MD3570834T2 - Inhibitori biciclici ai histon deacetilazei - Google Patents
Inhibitori biciclici ai histon deacetilazeiInfo
- Publication number
- MD3570834T2 MD3570834T2 MDE20191311T MDE20191311T MD3570834T2 MD 3570834 T2 MD3570834 T2 MD 3570834T2 MD E20191311 T MDE20191311 T MD E20191311T MD E20191311 T MDE20191311 T MD E20191311T MD 3570834 T2 MD3570834 T2 MD 3570834T2
- Authority
- MD
- Moldova
- Prior art keywords
- disease
- disorder
- compound
- pharmaceutically acceptable
- compounds
- Prior art date
Links
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-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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| US201762445022P | 2017-01-11 | 2017-01-11 | |
| US201762555298P | 2017-09-07 | 2017-09-07 | |
| PCT/US2018/013260 WO2018132531A1 (en) | 2017-01-11 | 2018-01-11 | Bicyclic inhibitors of histone deacetylase |
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| RS62639B1 (sr) | 2015-07-06 | 2021-12-31 | Alkermes Inc | Hetero-halo inhibitori histonskih deacetilaza |
| EP3319968A1 (en) | 2015-07-06 | 2018-05-16 | Rodin Therapeutics, Inc. | Heterobicyclic n-aminophenyl-amides as inhibitors of histone deacetylase |
| JP6756925B2 (ja) | 2017-01-11 | 2020-09-16 | ロダン・セラピューティクス，インコーポレーテッド | ヒストンデアセチラーゼの二環式阻害剤 |
| ES2914355T3 (es) | 2017-08-07 | 2022-06-09 | Alkermes Inc | Inhibidores bicíclicos de la histona desacetilasa |
| MA56213A (fr) * | 2019-06-13 | 2022-04-20 | Dana Farber Cancer Inst Inc | Développement d'inhibiteurs catalytiques de hdac3 et leurs utilisations |
| EP4003958A1 (en) | 2019-07-23 | 2022-06-01 | Alkermes, Inc. | Synthesis of bicyclic inhibitors of histone deacetylase |
| CN110734924B (zh) * | 2019-10-25 | 2020-10-23 | 山东大学第二医院 | 一种抑郁症检测、治疗和预后靶点及应用 |
| MX2024006684A (es) | 2021-12-03 | 2024-08-26 | Tango Therapeutics Inc | Inhibidores de hdac novedosos y uso terapéutico de estos. |
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