JP2011168609A5 - - Google Patents
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- JP2011168609A5 JP2011168609A5 JP2011092035A JP2011092035A JP2011168609A5 JP 2011168609 A5 JP2011168609 A5 JP 2011168609A5 JP 2011092035 A JP2011092035 A JP 2011092035A JP 2011092035 A JP2011092035 A JP 2011092035A JP 2011168609 A5 JP2011168609 A5 JP 2011168609A5
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- butyl
- methyl
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- 150000001875 compounds Chemical class 0.000 claims 19
- -1 s- butyl Chemical group 0.000 claims 11
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 5
- 125000001511 cyclopentyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 claims 5
- 229910052739 hydrogen Inorganic materials 0.000 claims 5
- 239000001257 hydrogen Substances 0.000 claims 5
- 125000000959 isobutyl group Chemical group [H]C([H])([H])C([H])(C([H])([H])[H])C([H])([H])* 0.000 claims 5
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims 4
- 125000005936 piperidyl group Chemical group 0.000 claims 4
- KUMUCXSUNUNKIJ-UHFFFAOYSA-N 2-[2-[[2-(cyclopentanecarbonyl)-5-methylphenyl]carbamoylamino]-1,3-thiazol-4-yl]acetic acid Chemical compound N=1C(CC(O)=O)=CSC=1NC(=O)NC1=CC(C)=CC=C1C(=O)C1CCCC1 KUMUCXSUNUNKIJ-UHFFFAOYSA-N 0.000 claims 3
- 125000000484 butyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])C([H])([H])[H] 0.000 claims 3
- 125000000113 cyclohexyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 claims 3
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 claims 3
- 125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 claims 3
- 125000001436 propyl group Chemical group [H]C([*])([H])C([H])([H])C([H])([H])[H] 0.000 claims 3
- 150000003839 salts Chemical class 0.000 claims 3
- 125000003718 tetrahydrofuranyl group Chemical group 0.000 claims 3
- 125000001412 tetrahydropyranyl group Chemical group 0.000 claims 3
- 125000000217 alkyl group Chemical group 0.000 claims 2
- 125000001995 cyclobutyl group Chemical group [H]C1([H])C([H])([H])C([H])(*)C1([H])[H] 0.000 claims 2
- 125000000582 cycloheptyl group Chemical group [H]C1([H])C([H])([H])C([H])([H])C([H])([H])C([H])(*)C([H])([H])C1([H])[H] 0.000 claims 2
- 125000001559 cyclopropyl group Chemical group [H]C1([H])C([H])([H])C1([H])* 0.000 claims 2
- 125000004634 hexahydroazepinyl group Chemical group N1(CCCCCC1)* 0.000 claims 2
- 239000012453 solvate Substances 0.000 claims 2
- 125000004632 tetrahydrothiopyranyl group Chemical group S1C(CCCC1)* 0.000 claims 2
- 125000001583 thiepanyl group Chemical group 0.000 claims 2
- 125000001166 thiolanyl group Chemical group 0.000 claims 2
- IGERFAHWSHDDHX-UHFFFAOYSA-N 1,3-dioxanyl Chemical group [CH]1OCCCO1 IGERFAHWSHDDHX-UHFFFAOYSA-N 0.000 claims 1
- JPRPJUMQRZTTED-UHFFFAOYSA-N 1,3-dioxolanyl Chemical group [CH]1OCCO1 JPRPJUMQRZTTED-UHFFFAOYSA-N 0.000 claims 1
- ILWJAOPQHOZXAN-UHFFFAOYSA-N 1,3-dithianyl Chemical group [CH]1SCCCS1 ILWJAOPQHOZXAN-UHFFFAOYSA-N 0.000 claims 1
- FLOJNXXFMHCMMR-UHFFFAOYSA-N 1,3-dithiolanyl Chemical group [CH]1SCCS1 FLOJNXXFMHCMMR-UHFFFAOYSA-N 0.000 claims 1
- 125000005940 1,4-dioxanyl group Chemical group 0.000 claims 1
- HKDFRDIIELOLTJ-UHFFFAOYSA-N 1,4-dithianyl Chemical group [CH]1CSCCS1 HKDFRDIIELOLTJ-UHFFFAOYSA-N 0.000 claims 1
- 125000003903 2-propenyl group Chemical group [H]C([*])([H])C([H])=C([H])[H] 0.000 claims 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 1
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 1
- 125000005411 dithiolanyl group Chemical group S1SC(CC1)* 0.000 claims 1
- 125000001972 isopentyl group Chemical group [H]C([H])([H])C([H])(C([H])([H])[H])C([H])([H])C([H])([H])* 0.000 claims 1
- 125000002757 morpholinyl group Chemical group 0.000 claims 1
- 125000003566 oxetanyl group Chemical group 0.000 claims 1
