5-beta-amidomethyloxazoliden-2-one |
US5231188A (en) * | 1989-11-17 | 1993-07-27 | The Upjohn Company | Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents |
JP3176626B2 (ja) | 1991-11-01 | 2001-06-18 | ファルマシア・アンド・アップジョン・カンパニー | 抗菌剤として有用な置換アリール−およびヘテロアリールフェニルオキサゾリジノン類 |
DE69329106T2 (de) * | 1992-04-30 | 2001-03-22 | Taiho Pharmaceutical Co Ltd | Oxazolidinderivat und sein pharmazeutisch verträgliches salz |
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
CA2136324A1 (en) | 1992-07-08 | 1994-01-20 | Steven Joseph Brickner | 5'-indolinyl oxazolidinones useful against mycobacterium tuberculosis |
HUT74099A (en) * | 1992-12-08 | 1996-11-28 | Upjohn Co | Tropone-substituted phenyloxazolidinone antibacterial agents and pharmaceutical compositions containing the same |
US5785976A (en) * | 1993-03-05 | 1998-07-28 | Pharmacia & Upjohn Ab | Solid lipid particles, particles of bioactive agents and methods for the manufacture and use thereof |
US5521202A (en) * | 1993-04-07 | 1996-05-28 | Taiho Pharmaceutical Co., Ltd. | Thiazolidine derivatives and pharmaceutical compositions containing the same |
DK0623615T3 (da) * | 1993-05-01 | 1999-12-13 | Merck Patent Gmbh | Adhæsionsreceptor-antagonister |
US5688792A (en) * | 1994-08-16 | 1997-11-18 | Pharmacia & Upjohn Company | Substituted oxazine and thiazine oxazolidinone antimicrobials |
DE4332384A1 (de) * | 1993-09-23 | 1995-03-30 | Merck Patent Gmbh | Adhäsionsrezeptor-Antagonisten III |
DE69419523T2 (de) * | 1993-11-22 | 1999-11-25 | Upjohn Co | Substituierte hydroxyacetyl piperazine phenyl oxazolidinonsäureester |
TW286317B (no) * | 1993-12-13 | 1996-09-21 | Hoffmann La Roche | |
US5668286A (en) * | 1994-03-15 | 1997-09-16 | Pharmacia & Upjohn Company | Oxazolidinone derivatives and pharmaceutical compositions containing them |
JPH07309850A (ja) | 1994-05-16 | 1995-11-28 | Canon Inc | 光学活性化合物、それを含有する液晶組成物、それを有する液晶素子及びそれらを用いた表示方法、表示装置 |
DE4425613A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
DE4425609A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | Benzofuranyl- und Benzothienyloxazolidinone |
DE4425612A1 (de) * | 1994-07-20 | 1996-04-04 | Bayer Ag | 6-gliedrige stickstoffhaltige Heteroaryl-oxazolidinone |
DE19514313A1 (de) * | 1994-08-03 | 1996-02-08 | Bayer Ag | Benzoxazolyl- und Benzothiazolyloxazolidinone |
ES2123889T3 (es) | 1994-11-02 | 1999-01-16 | Merck Patent Gmbh | Antagonistas de receptores de adhesion. |
CN1046520C (zh) * | 1994-11-15 | 1999-11-17 | 法玛西雅厄普约翰美国公司 | 二环噁嗪及噻嗪噁唑烷酮抗菌剂 |
NZ302844A (en) * | 1995-02-03 | 1999-06-29 | Upjohn Co | Antimicrobial hetero-aromatic ring substituted phenyloxazolidinones |
US6124334A (en) * | 1995-02-03 | 2000-09-26 | Pharmacia & Upjohn Company | Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials |
HRP960159A2 (en) * | 1995-04-21 | 1997-08-31 | Bayer Ag | Benzocyclopentane oxazolidinones containing heteroatoms |
DE19516483A1 (de) * | 1995-05-05 | 1996-11-07 | Merck Patent Gmbh | Adhäsionsrezeptor-Antagonisten |
CA2218088A1 (en) * | 1995-05-11 | 1996-11-14 | Pharmacia & Upjohn Company | Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
SK18898A3 (en) | 1995-08-14 | 1998-07-08 | Scripps Research Inst | Method compositions useful for inhibition of 'alpha'v'beta'5 mediated angiogenesis |
