DD247681A5 - Verfahren zur herstellung von 16,17-acetalsubstituierten androstan-17 beta- carbonsaeureestern - Google Patents

Verfahren zur herstellung von 16,17-acetalsubstituierten androstan-17 beta- carbonsaeureestern Download PDF

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Publication number
DD247681A5
DD247681A5 DD86288744A DD28874486A DD247681A5 DD 247681 A5 DD247681 A5 DD 247681A5 DD 86288744 A DD86288744 A DD 86288744A DD 28874486 A DD28874486 A DD 28874486A DD 247681 A5 DD247681 A5 DD 247681A5
Authority
DD
German Democratic Republic
Prior art keywords
sub
hydrogen
hydroxy
dien
carboxylate
Prior art date
Application number
DD86288744A
Other languages
German (de)
English (en)
Inventor
Paul H Andersson
Per T Andersson
Bengt I Axelsson
Bror A Thalen
Jan W Trofast
Original Assignee
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Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by ������@������������k�� filed Critical ������@������������k��
Publication of DD247681A5 publication Critical patent/DD247681A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/0026—Oxygen-containing hetero ring cyclic ketals
    • C07J71/0031—Oxygen-containing hetero ring cyclic ketals at positions 16, 17
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/38—Drugs for disorders of the endocrine system of the suprarenal hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Fats And Perfumes (AREA)
  • Threshing Machine Elements (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Crystals, And After-Treatments Of Crystals (AREA)
DD86288744A 1985-04-04 1986-04-03 Verfahren zur herstellung von 16,17-acetalsubstituierten androstan-17 beta- carbonsaeureestern DD247681A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
SE8501693A SE8501693D0 (sv) 1985-04-04 1985-04-04 Novel 16,17-acetalsubstituted androstane-17beta-carboxylic acid esters

Publications (1)

Publication Number Publication Date
DD247681A5 true DD247681A5 (de) 1987-07-15

Family

ID=20359775

Family Applications (2)

Application Number Title Priority Date Filing Date
DD86288744A DD247681A5 (de) 1985-04-04 1986-04-03 Verfahren zur herstellung von 16,17-acetalsubstituierten androstan-17 beta- carbonsaeureestern
DD87305598A DD261364A5 (de) 1985-04-04 1987-07-31 Verfahren zur herstellung von ausgangsverbindungen fuer glucocorticosteroiden, die in der humanmedizin und veterinaermedizin angewendet werden kann

Family Applications After (1)

Application Number Title Priority Date Filing Date
DD87305598A DD261364A5 (de) 1985-04-04 1987-07-31 Verfahren zur herstellung von ausgangsverbindungen fuer glucocorticosteroiden, die in der humanmedizin und veterinaermedizin angewendet werden kann

Country Status (31)

Country Link
US (1) US4950659A (es)
EP (2) EP0355859B1 (es)
JP (1) JPH0762028B2 (es)
KR (1) KR930009444B1 (es)
CN (1) CN1021444C (es)
AT (2) ATE107657T1 (es)
AU (1) AU590545B2 (es)
CA (1) CA1333597C (es)
CS (1) CS266581B2 (es)
DD (2) DD247681A5 (es)
DE (2) DE3689936T2 (es)
DK (3) DK165638C (es)
ES (2) ES8800264A1 (es)
FI (1) FI85378C (es)
GR (1) GR860902B (es)
HU (2) HU196830B (es)
IE (1) IE61474B1 (es)
IL (1) IL78143A0 (es)
JO (1) JO1479B1 (es)
LT (3) LT3812B (es)
LV (3) LV10281B (es)
MY (1) MY102056A (es)
NO (1) NO165298C (es)
NZ (1) NZ215586A (es)
PH (2) PH23547A (es)
PL (2) PL150052B1 (es)
PT (1) PT82340B (es)
RU (3) RU1795972C (es)
SE (1) SE8501693D0 (es)
UA (2) UA13319A (es)
ZA (1) ZA861884B (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE8501693D0 (sv) 1985-04-04 1985-04-04 Draco Ab Novel 16,17-acetalsubstituted androstane-17beta-carboxylic acid esters
HU203769B (en) * 1989-03-09 1991-09-30 Richter Gedeon Vegyeszet Process for producing new steroide derivatives and pharmaceutical compositions containing them
ATE154607T1 (de) * 1992-12-24 1997-07-15 Rhone Poulenc Rorer Ltd Neue steroide
GB9423919D0 (en) * 1994-11-26 1995-01-11 Rhone Poulenc Rorer Ltd Chemical process
GB0110411D0 (en) * 2001-04-27 2001-06-20 Astrazeneca Ab Chemical process

