ATE258552T1 - Oxazolidinon-derivate als antibiotika, verfahren zu ihrer herstellung und diese derivate enthaltende pharmazeutische zusammensetzungen - Google Patents
Oxazolidinon-derivate als antibiotika, verfahren zu ihrer herstellung und diese derivate enthaltende pharmazeutische zusammensetzungenInfo
- Publication number
- ATE258552T1 ATE258552T1 AT99925181T AT99925181T ATE258552T1 AT E258552 T1 ATE258552 T1 AT E258552T1 AT 99925181 T AT99925181 T AT 99925181T AT 99925181 T AT99925181 T AT 99925181T AT E258552 T1 ATE258552 T1 AT E258552T1
- Authority
- AT
- Austria
- Prior art keywords
- derivatives
- antibiotics
- production
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9812019.9A GB9812019D0 (en) | 1998-06-05 | 1998-06-05 | Chemical compounds |
PCT/GB1999/001737 WO1999064416A2 (en) | 1998-06-05 | 1999-06-03 | Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them |
Publications (1)
Publication Number | Publication Date |
---|---|
ATE258552T1 true ATE258552T1 (de) | 2004-02-15 |
Family
ID=10833201
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AT99925181T ATE258552T1 (de) | 1998-06-05 | 1999-06-03 | Oxazolidinon-derivate als antibiotika, verfahren zu ihrer herstellung und diese derivate enthaltende pharmazeutische zusammensetzungen |
Country Status (16)
Country | Link |
---|---|
EP (2) | EP1082322B1 (de) |
JP (1) | JP2002517497A (de) |
KR (1) | KR20010052590A (de) |
CN (1) | CN1304410A (de) |
AT (1) | ATE258552T1 (de) |
AU (1) | AU753865B2 (de) |
BR (1) | BR9910915A (de) |
CA (1) | CA2332831A1 (de) |
DE (1) | DE69914478T2 (de) |
GB (1) | GB9812019D0 (de) |
HU (1) | HUP0103404A3 (de) |
IL (1) | IL140085A0 (de) |
NO (1) | NO20006149L (de) |
NZ (1) | NZ507973A (de) |
WO (1) | WO1999064416A2 (de) |
ZA (1) | ZA200006697B (de) |
Families Citing this family (35)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6608081B2 (en) | 1999-08-12 | 2003-08-19 | Ortho-Mcneil Pharmaceutical, Inc. | Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods |
PE20010851A1 (es) * | 1999-12-14 | 2001-08-17 | Upjohn Co | Esteres del acido benzoico de oxazolidinonas que tienen un substituyente hidroxiacetilpiperazina |
GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
PE20030044A1 (es) | 2000-11-17 | 2003-02-09 | Upjohn Co | Isoxazolinonas biciclicas de formula i |
PE20020689A1 (es) * | 2000-11-17 | 2002-08-03 | Upjohn Co | Oxazolidinonas con un heterociclo de 6 o 7 miembros unidos con enlace anular al benceno |
JP2004518724A (ja) * | 2001-02-07 | 2004-06-24 | オーソーマクニール ファーマシューティカル, インコーポレイテッド | ピリドアリールフェニル・オキサゾリジノン抗菌剤、および関連の組成物および方法 |
RU2004111285A (ru) | 2001-09-11 | 2005-10-10 | Астразенека Аб (Se) | Оксазолидинон и/или изоксазолин в качестве антибактериальных средств |
JP2005512975A (ja) | 2001-10-25 | 2005-05-12 | アストラゼネカ アクチボラグ | 抗菌薬として有用なイソキサゾリン誘導体 |
WO2003035648A1 (en) * | 2001-10-25 | 2003-05-01 | Astrazeneca Ab | Aryl substituted oxazolidinones with antibacterial activity |
