AU2003253418B2 - 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments - Google Patents

8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments Download PDF

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Publication number
AU2003253418B2
AU2003253418B2 AU2003253418A AU2003253418A AU2003253418B2 AU 2003253418 B2 AU2003253418 B2 AU 2003253418B2 AU 2003253418 A AU2003253418 A AU 2003253418A AU 2003253418 A AU2003253418 A AU 2003253418A AU 2003253418 B2 AU2003253418 B2 AU 2003253418B2
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Australia
Prior art keywords
methyl
xanthine
piperidin
mass spectrum
butyn
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active, expires
Application number
AU2003253418A
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AU2003253418A1 (en
Inventor
Matthias Eckhardt
Frank Himmelsbach
Elke Langkopf
Ralf Richard Hermann Lotz
Roland Maier
Michael Mark
Mohammad Tadayyon
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
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Boehringer Ingelheim Pharma GmbH and Co KG
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=31947613&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AU2003253418(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from DE10238243A external-priority patent/DE10238243A1/de
Priority claimed from DE10312353A external-priority patent/DE10312353A1/de
Application filed by Boehringer Ingelheim Pharma GmbH and Co KG filed Critical Boehringer Ingelheim Pharma GmbH and Co KG
Publication of AU2003253418A1 publication Critical patent/AU2003253418A1/en
Priority to AU2010201384A priority Critical patent/AU2010201384C1/en
Application granted granted Critical
Publication of AU2003253418B2 publication Critical patent/AU2003253418B2/en
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
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    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • C07D473/12Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1, 3, and 7, e.g. caffeine

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AU2003253418A 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments Active 2026-11-01 AU2003253418B2 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU2010201384A AU2010201384C1 (en) 2002-08-21 2010-04-07 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DE10238243A DE10238243A1 (de) 2002-08-21 2002-08-21 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
DE10238243.3 2002-08-21
DE10312353.9 2003-03-20
DE10312353A DE10312353A1 (de) 2003-03-20 2003-03-20 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel
PCT/EP2003/009127 WO2004018468A2 (de) 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-yl]-xanthine, deren herstellung und deren verwendung als arzneimittel

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AU2010201384A Division AU2010201384C1 (en) 2002-08-21 2010-04-07 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

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AU2003253418A1 AU2003253418A1 (en) 2004-03-11
AU2003253418B2 true AU2003253418B2 (en) 2010-04-22

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AU2003253418A Active 2026-11-01 AU2003253418B2 (en) 2002-08-21 2003-08-18 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments
AU2010201384A Active 2028-05-21 AU2010201384C1 (en) 2002-08-21 2010-04-07 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments

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EP (6) EP2058311A3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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