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3828080A (en) * 1972-01-20 1974-08-06 Glaxo Lab Ltd Androstane-17beta-carboxylic acids and processes for the preparation thereof
SE378109B (es) * 1972-05-19 1975-08-18 Bofors Ab
GB1438940A (en) * 1972-07-19 1976-06-09 Glaxo Lab Ltd 17beta-haloalkoxycarbonyl-17alpha-oxysteroids
GB1517278A (en) * 1974-08-30 1978-07-12 Glaxo Lab Ltd Alkyl and haloalkyl androsta-1,4,15-triene and-4,15-diene-17beta-carboxylates
CH628355A5 (de) * 1976-02-24 1982-02-26 Ciba Geigy Ag Verfahren zur herstellung neuer androstadien-17beta-carbonsaeuren und ihrer ester und salze.
US4198336A (en) 1978-04-05 1980-04-15 Syntex (U.S.A.) Inc. Chemical process for preparing androsta-4-ene 17α-carboxylic acids
ZA814440B (en) * 1980-07-10 1982-10-27 Otsuka Pharma Co Ltd Soft steroids having anti-inflammatory activity
SE449106B (sv) * 1980-07-10 1987-04-06 Otsuka Pharma Co Ltd Steroid med anti-inflammatorisk verkan samt komposition innehallande denna
ZA817929B (en) * 1980-12-22 1982-10-27 Upjohn Co 5alpha-and 5beta-androstane-17beta-carboxylates
SE8306370D0 (sv) * 1983-11-18 1983-11-18 Draco Ab Novel androstane-17beta-carboxylic acid esters, a process and intermediates for their preparation, compositions and method for the treatment of inflammatory conditions
SE8403905D0 (sv) * 1984-07-30 1984-07-30 Draco Ab Liposomes and steroid esters
SE8501693D0 (sv) 1985-04-04 1985-04-04 Draco Ab Novel 16,17-acetalsubstituted androstane-17beta-carboxylic acid esters
JP2687768B2 (ja) * 1991-07-30 1997-12-08 トヨタ自動車株式会社 エンジンの制御装置

Also Published As

Publication number Publication date
LT3913B (en) 1996-04-25
DK165638C (da) 1993-06-01
KR930009444B1 (ko) 1993-10-04
SE8501693D0 (sv) 1985-04-04
PH23547A (en) 1989-08-25
DK59693A (da) 1993-05-21
FI85378C (fi) 1992-04-10
FI861275A (fi) 1986-10-05
GR860902B (en) 1986-07-29
PL265699A1 (en) 1988-03-03
HU196830B (en) 1989-01-30
PT82340A (en) 1986-05-01
IL78143A0 (en) 1986-07-31
LT3811B (en) 1996-03-25
HUT40809A (en) 1987-02-27
DK167150B1 (da) 1993-09-06
JO1479B1 (en) 1988-03-10
LTIP1677A (en) 1995-07-25
DK167574B1 (da) 1993-11-22
LV10960B (en) 1996-08-20
JPS61236794A (ja) 1986-10-22
DK59693D0 (da) 1993-05-21
CN86102193A (zh) 1987-09-02
LV10960A (lv) 1995-12-20
NO165298B (no) 1990-10-15
LTIP1678A (en) 1995-07-25
NZ215586A (en) 1990-01-29
DK138386A (da) 1986-10-05
UA19288A (uk) 1997-12-25
DK138386D0 (da) 1986-03-25
IE860879L (en) 1986-10-04
ES557314A0 (es) 1988-05-16
LV10281A (lv) 1994-10-20
FI85378B (fi) 1991-12-31
DK165638B (da) 1992-12-28
AU5486886A (en) 1986-10-16
RU1779257C (ru) 1992-11-30
DE3689936T2 (de) 1994-09-29
DE3687239T2 (de) 1993-04-15
EP0355859B1 (en) 1994-06-22
NO861313L (no) 1986-10-06
LV10957A (lv) 1995-12-20
ATE83241T1 (de) 1992-12-15
LV10281B (en) 1995-04-20
LTIP1676A (en) 1995-07-25
JPH0762028B2 (ja) 1995-07-05
IE61474B1 (en) 1994-11-02
MY102056A (en) 1992-03-31
LT3812B (en) 1996-03-25
EP0197018B1 (en) 1992-12-09
FI861275A0 (fi) 1986-03-25
US4950659A (en) 1990-08-21
CA1333597C (en) 1994-12-20
ES8800264A1 (es) 1987-10-16
ATE107657T1 (de) 1994-07-15
DE3687239D1 (de) 1993-01-21
DK59392D0 (da) 1992-05-05
CN1021444C (zh) 1993-06-30
UA13319A (uk) 1997-02-28
DE3689936D1 (de) 1994-07-28
RU2081879C1 (ru) 1997-06-20
KR860008208A (ko) 1986-11-14
AU590545B2 (en) 1989-11-09
PH24369A (en) 1990-06-13
DK59392A (da) 1992-05-05
LV10957B (en) 1996-04-20
HU199872B (en) 1990-03-28
ES8802392A1 (es) 1988-05-16
EP0355859A1 (en) 1990-02-28
EP0197018A1 (en) 1986-10-08
ES553675A0 (es) 1987-10-16
PT82340B (pt) 1988-10-14
NO165298C (no) 1991-01-23
CS266581B2 (en) 1990-01-12
CS232886A2 (en) 1989-04-14
PL150052B1 (en) 1990-04-30
ZA861884B (en) 1987-07-29
DD261364A5 (de) 1988-10-26
RU1795972C (ru) 1993-02-15
PL148272B1 (en) 1989-09-30

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IF04 In force in the year 2004

Expiry date: 20060404