JP2011037901A5 - - Google Patents

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Publication number
JP2011037901A5
JP2011037901A5 JP2010261857A JP2010261857A JP2011037901A5 JP 2011037901 A5 JP2011037901 A5 JP 2011037901A5 JP 2010261857 A JP2010261857 A JP 2010261857A JP 2010261857 A JP2010261857 A JP 2010261857A JP 2011037901 A5 JP2011037901 A5 JP 2011037901A5
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JP
Japan
Prior art keywords
compound
hydrochloride
tandospirone
buspirone
amd
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
JP2010261857A
Other languages
English (en)
Japanese (ja)
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JP2011037901A (ja
Filing date
Publication date
Application filed filed Critical
Publication of JP2011037901A publication Critical patent/JP2011037901A/ja
Publication of JP2011037901A5 publication Critical patent/JP2011037901A5/ja
Withdrawn legal-status Critical Current

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JP2010261857A 2000-03-17 2010-11-24 網膜外縁部障害の処置に有用な５−ｈｔ１ａ活性を有する化合物 Withdrawn JP2011037901A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US19027900P 2000-03-17 2000-03-17

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
JP2001568420A Division JP4789231B2 (ja) 2000-03-17 2001-02-23 網膜外縁部障害の処置に有用な５−ｈｔ１ａ活性を有する化合物

Publications (2)

Publication Number Publication Date
JP2011037901A JP2011037901A (ja) 2011-02-24
JP2011037901A5 true JP2011037901A5 (enExample) 2012-01-05

Family

ID=22700682

Family Applications (5)

Application Number Title Priority Date Filing Date
JP2001568421A Pending JP2003527423A (ja) 2000-03-17 2001-02-20 緑内障処置用の５−ｈｔ２および５−ｈｔ１ａアゴニスト活性を有する化合物
JP2001568428A Withdrawn JP2003527427A (ja) 2000-03-17 2001-02-23 視野損失を抑制するのに有用な５−ｈｔ活性を有する化合物
JP2001568420A Expired - Fee Related JP4789231B2 (ja) 2000-03-17 2001-02-23 網膜外縁部障害の処置に有用な５−ｈｔ１ａ活性を有する化合物
JP2010261857A Withdrawn JP2011037901A (ja) 2000-03-17 2010-11-24 網膜外縁部障害の処置に有用な５−ｈｔ１ａ活性を有する化合物
JP2011108785A Withdrawn JP2011153158A (ja) 2000-03-17 2011-05-13 網膜外縁部障害の処置に有用な５−ｈｔ１ａ活性を有する化合物

Family Applications Before (3)

Application Number Title Priority Date Filing Date
JP2001568421A Pending JP2003527423A (ja) 2000-03-17 2001-02-20 緑内障処置用の５−ｈｔ２および５−ｈｔ１ａアゴニスト活性を有する化合物
JP2001568428A Withdrawn JP2003527427A (ja) 2000-03-17 2001-02-23 視野損失を抑制するのに有用な５−ｈｔ活性を有する化合物
JP2001568420A Expired - Fee Related JP4789231B2 (ja) 2000-03-17 2001-02-23 網膜外縁部障害の処置に有用な５−ｈｔ１ａ活性を有する化合物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2011108785A Withdrawn JP2011153158A (ja) 2000-03-17 2011-05-13 網膜外縁部障害の処置に有用な５−ｈｔ１ａ活性を有する化合物

Country Status (18)