BR0308018A (pt) | 2002-02-28 | 2005-01-04 | Astrazeneca Ab | Composto ou um seu sal farmaceuticamente aceitável ou um seu éster hidrolisável in vivo, pró-droga, método para produzir um efeito antibacteriano em um animal de sangue quente, uso de um composto ou um seu sal farmaceuticamente aceitável ou um seu éster hirolisável in vivo, composição farmacêutica, e, processo para a preparação de um composto ou um seu sal farmaceuticamente aceitável ou um seu éster hidrolisável in vivo |
MXPA04008312A (es) | 2002-02-28 | 2004-11-26 | Astrazeneca Ab | Derivados de 3-cilil-5-(anillo de 5 miembros que contienen nitrogeno)-metil-oxazolidinona y sus uso como agentes antibacterianos. |
AR043050A1 (es) | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
US7012088B2 (en) * | 2003-02-24 | 2006-03-14 | Pharmacia & Upjohn Company | Indolone oxazolidinones and derivatives thereof |
GB0306358D0 (en) | 2003-03-20 | 2003-04-23 | Astrazeneca Ab | Chemical compounds |
US8324398B2 (en) | 2003-06-03 | 2012-12-04 | Rib-X Pharmaceuticals, Inc. | Process for the synthesis of biaryl oxazolidinones |
MXPA05013132A (es) | 2003-06-03 | 2006-05-25 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos de biarilo y metodos de produccion y su uso. |
JP2007514782A (ja) | 2003-12-17 | 2007-06-07 | リブ−エックス ファーマシューティカルズ,インコーポレイテッド | ハロゲン化ビアリール複素環式化合物ならびにその作製方法および使用方法 |
CN102816194A (zh) | 2004-02-27 | 2012-12-12 | 瑞伯-X医药品有限公司 | 大环化合物以及其制作和使用方法 |
CN101001853A (zh) * | 2004-08-06 | 2007-07-18 | 法玛西雅厄普约翰有限责任公司 | 作为抗细菌剂的含羟吲哚的唑烷酮类 |
MX2007003319A (es) | 2004-09-20 | 2007-06-05 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como agentes terapeuticos. |
WO2006034279A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as therapeutic agents |
CN101083994A (zh) | 2004-09-20 | 2007-12-05 | 泽农医药公司 | 杂环衍生物及其用作硬脂酰CoA去饱和酶抑制剂的用途 |
CA2580856A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors |
AR051026A1 (es) | 2004-09-20 | 2006-12-13 | Xenon Pharmaceuticals Inc | Derivados heterociclicos y su uso como inhibidores de la estearoil-coa desaturasa |
CA2580844A1 (en) | 2004-09-20 | 2006-03-30 | Xenon Pharmaceuticals Inc. | Heterocyclic derivatives and their use as mediators of stearoyl-coa desaturase |
CN101083993A (zh) | 2004-09-20 | 2007-12-05 | 泽农医药公司 | 杂环衍生物及其作为硬脂酰CoA去饱和酶抑制剂的用途 |
WO2006043121A1 (en) * | 2004-10-20 | 2006-04-27 | Ranbaxy Laboratories Limited | Oxazolidinone derivatives as antimicrobials |
AU2006343359A1 (en) | 2005-06-03 | 2007-11-15 | Xenon Pharmaceuticals Inc. | Aminothiazole derivatives as human stearoyl-coa desaturase inhibitors |
KR101394307B1 (ko) | 2005-06-08 | 2014-05-13 | 멜린타 테라퓨틱스, 인크. | 트리아졸의 합성 방법 |
WO2008021309A1 (en) | 2006-08-15 | 2008-02-21 | Wyeth | Imidazolidin-2-one derivatives useful as pr modulators |
WO2008021338A2 (en) | 2006-08-15 | 2008-02-21 | Wyeth | Tricyclic oxazolidone derivatives useful as pr modulators |
US7538107B2 (en) | 2006-08-15 | 2009-05-26 | Wyeth | Oxazinan-2-one derivatives useful as PR modulators |
US7649007B2 (en) | 2006-08-15 | 2010-01-19 | Wyeth Llc | Oxazolidine derivatives as PR modulators |
CN101798302B (zh) | 2009-02-06 | 2014-11-05 | 上海盟科药业有限公司 | 抗生素类药物1-(邻-氟苯基)二氢吡啶酮的合成及生产的方法和工艺 |