- 125000003538 pentan-3-yl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])C([H])([H])[H] 0.000 claims 1
- SNOOUWRIMMFWNE-UHFFFAOYSA-M sodium;6-[(3,4,5-trimethoxybenzoyl)amino]hexanoate Chemical compound [Na+].COC1=CC(C(=O)NCCCCCC([O-])=O)=CC(OC)=C1OC SNOOUWRIMMFWNE-UHFFFAOYSA-M 0.000 claims 1
- 125000001424 substituent group Chemical group 0.000 claims 1
- 125000004568 thiomorpholinyl group Chemical group 0.000 claims 1
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DKPA200200999 | 2002-06-27 | ||
| DKPA200200999 | 2002-06-27 | ||
| US39414402P | 2002-07-03 | 2002-07-03 | |
| US60/394,144 | 2002-07-03 | ||
| DKPA200300286 | 2003-02-25 | ||
| DKPA200300286 | 2003-02-25 | ||
| US45222803P | 2003-03-05 | 2003-03-05 | |
| US60/452,228 | 2003-03-05 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004548878A Division JP4881559B2 (ja) | 2002-06-27 | 2003-06-27 | 治療薬としてのアリールカルボニル誘導体 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2011168609A JP2011168609A (ja) | 2011-09-01 |
| JP2011168609A5 true JP2011168609A5 (enExample) | 2012-05-31 |
Family
ID=30003872
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004548878A Expired - Fee Related JP4881559B2 (ja) | 2002-06-27 | 2003-06-27 | 治療薬としてのアリールカルボニル誘導体 |
| JP2010162302A Pending JP2010265306A (ja) | 2002-06-27 | 2010-07-16 | 治療薬としてのアリールカルボニル誘導体 |
| JP2011092035A Withdrawn JP2011168609A (ja) | 2002-06-27 | 2011-04-18 | 治療薬としてのアリールカルボニル誘導体 |
Family Applications Before (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2004548878A Expired - Fee Related JP4881559B2 (ja) | 2002-06-27 | 2003-06-27 | 治療薬としてのアリールカルボニル誘導体 |
| JP2010162302A Pending JP2010265306A (ja) | 2002-06-27 | 2010-07-16 | 治療薬としてのアリールカルボニル誘導体 |
Country Status (12)
| Country | Link |
|---|---|
| US (5) | US7384967B2 (enExample) |
| EP (2) | EP2471533A1 (enExample) |
| JP (3) | JP4881559B2 (enExample) |
| KR (1) | KR101116627B1 (enExample) |
| AU (1) | AU2003243921B2 (enExample) |
| BR (1) | BR0312023A (enExample) |
| CA (2) | CA2744893A1 (enExample) |
| IL (1) | IL165532A (enExample) |
| MX (1) | MXPA05000130A (enExample) |
| NO (1) | NO20111028L (enExample) |
| PL (1) | PL215132B1 (enExample) |
| WO (1) | WO2004002481A1 (enExample) |
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2003
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- 2003-06-27 CA CA2488642A patent/CA2488642C/en not_active Expired - Fee Related
- 2003-06-27 WO PCT/DK2003/000449 patent/WO2004002481A1/en not_active Ceased
- 2003-06-27 AU AU2003243921A patent/AU2003243921B2/en not_active Ceased
- 2003-06-27 MX MXPA05000130A patent/MXPA05000130A/es active IP Right Grant
- 2003-06-27 EP EP11189145A patent/EP2471533A1/en not_active Withdrawn
- 2003-06-27 KR KR1020047021359A patent/KR101116627B1/ko not_active Expired - Fee Related
- 2003-06-27 BR BR0312023-6A patent/BR0312023A/pt not_active Application Discontinuation
- 2003-06-27 EP EP03761446.8A patent/EP1531815B1/en not_active Expired - Lifetime
- 2003-06-27 PL PL374920A patent/PL215132B1/pl unknown
- 2003-06-27 JP JP2004548878A patent/JP4881559B2/ja not_active Expired - Fee Related
- 2003-10-06 US US10/679,887 patent/US7384967B2/en not_active Expired - Fee Related
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2004
- 2004-12-02 IL IL165532A patent/IL165532A/en active IP Right Grant
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2007
- 2007-10-31 US US11/981,997 patent/US8063081B2/en not_active Expired - Lifetime
- 2007-10-31 US US11/982,248 patent/US7897628B2/en not_active Expired - Lifetime
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2010
- 2010-07-16 JP JP2010162302A patent/JP2010265306A/ja active Pending
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2011
- 2011-04-18 JP JP2011092035A patent/JP2011168609A/ja not_active Withdrawn
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2013
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