CN1072222C (zh) * | 1995-09-01 | 2001-10-03 | 法玛西雅厄普约翰公司 | 以c-c键连接于4-8元杂环环的苯基噁唑烷酮 |
MX9703040A (es) * | 1995-09-12 | 1997-07-31 | Upjohn Co | Antimicrobianos de feniloxazolidinona. |
DE69625238T2 (de) * | 1995-09-15 | 2003-07-24 | Upjohn Co | Alpha,beta-gesättigte und -ungesättigte 3-aryl-5-aminomethyl-butyrolactone antibakterielle mittel |
ES2214546T3 (es) | 1995-09-15 | 2004-09-16 | PHARMACIA & UPJOHN COMPANY | N-oxidos de aminoariloxazolidinona. |
GB9521508D0 (en) | 1995-10-20 | 1995-12-20 | Zeneca Ltd | Chemical compounds |
ZA968661B (en) * | 1995-11-17 | 1998-04-14 | Upjohn Co | Oxazolidinone antibacterial agent with tricyclic substituents. |
ZA969622B (en) * | 1995-12-13 | 1998-05-15 | Upjohn Co | Oxazolidinone antibacterial agents having a six-membered heteroaromatic ring. |
EP0874629B1 (en) | 1995-12-21 | 2004-05-19 | Bristol-Myers Squibb Pharma Company | ISOXAZOLINE, ISOTHIAZOLINE AND PYRAZOLINE FACTOR Xa INHIBITORS |
DE19601265A1 (de) * | 1996-01-16 | 1997-07-17 | Bayer Ag | 2-Oxo- und 2-Thio-1,2-dihydrochinolinyl-oxazolidinone |
DE19601264A1 (de) * | 1996-01-16 | 1997-07-17 | Bayer Ag | Pyrido-annellierte Thienyl- und Furanyl-Oxazolidinone |
DE19601627A1 (de) * | 1996-01-18 | 1997-07-24 | Bayer Ag | Heteroatomhaltige Cyclopentanopyridyl-Oxazolidinone |
GB9601666D0 (en) * | 1996-01-27 | 1996-03-27 | Zeneca Ltd | Chemical compounds |
DE19604223A1 (de) * | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
HRP970049A2 (en) * | 1996-02-06 | 1998-04-30 | Bayer Ag | New heteroaryl oxazolidinones |
GB9702213D0 (en) * | 1996-02-24 | 1997-03-26 | Zeneca Ltd | Chemical compounds |
MY116093A (en) * | 1996-02-26 | 2003-11-28 | Upjohn Co | Azolyl piperazinyl phenyl oxazolidinone antimicrobials |
GB9604301D0 (en) | 1996-02-29 | 1996-05-01 | Zeneca Ltd | Chemical compounds |
RU2176643C2 (ru) * | 1996-04-11 | 2001-12-10 | Фармация Энд Апджон Компани | Способ получения 5-гидроксиметил замещенных оксазолидинонов, способ получения 5-аминометил замещенных оксазолидиноновых аминов, оксазолидинонсульфонат |
GB9609919D0 (en) * | 1996-05-11 | 1996-07-17 | Zeneca Ltd | Chemical compounds |
GB9614236D0 (en) | 1996-07-06 | 1996-09-04 | Zeneca Ltd | Chemical compounds |
GB9614238D0 (en) | 1996-07-06 | 1996-09-04 | Zeneca Ltd | Chemical compounds |
AU3973697A (en) | 1996-08-21 | 1998-03-06 | Pharmacia & Upjohn Company | Isoxazoline derivatives useful as antimicrobials |
DE19707628A1 (de) * | 1997-02-26 | 1998-08-27 | Merck Patent Gmbh | Oxazolidinone |
KR100307211B1 (ko) * | 1997-05-24 | 2001-11-30 | 손 경 식 | 옥사졸리디논유도체,이의제조방법및그를함유한항균제조성물 |
EP0984947B8 (en) | 1997-05-30 | 2005-06-15 | Pharmacia & Upjohn Company LLC | Oxazolidinone antibacterial agents having a thiocarbonyl functionality |
GB9717804D0 (en) * | 1997-08-22 | 1997-10-29 | Zeneca Ltd | Chemical compounds |
JP2001514259A (ja) * | 1997-08-29 | 2001-09-11 | ゼネカ・リミテッド | アミノメチルオキソオキサゾリジニルベンゼン誘導体 |
US6140318A (en) * | 1997-10-23 | 2000-10-31 | Merck & Co., Inc. | Carbapenem antibacterial compounds, compositions containing such compounds and methods of treatment |
RU2205822C2 (ru) * | 1997-11-07 | 2003-06-10 | Фармация Энд Апджон Компани | Способы получения (s)-оксазолидинонов, (s)-вторичный спирт, соединение, способ получения спирта |
