LU82120A1 - Procede de preparation de composes b-lactame - Google Patents

Procede de preparation de composes b-lactame Download PDF

Info

Publication number
LU82120A1
LU82120A1 LU82120A LU82120A LU82120A1 LU 82120 A1 LU82120 A1 LU 82120A1 LU 82120 A LU82120 A LU 82120A LU 82120 A LU82120 A LU 82120A LU 82120 A1 LU82120 A1 LU 82120A1
Authority
LU
Luxembourg
Prior art keywords
group
formula
protected
alkyl
chlorine
Prior art date
Application number
LU82120A
Other languages
English (en)
French (fr)
Inventor
J Fisher
L Hatfield
L Blaszczak
C Bunnell
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27358615&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=LU82120(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US06/008,647 external-priority patent/US4226986A/en
Priority claimed from US06/008,470 external-priority patent/US4211702A/en
Priority claimed from US06/008,645 external-priority patent/US4223133A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of LU82120A1 publication Critical patent/LU82120A1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04—Preparation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/02—Preparation
    • C07D501/04—Preparation from compounds already containing the ring or condensed ring systems, e.g. by dehydrogenation of the ring, by introduction, elimination or modification of substituents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D505/00—Heterocyclic compounds containing 5-oxa-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. oxacephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
LU82120A 1979-02-01 1980-01-31 Procede de preparation de composes b-lactame LU82120A1 (fr)

Applications Claiming Priority (6)

Application Number Priority Date Filing Date Title
US06/008,647 US4226986A (en) 1979-02-01 1979-02-01 Process for halogenation of β-lactam compounds
US06/008,470 US4211702A (en) 1979-02-01 1979-02-01 Process for preparation of penicillin and cephalosporin imino halides
US864579 1979-02-01
US847079 1979-02-01
US06/008,645 US4223133A (en) 1979-02-01 1979-02-01 Cephalosporin reduction process
US864779 1979-02-01

Publications (1)

Publication Number Publication Date
LU82120A1 true LU82120A1 (fr) 1980-04-23

Family

ID=27358615

Family Applications (1)

Application Number Title Priority Date Filing Date
LU82120A LU82120A1 (fr) 1979-02-01 1980-01-31 Procede de preparation de composes b-lactame

Country Status (32)

Country Link
EP (1) EP0014567B1 (ru)
JP (12) JPS55113789A (ru)
KR (1) KR830001901B1 (ru)
AT (1) AT372684B (ru)
AU (1) AU538175B2 (ru)
BE (1) BE881425A (ru)
BG (1) BG35899A3 (ru)
CA (1) CA1133468A (ru)
CH (3) CH652405A5 (ru)
DD (1) DD153374A5 (ru)
DE (1) DE3066119D1 (ru)
DK (2) DK163513C (ru)
ES (1) ES488231A0 (ru)
FI (1) FI74968C (ru)
FR (1) FR2447924A1 (ru)
GB (1) GB2044256B (ru)
GR (1) GR72278B (ru)
IE (1) IE49377B1 (ru)
IL (1) IL59269A (ru)
IT (1) IT1193908B (ru)
LU (1) LU82120A1 (ru)
MA (1) MA18715A1 (ru)
MW (1) MW880A1 (ru)
MY (1) MY8500598A (ru)
NL (1) NL191791C (ru)
NO (1) NO160660C (ru)
NZ (1) NZ192749A (ru)
OA (1) OA06451A (ru)
PH (1) PH15158A (ru)
PL (4) PL129604B1 (ru)
PT (1) PT70744A (ru)
YU (4) YU22580A (ru)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0348124B1 (en) * 1988-06-22 1994-04-27 Eli Lilly And Company Intermediate for 1-carba(dethia)cephalosporin
EP1961636B1 (en) 2007-02-20 2013-04-24 Yamaha Hatsudoki Kabushiki Kaisha Hydraulic master cylinder and vehicle provided with the same
JP5319035B1 (ja) 2012-03-09 2013-10-16 真一郎 谷 トレーニングラダー
US9741942B2 (en) 2012-10-11 2017-08-22 Merck Patent Gmbh Materials for organic electroluminescent devices
JP6202969B2 (ja) * 2013-10-01 2017-09-27 富士電機株式会社 情報処理装置、暗号化方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK118506B (da) * 1963-02-18 1970-08-31 Ciba Geigy Fremgangsmåde til fremstilling af 7-aminocephalosporansyre eller estere deraf.
US3641014A (en) * 1968-10-03 1972-02-08 Lilly Co Eli Reduction of delta**3-cephalosporin sulfoxides
US3925372A (en) * 1973-02-23 1975-12-09 Lilly Co Eli Alpha-aminoacyl-3-halo cephalosporins

