ATE248153T1 - Neue benzoxazole - Google Patents

Neue benzoxazole

Info

Publication number
ATE248153T1
ATE248153T1 AT95940634T AT95940634T ATE248153T1 AT E248153 T1 ATE248153 T1 AT E248153T1 AT 95940634 T AT95940634 T AT 95940634T AT 95940634 T AT95940634 T AT 95940634T AT E248153 T1 ATE248153 T1 AT E248153T1
Authority
AT
Austria
Prior art keywords
pde
benzoxazoles
new
inhibition
new benzoxazoles
Prior art date
Application number
AT95940634T
Other languages
English (en)
Inventor
David John Cavalla
Mark Chasin
Peter Hofer
Lloyd Dolby
Original Assignee
Euro Celtique Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08321730 external-priority patent/US5665737B1/en
Application filed by Euro Celtique Sa filed Critical Euro Celtique Sa
Application granted granted Critical
Publication of ATE248153T1 publication Critical patent/ATE248153T1/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/56Benzoxazoles; Hydrogenated benzoxazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
    • C07D263/57Aryl or substituted aryl radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
AT95940634T 1994-10-12 1995-10-11 Neue benzoxazole ATE248153T1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08321730 US5665737B1 (en) 1994-10-12 1994-10-12 Substituted benzoxazoles
US46709195A 1995-06-06 1995-06-06
PCT/US1995/014399 WO1996011917A1 (en) 1994-10-12 1995-10-11 Novel benzoxazoles

Publications (1)

Publication Number Publication Date
ATE248153T1 true ATE248153T1 (de) 2003-09-15

Family

ID=26983104

Family Applications (1)

Application Number Title Priority Date Filing Date
AT95940634T ATE248153T1 (de) 1994-10-12 1995-10-11 Neue benzoxazole

Country Status (12)

Country Link
EP (1) EP0785927B1 (de)
KR (1) KR100237962B1 (de)
AT (1) ATE248153T1 (de)
AU (1) AU699489B2 (de)
BG (1) BG101422A (de)
CA (1) CA2202273A1 (de)
DE (1) DE69531623T2 (de)
FI (1) FI971489A (de)
NO (1) NO971684L (de)
PL (1) PL319605A1 (de)
SK (1) SK45497A3 (de)
WO (1) WO1996011917A1 (de)

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Also Published As

Publication number Publication date
DE69531623D1 (de) 2003-10-02
FI971489A (fi) 1997-06-05
FI971489A0 (fi) 1997-04-10
PL319605A1 (en) 1997-08-18
CA2202273A1 (en) 1996-04-25
EP0785927A1 (de) 1997-07-30
AU699489B2 (en) 1998-12-03
SK45497A3 (en) 1997-10-08
EP0785927A4 (de) 1997-12-29
BG101422A (en) 1997-11-28
EP0785927B1 (de) 2003-08-27
DE69531623T2 (de) 2004-06-17
AU4231796A (en) 1996-05-06
KR100237962B1 (ko) 2000-02-01
NO971684L (no) 1997-06-12
WO1996011917A1 (en) 1996-04-25
NO971684D0 (no) 1997-04-11

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