HUP0204137A2 - Fulvesztrantot tartalmazó gyógyászati készítmény - Google Patents

Fulvesztrantot tartalmazó gyógyászati készítmény

Info

Publication number
HUP0204137A2
HUP0204137A2 HU0204137A HUP0204137A HUP0204137A2 HU P0204137 A2 HUP0204137 A2 HU P0204137A2 HU 0204137 A HU0204137 A HU 0204137A HU P0204137 A HUP0204137 A HU P0204137A HU P0204137 A2 HUP0204137 A2 HU P0204137A2
Authority
HU
Hungary
Prior art keywords
fulvestrant
pharmaceutical composition
active ingredient
ricinoleate carrier
ricinoleate
Prior art date
Application number
HU0204137A
Other languages
English (en)
Inventor
John Raymond Evans
Rosalind Ursula Grundy
Original Assignee
Astrazeneca Ab,
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26243352&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HUP0204137(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab, filed Critical Astrazeneca Ab,
Publication of HUP0204137A2 publication Critical patent/HUP0204137A2/hu
Publication of HUP0204137A3 publication Critical patent/HUP0204137A3/hu
Publication of HU230162B1 publication Critical patent/HU230162B1/hu

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32Antioestrogens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/44Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

A találmány injekció formájában beadható, hatóanyagként 7a-[9-(4,4,5,5,5-pentafluor-pentilszulfinil)-nonil]-ösztra-1,3,5(10)-trién-3,17b-diolt (azaz fulvesztrantot) tartalmazó, nyújtott hatóanyag-felszabadulású gyógyászati készítményre vonatkozik. A találmányszerinti készítmény a hatóanyagot olyan ricinoleát hordozóban oldvatartalmazza, amely még legalább egy alkoholt és a ricinoleáthordozóanyaggal elegyíthető nemvizes észter oldószert is tartalmaz. Ó
HU0204137A 2000-01-10 2001-01-08 Fulvesztrantot tartalmazó gyógyászati készítmény HU230162B1 (hu)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB0000313.7 2000-01-10
GBGB0000313.7A GB0000313D0 (en) 2000-01-10 2000-01-10 Formulation
GB0008837.7 2000-04-12
GBGB0008837.7A GB0008837D0 (en) 2000-01-10 2000-04-12 Formulation
PCT/GB2001/000049 WO2001051056A1 (en) 2000-01-10 2001-01-08 Fulvestrant formulation

Publications (3)

Publication Number Publication Date
HUP0204137A2 true HUP0204137A2 (hu) 2003-04-28
HUP0204137A3 HUP0204137A3 (en) 2005-03-29
HU230162B1 HU230162B1 (hu) 2015-09-28

Family

ID=26243352

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0204137A HU230162B1 (hu) 2000-01-10 2001-01-08 Fulvesztrantot tartalmazó gyógyászati készítmény

Country Status (41)

Country Link
US (5) US20030125387A1 (hu)
EP (4) EP1250138B2 (hu)
JP (3) JP3713237B2 (hu)
KR (1) KR100802366B1 (hu)
CN (1) CN1222292C (hu)
AR (1) AR027510A1 (hu)
AT (1) ATE306928T1 (hu)
AU (1) AU762080B2 (hu)
BE (1) BE1013477A3 (hu)
BG (1) BG65776B1 (hu)
BR (1) BR0107445B1 (hu)
CA (1) CA2351004C (hu)
CH (1) CH696260A5 (hu)
CO (1) CO5280206A1 (hu)
CY (1) CY1116520T1 (hu)
CZ (1) CZ304689B6 (hu)
DE (2) DE60114145T3 (hu)
DK (2) DK1250138T4 (hu)
EE (1) EE05421B1 (hu)
EG (1) EG24074A (hu)
ES (3) ES2248272T5 (hu)
FR (1) FR2803516B1 (hu)
GB (3) GB0000313D0 (hu)
HK (3) HK1049286B (hu)
HU (1) HU230162B1 (hu)
IL (2) IL150230A0 (hu)
IS (1) IS2932B (hu)
IT (2) ITTO20010005A1 (hu)
MX (1) MXPA02006698A (hu)
MY (1) MY118583A (hu)
NL (1) NL1017075C2 (hu)
NO (2) NO336286B1 (hu)
PL (1) PL202525B1 (hu)
PT (2) PT2266573E (hu)
RU (1) RU2263507C9 (hu)
SI (2) SI2266573T1 (hu)
SK (1) SK287221B6 (hu)
TW (1) TWI259086B (hu)
UA (1) UA75879C2 (hu)
WO (1) WO2001051056A1 (hu)
ZA (1) ZA200204165B (hu)

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