GB2332387A (en) * | 1997-12-16 | 1999-06-23 | Nestle Sa | Method and apparatus for moulding food articles |
JPH11322729A (ja) | 1998-03-09 | 1999-11-24 | Hokuriku Seiyaku Co Ltd | ジチオカルバミド酸誘導体 |
JP3334595B2 (ja) * | 1998-03-10 | 2002-10-15 | ダイソー株式会社 | オキサゾリジン−2−オン誘導体の製造法 |
CA2333332A1 (en) * | 1998-06-05 | 1999-12-16 | Astrazeneca Ab | Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them |
GB9812019D0 (en) * | 1998-06-05 | 1998-07-29 | Zeneca Ltd | Chemical compounds |
GB9821938D0 (en) * | 1998-10-09 | 1998-12-02 | Zeneca Ltd | Chemical compounds |
JP3973304B2 (ja) | 1998-10-29 | 2007-09-12 | 三井化学株式会社 | 2−オキサゾリドン誘導体の製造方法 |
JP2000204084A (ja) | 1998-11-11 | 2000-07-25 | Hokuriku Seiyaku Co Ltd | チオカルバミド酸誘導体 |
DE19901306A1 (de) | 1999-01-15 | 2000-07-20 | Bayer Ag | Neue Oxazolidinone |
DE19905278A1 (de) | 1999-02-09 | 2000-08-10 | Bayer Ag | Oxazolidinone und ihre Verwendung als antibakterielle Mittel |
DE19907701A1 (de) | 1999-02-23 | 2000-08-24 | Bayer Ag | Mit tricyclischen Indolen substituierte Oxazolidinone |
DE19909785A1 (de) | 1999-03-05 | 2000-09-07 | Bayer Ag | Neue, substituierte Isoxazoline |
DE10014961A1 (de) | 1999-07-08 | 2001-01-11 | Merck Patent Gmbh | Enantiomerentrennung von 3,5-disubstituierten 2-Oxazolidinonen |
DE10034625A1 (de) | 2000-07-17 | 2002-01-31 | Bayer Ag | Heterocyclisch substituierte Thienyl-Phenyl-Oxazolidinone |
DE10034624A1 (de) | 2000-07-17 | 2002-01-31 | Bayer Ag | Aryl-substituierte Thienyl-1,3-oxazolidin-2-one als Cytokin-Inhibitoren |
HUP0302918A2 (hu) * | 2000-07-17 | 2003-12-29 | Ranbaxy Laboratories Limited | Mikrobaellenes oxazolidinonszármazékok és a vegyületeket tartalmazó gyógyászati készítmények és eljárás a vegyületek előállítására |
US6410728B1 (en) * | 2000-08-31 | 2002-06-25 | Abbott Laboratories | Oxazolidinone chemotherapeutic agents |
-
2000
- 2000-04-25 GB GBGB0009803.8A patent/GB0009803D0/en not_active Ceased
-
2001
- 2001-04-23 SI SI200130129T patent/SI1286998T2/sl unknown
- 2001-04-23 CZ CZ20023527A patent/CZ20023527A3/cs unknown
- 2001-04-23 MX MXPA02010453A patent/MXPA02010453A/es active IP Right Grant
- 2001-04-23 AU AU48636/01A patent/AU781784B2/en not_active Ceased
- 2001-04-23 PL PL01358326A patent/PL358326A1/xx not_active Application Discontinuation
- 2001-04-23 DE DE60103754T patent/DE60103754T3/de not_active Expired - Lifetime
- 2001-04-23 EE EEP200200598A patent/EE200200598A/xx unknown
- 2001-04-23 US US10/258,355 patent/US7141583B2/en not_active Expired - Fee Related
- 2001-04-23 JP JP2001578439A patent/JP2003531211A/ja active Pending
- 2001-04-23 IL IL15228401A patent/IL152284A0/xx unknown
- 2001-04-23 TR TR2004/02261T patent/TR200402261T4/xx unknown
- 2001-04-23 CN CNB01811640XA patent/CN1277829C/zh not_active Expired - Fee Related
- 2001-04-23 EP EP01921669A patent/EP1286998B2/en not_active Expired - Lifetime
- 2001-04-23 NZ NZ521765A patent/NZ521765A/en not_active IP Right Cessation
- 2001-04-23 HU HU0300416A patent/HUP0300416A2/hu unknown
- 2001-04-23 PT PT01921669T patent/PT1286998E/pt unknown
- 2001-04-23 AT AT01921669T patent/ATE268778T1/de active
- 2001-04-23 DK DK01921669T patent/DK1286998T4/da active