Country Link
EP (3) EP1263434A1 (enExample)
JP (5) JP2003527423A (enExample)
KR (3) KR20030016239A (enExample)
CN (2) CN1198605C (enExample)
AR (1) AR028258A1 (enExample)
AT (1) ATE247507T1 (enExample)
AU (5) AU2001238552A1 (enExample)
BR (3) BR0109193A (enExample)
CA (3) CA2400637A1 (enExample)
DE (1) DE60100625T2 (enExample)
DK (1) DK1263504T3 (enExample)
ES (1) ES2204848T3 (enExample)
MX (3) MXPA02009071A (enExample)
PL (1) PL203709B1 (enExample)
PT (1) PT1263504E (enExample)
TW (1) TWI268777B (enExample)
WO (3) WO2001070223A1 (enExample)
ZA (1) ZA200206350B (enExample)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6960579B1 (en) 1998-05-19 2005-11-01 Alcon Manufacturing, Ltd. Serotonergic 5HT7 receptor compounds for treating ocular and CNS disorders
US20030207890A1 (en) 2001-02-23 2003-11-06 Collier Robert J Compounds with 5-ht1a activity useful for treating disorders of the outer retina
EP1263434A1 (en) * 2000-03-17 2002-12-11 Alcon, Inc Compounds with 5-ht 2 and 5-ht 1a agonist activity for treating glaucoma
TW593302B (en) * 2001-12-20 2004-06-21 Alcon Inc Novel benzodifuranimidazoline and benzofuranimidazoline derivatives and their use for the treatment of glaucoma
BR0316775A (pt) 2002-12-13 2005-11-01 Alcon Inc Novos análogos de benzopirano e seu uso para o tratamento de glaucoma
JP2004262812A (ja) * 2003-02-28 2004-09-24 Rohto Pharmaceut Co Ltd 眼圧低下剤
EP1617838A4 (en) * 2003-04-25 2011-07-06 Mitsubishi Tanabe Pharma Corp COMPOSITION FOR ORAL ADMINISTRATION WITH ALKYLENEDIOXYBENZOLE DERIVATIVES
US7476687B2 (en) 2003-11-26 2009-01-13 Alcon, Inc. Substituted furo[2,3-g]indazoles for the treatment of glaucoma
AR046890A1 (es) 2003-12-15 2005-12-28 Alcon Inc [1,4] oxazino [2,3-g] indazoles sustituidos para el tratamiento del glaucoma.
US7338972B1 (en) 2003-12-15 2008-03-04 Alcon, Inc. Substituted 1-alkylamino-1H-indazoles for the treatment of glaucoma
US7129257B1 (en) 2003-12-15 2006-10-31 Alcon, Inc. Pyrazolo[3,4- e]benzoxazoles for the treatment of glaucoma
US20050244463A1 (en) 2004-04-30 2005-11-03 Allergan, Inc. Sustained release intraocular implants and methods for treating ocular vasculopathies
JP5173190B2 (ja) 2004-08-25 2013-03-27 武田薬品工業株式会社 腹圧性尿失禁の予防・治療剤及びそのスクリーニング方法
WO2006062839A1 (en) 2004-12-08 2006-06-15 Alcon, Inc. Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma
JP5528699B2 (ja) 2006-05-16 2014-06-25 武田薬品工業株式会社 縮合複素環化合物およびその用途
WO2008024846A2 (en) * 2006-08-25 2008-02-28 Allergan, Inc. Brimonidine and timolol compositions
EP2896624B1 (en) 2007-03-28 2016-07-13 Atir Holding S.A. Heterotricyclic compounds as serotonergic and/or dopaminergic agents and uses thereof
JP5520051B2 (ja) 2007-11-15 2014-06-11 武田薬品工業株式会社 縮合ピリジン誘導体およびその用途
TW201010727A (en) * 2008-09-03 2010-03-16 Alcon Res Ltd Pharmaceutical composition having relatively low ionic strength
NZ716349A (en) 2009-11-09 2017-07-28 Allergan Inc Compositions and methods for stimulating hair growth
WO2011071136A1 (ja) 2009-12-11 2011-06-16 アステラス製薬株式会社 線維筋痛症治療剤
EP2956096A1 (en) 2013-02-15 2015-12-23 Allergan, Inc. Sustained drug delivery implant
EP3519816A4 (en) 2016-09-29 2020-05-06 The Regents of the University of California CONNECTIONS FOR INCREASING NEURONAL PLASTICITY
WO2019131902A1 (ja) 2017-12-27 2019-07-04 武田薬品工業株式会社 腹圧性尿失禁および便失禁の治療薬
WO2020176597A1 (en) 2019-02-27 2020-09-03 The Regents Of The University Of California N-substituted indoles and other heterocycles for treating brain disorders
KR102946120B1 (ko) 2019-02-27 2026-03-30 더 리젠츠 오브 더 유니버시티 오브 캘리포니아 뇌 장애를 치료하기 위한 아제피노-인돌 및 다른 헤테로사이클
WO2022221415A2 (en) 2021-04-13 2022-10-20 The Regents Of The University Of California Tetracyclic compounds for treating brain disorders
JP2025502615A (ja) 2021-12-15 2025-01-28 デリックス セラピューティクス，インク． フェノキシおよびベンジルオキシ置換サイコプラストゲンならびにその使用
DK4452267T3 (da) * 2021-12-23 2025-05-26 Cilcare Dev 4-phenyl-tetrahydropyridinderivater til behandling af hørelidelser

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH02262518A (ja) * 1989-04-03 1990-10-25 Kaken Pharmaceut Co Ltd 眼圧調整剤
JP2824863B2 (ja) * 1989-07-12 1998-11-18 エーザイ株式会社 α▲下１▼―ブロッカー点眼剤
TW270114B (enExample) * 1993-10-22 1996-02-11 Hoffmann La Roche
US5521183A (en) * 1994-08-30 1996-05-28 Allergan Use of 5-HT ligands as anti-pruritic agents
US5998467A (en) * 1995-10-25 1999-12-07 Mitsubishi Chemical Corporation Medicine for oculopathy
JP3958391B2 (ja) * 1995-10-25 2007-08-15 三菱化学株式会社 眼疾患用薬剤
WO1998018458A1 (en) * 1996-10-31 1998-05-07 Alcon Laboratories, Inc. Opthalmological compositions containing serotonin 5-ht1a receptor agonist and their use in the treatment of glaucoma
DE19751949A1 (de) * 1997-11-24 1999-05-27 Bayer Ag Verwendung von substituierten Aminomethyl-Chromanen zur Verhinderung der neuronalen Degeneration und zur Förderung der neuronalen Regeneration
GB9819033D0 (en) * 1998-09-01 1998-10-28 Cerebrus Ltd Chemical compounds VI
EP1263434A1 (en) * 2000-03-17 2002-12-11 Alcon, Inc Compounds with 5-ht 2 and 5-ht 1a agonist activity for treating glaucoma

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