KR20220025926A - 당뇨병 요법 - Google Patents

당뇨병 요법 Download PDF

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Publication number
KR20220025926A
KR20220025926A KR1020227004998A KR20227004998A KR20220025926A KR 20220025926 A KR20220025926 A KR 20220025926A KR 1020227004998 A KR1020227004998 A KR 1020227004998A KR 20227004998 A KR20227004998 A KR 20227004998A KR 20220025926 A KR20220025926 A KR 20220025926A
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KR
South Korea
Prior art keywords
insulin
dpp
inhibitor
diabetes
combination
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020227004998A
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English (en)
Korean (ko)
Inventor
토마스 클라인
미하엘 마르크
레오 토마스
Original Assignee
베링거 인겔하임 인터내셔날 게엠베하
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Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44509854&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20220025926(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 베링거 인겔하임 인터내셔날 게엠베하 filed Critical 베링거 인겔하임 인터내셔날 게엠베하
Priority to KR1020237011271A priority Critical patent/KR20230051307A/ko
Publication of KR20220025926A publication Critical patent/KR20220025926A/ko
Ceased legal-status Critical Current

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/28—Insulins
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    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
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    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Ophthalmology & Optometry (AREA)
  • Urology & Nephrology (AREA)
  • Rheumatology (AREA)
  • Reproductive Health (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Vascular Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Dermatology (AREA)
  • Gynecology & Obstetrics (AREA)
KR1020227004998A 2010-06-24 2011-06-22 당뇨병 요법 Ceased KR20220025926A (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1020237011271A KR20230051307A (ko) 2010-06-24 2011-06-22 당뇨병 요법

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP10167243.4 2010-06-24
EP10167243 2010-06-24
KR1020207006530A KR20200028498A (ko) 2010-06-24 2011-06-22 당뇨병 요법
PCT/EP2011/060449 WO2011161161A1 (en) 2010-06-24 2011-06-22 Diabetes therapy

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020207006530A Division KR20200028498A (ko) 2010-06-24 2011-06-22 당뇨병 요법

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020237011271A Division KR20230051307A (ko) 2010-06-24 2011-06-22 당뇨병 요법

Publications (1)

Publication Number Publication Date
KR20220025926A true KR20220025926A (ko) 2022-03-03

Family

ID=44509854

Family Applications (6)

Application Number Title Priority Date Filing Date
KR1020227004998A Ceased KR20220025926A (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR20127033437A Ceased KR20130093012A (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020197012928A Ceased KR20190050871A (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020187017848A Active KR102018038B1 (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020237011271A Ceased KR20230051307A (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020207006530A Ceased KR20200028498A (ko) 2010-06-24 2011-06-22 당뇨병 요법

Family Applications After (5)

Application Number Title Priority Date Filing Date
KR20127033437A Ceased KR20130093012A (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020197012928A Ceased KR20190050871A (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020187017848A Active KR102018038B1 (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020237011271A Ceased KR20230051307A (ko) 2010-06-24 2011-06-22 당뇨병 요법
KR1020207006530A Ceased KR20200028498A (ko) 2010-06-24 2011-06-22 당뇨병 요법

Country Status (18)

Country Link
US (1) US9149478B2 (enExample)
EP (4) EP3124041A1 (enExample)
JP (3) JP5843855B2 (enExample)
KR (6) KR20220025926A (enExample)
CN (2) CN106975074A (enExample)
AR (1) AR082767A1 (enExample)
AU (1) AU2011268940B2 (enExample)
BR (1) BR112012032579B1 (enExample)
CA (2) CA2803504C (enExample)
CL (1) CL2012003393A1 (enExample)
EA (2) EA201201657A1 (enExample)
ES (2) ES2953123T3 (enExample)
IL (1) IL222778A0 (enExample)
MX (1) MX2012014247A (enExample)
NZ (1) NZ603319A (enExample)
PH (1) PH12012502524A1 (enExample)
TW (1) TWI618537B (enExample)
WO (1) WO2011161161A1 (enExample)

Families Citing this family (49)

* Cited by examiner, † Cited by third party
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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7501426B2 (en) 2004-02-18 2009-03-10 Boehringer Ingelheim International Gmbh 8-[3-amino-piperidin-1-yl]-xanthines, their preparation and their use as pharmaceutical compositions
DE102004054054A1 (de) 2004-11-05 2006-05-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Verfahren zur Herstellung chiraler 8-(3-Amino-piperidin-1-yl)-xanthine
DE102005035891A1 (de) 2005-07-30 2007-02-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-(3-Amino-piperidin-1-yl)-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
EP1852108A1 (en) 2006-05-04 2007-11-07 Boehringer Ingelheim Pharma GmbH & Co.KG DPP IV inhibitor formulations
MX2008014024A (es) 2006-05-04 2008-11-14 Boehringer Ingelheim Int Formas poliformas.
PE20080251A1 (es) 2006-05-04 2008-04-25 Boehringer Ingelheim Int Usos de inhibidores de dpp iv
PE20090938A1 (es) 2007-08-16 2009-08-08 Boehringer Ingelheim Int Composicion farmaceutica que comprende un derivado de benceno sustituido con glucopiranosilo
US10058593B2 (en) 2008-03-26 2018-08-28 Oramed Ltd. Methods and compositions for oral administration of proteins
PE20091730A1 (es) 2008-04-03 2009-12-10 Boehringer Ingelheim Int Formulaciones que comprenden un inhibidor de dpp4
UY32030A (es) 2008-08-06 2010-03-26 Boehringer Ingelheim Int "tratamiento para diabetes en pacientes inapropiados para terapia con metformina"
BRPI0916997A2 (pt) 2008-08-06 2020-12-15 Boehringer Ingelheim International Gmbh Inibidor de dpp-4 e seu uso
MX2011002558A (es) 2008-09-10 2011-04-26 Boehringer Ingelheim Int Terapia de combinacion para el tratamiento de diabetes y estados relacionados.
US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
EP2382216A1 (en) 2008-12-23 2011-11-02 Boehringer Ingelheim International GmbH Salt forms of organic compound
TW201036975A (en) 2009-01-07 2010-10-16 Boehringer Ingelheim Int Treatment for diabetes in patients with inadequate glycemic control despite metformin therapy
EP2395983B1 (en) 2009-02-13 2020-04-08 Boehringer Ingelheim International GmbH Pharmaceutical composition comprisng a sglt2 inhibitor, a dpp-iv inhibitor and optionally a further antidiabetic agent and uses thereof
EP3646859A1 (en) 2009-11-27 2020-05-06 Boehringer Ingelheim International GmbH Treatment of genotyped diabetic patients with dpp-iv inhibitors such as linagliptin
AU2011249722B2 (en) 2010-05-05 2015-09-17 Boehringer Ingelheim International Gmbh Combination therapy
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