- 2001-04-23 CA CA2405349A patent/CA2405349C/en not_active Expired - Lifetime
- 2001-04-23 RU RU2002131455/04A patent/RU2002131455A/ru not_active Application Discontinuation
- 2001-04-23 BR BR0110240-0A patent/BR0110240A/pt not_active Application Discontinuation
- 2001-04-23 KR KR1020027014321A patent/KR100858771B1/ko not_active IP Right Cessation
- 2001-04-23 WO PCT/GB2001/001815 patent/WO2001081350A1/en active IP Right Grant
- 2001-04-23 ES ES01921669T patent/ES2220759T5/es not_active Expired - Lifetime
-
2002
- 2002-10-10 ZA ZA200208187A patent/ZA200208187B/en unknown
- 2002-10-14 IL IL152284A patent/IL152284A/en not_active IP Right Cessation
- 2002-10-16 IS IS6583A patent/IS6583A/is unknown
- 2002-10-23 NO NO20025091A patent/NO328549B1/no not_active IP Right Cessation
-
2003
- 2003-07-25 HK HK03105394A patent/HK1053114A1/xx not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
DK1286998T4 (da) | Oxazolidinonderivater med antibiotisk aktivitet | |
BG105001A (en) | Oxazolidinone derivatives, process for their preparartion and pharmaceutical compositions containing them | |
AU1714801A (en) | Substituted isoxazolines and their use as antibacterial agents | |
ATE258552T1 (de) | Oxazolidinon-derivate als antibiotika, verfahren zu ihrer herstellung und diese derivate enthaltende pharmazeutische zusammensetzungen | |
PL373888A1 (en) | 3-heteroaryl substituted 5-methyloxymethyl isoxazolines used as herbicides | |
HUP0302918A2 (hu) | Mikrobaellenes oxazolidinonszármazékok és a vegyületeket tartalmazó gyógyászati készítmények és eljárás a vegyületek előállítására | |
HUP0300350A2 (hu) | Új 3-amino-azetidin-származékok, előállításuk és ezeket tartalmazó gyógyszerkészítmények | |
NO20062269L (no) | Pyridin-karboksylsyrederivater som glucokinasemodulatorer | |
AU2001235838A1 (en) | Imidazol derivatives as raf kinase inhibitors | |
ATE332299T1 (de) | Eine sulfonimid-gruppe enthaltende oxazolidinone als antibiotika | |
AU2003267791A1 (en) | Triazole compounds for the treatment of dysmenorrhoea | |
SE0201937D0 (sv) | Therapeutic agents | |
NO922028L (no) | Azol-derivater | |
AU8824391A (en) | New guanidine compounds, process for preparing these and pharmaceutical compositions containing them | |
WO2003072576A3 (en) | Oxazolidinone derivatives, processes for their preparation, and pharmaceutical compositions containing them | |
AU8454998A (en) | (hetero)aryl-sulfonamide derivatives, their preparation and their use as factor xa inhibitors | |
KR930006024A (ko) | 이미다조 인돌리진 유도체 및 그의 제조방법 | |
KR920009834A (ko) | 7-아실-3-(치환 카르바모일옥시)세펨 화합물 및 그의 제조 방법 | |
NO20053302D0 (no) | Imidazolderivater med affinitet for alfa 2-reseptoraktivitet. | |
TW360655B (en) | Heterocyclyl-ergoline derivatives | |
HUP9901211A2 (hu) | Benzopiránszármazékok alkalmazása implantátum kilökődést magakadályozó gyógyszerkészítmények előállítására | |
HUP0002715A2 (hu) | Benzotiofénszármazékok alkalmazása trombocitaszám csökkentésére szolgáló gyógyszerkészítmények előállítására | |
CA2238723A1 (en) | Arylethenesulfonamide derivatives and drug composition containing the same | |
JO1684B1 (en) | Azole derivatives | |
TH13393A (th) | อนุพันธ์ของอินโดล |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM1K | Lapsed by not paying the annual fees |