Also Published As

Publication number Publication date
IT1193908B (it) 1988-08-31
DK41480A (da) 1980-08-02
JPH0372633B2 (ru) 1991-11-19
IL59269A0 (en) 1980-05-30
DK179991A (da) 1991-10-30
IT8019609A0 (it) 1980-01-31
MY8500598A (en) 1985-12-31
JPH0372631B2 (ru) 1991-11-19
GR72278B (ru) 1983-10-11
EP0014567A1 (en) 1980-08-20
DE3066119D1 (en) 1984-02-23
FR2447924B1 (ru) 1983-10-21
PL128595B1 (en) 1984-02-29
MA18715A1 (fr) 1980-10-01
PH15158A (en) 1982-08-24
YU22580A (en) 1983-06-30
JPH0649706B2 (ja) 1994-06-29
EP0014567B1 (en) 1984-01-18
JPH0371435B2 (ru) 1991-11-13
JPH0649705B2 (ja) 1994-06-29
ES8101603A1 (es) 1980-12-16
IE800190L (en) 1980-08-01
JPH0372634B2 (ru) 1991-11-19
PL126947B1 (en) 1983-09-30
JPH04356490A (ja) 1992-12-10
IE49377B1 (en) 1985-10-02
YU16483A (en) 1984-02-29
MW880A1 (en) 1981-09-09
BG35899A3 (en) 1984-07-16
AT372684B (de) 1983-11-10
PL129604B1 (en) 1984-05-31
JPH0334982A (ja) 1991-02-14
JPH0565513B2 (ru) 1993-09-17
FR2447924A1 (fr) 1980-08-29
CH652405A5 (fr) 1985-11-15
CH656385A5 (fr) 1986-06-30
NL191791C (nl) 1996-08-02
DK163513B (da) 1992-03-09
YU18283A (en) 1984-02-29
JPH07121950B2 (ja) 1995-12-25
YU16383A (en) 1984-02-29
JPS55113789A (en) 1980-09-02
JPH04364187A (ja) 1992-12-16
ATA50280A (de) 1983-03-15
DK179991D0 (da) 1991-10-30
AU538175B2 (en) 1984-08-02
NO160660C (no) 1989-05-16
PT70744A (en) 1980-02-01
JPH0517483A (ja) 1993-01-26
JPH089629B2 (ja) 1996-01-31
GB2044256B (en) 1983-05-05
YU44734B (en) 1991-02-28
BE881425A (fr) 1980-07-30
JPH0334981A (ja) 1991-02-14
DD153374A5 (de) 1982-01-06
ES488231A0 (es) 1980-12-16
JPH0565514B2 (ru) 1993-09-17
JPH0334984A (ja) 1991-02-14
OA06451A (fr) 1981-07-31
JPH0372632B2 (ru) 1991-11-19
NL8000545A (nl) 1980-08-05
IL59269A (en) 1984-04-30
JPH0532669A (ja) 1993-02-09
NO160660B (no) 1989-02-06
JPH0334985A (ja) 1991-02-14
GB2044256A (en) 1980-10-15
DK163667B (da) 1992-03-23
NO800251L (no) 1980-08-04
KR830001943A (ko) 1983-05-19
FI74968C (fi) 1988-04-11
JPH054991A (ja) 1993-01-14
FI800303A (fi) 1980-08-02
DK163667C (da) 1992-08-17
PL221744A1 (ru) 1980-12-01
DK163513C (da) 1992-07-27
NZ192749A (en) 1983-06-17
JPH054990A (ja) 1993-01-14
CH648318A5 (fr) 1985-03-15
NL191791B (nl) 1996-04-01
FI74968B (fi) 1987-12-31
AU5502980A (en) 1980-08-07
JPH0334983A (ja) 1991-02-14
JPH0372231B2 (ru) 1991-11-18
CA1133468A (en) 1982-10-12
PL129399B1 (en) 1984-05-31
KR830001901B1 (ko) 1983-09-19

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