WO2013182070A1 (zh) * | 2012-06-08 | 2013-12-12 | 四川贝力克生物技术有限责任公司 | 一种用于预防或治疗分支杆菌疾病的药物 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0605729B1 (de) * | 1992-04-30 | 2000-07-26 | Taiho Pharmaceutical Co., Ltd. | Oxazolidinderivat und sein pharmazeutisch verträgliches salz |
SK283420B6 (sk) * | 1992-05-08 | 2003-07-01 | Pharmacia & Upjohn Company | Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny |
US5521202A (en) * | 1993-04-07 | 1996-05-28 | Taiho Pharmaceutical Co., Ltd. | Thiazolidine derivatives and pharmaceutical compositions containing the same |
DE4332384A1 (de) * | 1993-09-23 | 1995-03-30 | Merck Patent Gmbh | Adhäsionsrezeptor-Antagonisten III |
EP0710657B1 (de) * | 1994-11-02 | 1998-08-26 | MERCK PATENT GmbH | Adhäsionsrezeptor-Antagonisten |
CZ40998A3 (cs) * | 1995-08-14 | 1998-09-16 | The Scripps Research Institute | Použití antagonisty anb5 pro výrobu prostředků, schopných inhibovat angiogenezi v tkáních |
US5968962A (en) * | 1995-09-01 | 1999-10-19 | Pharmacia & Upjohn Company | Phenyloxazolidinones having a C-C bond to 4-8 membered heterocyclic rings |
-
1998
- 1998-06-05 GB GBGB9812019.9A patent/GB9812019D0/en not_active Ceased
-
1999
- 1999-06-03 CA CA002332831A patent/CA2332831A1/en not_active Abandoned
- 1999-06-03 JP JP2000553425A patent/JP2002517497A/ja active Pending
- 1999-06-03 IL IL14008599A patent/IL140085A0/xx unknown
- 1999-06-03 NZ NZ507973A patent/NZ507973A/en unknown
- 1999-06-03 CN CN99806910A patent/CN1304410A/zh active Pending
- 1999-06-03 BR BR9910915-8A patent/BR9910915A/pt not_active IP Right Cessation
- 1999-06-03 EP EP99925181A patent/EP1082322B1/de not_active Expired - Lifetime
- 1999-06-03 AT AT99925181T patent/ATE258552T1/de not_active IP Right Cessation
- 1999-06-03 KR KR1020007013774A patent/KR20010052590A/ko not_active Application Discontinuation
- 1999-06-03 EP EP03012958A patent/EP1357122A3/de not_active Withdrawn
- 1999-06-03 DE DE69914478T patent/DE69914478T2/de not_active Expired - Fee Related
- 1999-06-03 HU HU0103404A patent/HUP0103404A3/hu unknown
- 1999-06-03 AU AU41565/99A patent/AU753865B2/en not_active Ceased
- 1999-06-03 WO PCT/GB1999/001737 patent/WO1999064416A2/en not_active Application Discontinuation
-
2000
- 2000-11-18 ZA ZA200006697A patent/ZA200006697B/en unknown
- 2000-12-04 NO NO20006149A patent/NO20006149L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
DE69914478T2 (de) | 2004-11-11 |
HUP0103404A3 (en) | 2002-08-28 |
NO20006149D0 (no) | 2000-12-04 |
EP1082322B1 (de) | 2004-01-28 |
BR9910915A (pt) | 2001-03-06 |
CA2332831A1 (en) | 1999-12-16 |
WO1999064416A2 (en) | 1999-12-16 |
EP1082322A2 (de) | 2001-03-14 |
AU753865B2 (en) | 2002-10-31 |
JP2002517497A (ja) | 2002-06-18 |
IL140085A0 (en) | 2002-02-10 |
ZA200006697B (en) | 2002-02-18 |
CN1304410A (zh) | 2001-07-18 |
EP1357122A2 (de) | 2003-10-29 |
NZ507973A (en) | 2003-10-31 |
NO20006149L (no) | 2001-02-02 |
WO1999064416A3 (en) | 2000-01-27 |
AU4156599A (en) | 1999-12-30 |
DE69914478D1 (de) | 2004-03-04 |
GB9812019D0 (en) | 1998-07-29 |
HUP0103404A2 (hu) | 2002-05-29 |
KR20010052590A (ko) | 2001-06-25 |
EP1357122A3 (de) | 2003-12-10 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |