AU2003253418B2 - 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments - Google Patents
8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments Download PDFInfo
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- AU2003253418B2 AU2003253418B2 AU2003253418A AU2003253418A AU2003253418B2 AU 2003253418 B2 AU2003253418 B2 AU 2003253418B2 AU 2003253418 A AU2003253418 A AU 2003253418A AU 2003253418 A AU2003253418 A AU 2003253418A AU 2003253418 B2 AU2003253418 B2 AU 2003253418B2
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- methyl
- xanthine
- piperidin
- mass spectrum
- butyn
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- C—CHEMISTRY; METALLURGY
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- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- General Health & Medical Sciences (AREA)
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Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AU2010201384A AU2010201384C1 (en) | 2002-08-21 | 2010-04-07 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10238243A DE10238243A1 (de) | 2002-08-21 | 2002-08-21 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
DE10238243.3 | 2002-08-21 | ||
DE10312353.9 | 2003-03-20 | ||
DE10312353A DE10312353A1 (de) | 2003-03-20 | 2003-03-20 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
PCT/EP2003/009127 WO2004018468A2 (de) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-yl]-xanthine, deren herstellung und deren verwendung als arzneimittel |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2010201384A Division AU2010201384C1 (en) | 2002-08-21 | 2010-04-07 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2003253418A1 AU2003253418A1 (en) | 2004-03-11 |
AU2003253418B2 true AU2003253418B2 (en) | 2010-04-22 |
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Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU2003253418A Active 2026-11-01 AU2003253418B2 (en) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
AU2010201384A Active 2028-05-21 AU2010201384C1 (en) | 2002-08-21 | 2010-04-07 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
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AU2010201384A Active 2028-05-21 AU2010201384C1 (en) | 2002-08-21 | 2010-04-07 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
Country Status (38)
Families Citing this family (182)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1509525B9 (en) * | 2002-05-31 | 2007-10-31 | Schering Corporation | Process for preparing xanthine phosphodiesterase v inhibitors and precursors thereof |
GB0215293D0 (en) | 2002-07-03 | 2002-08-14 | Rega Foundation | Viral inhibitors |
SI1532149T1 (sl) * | 2002-08-21 | 2010-05-31 | Boehringer Ingelheim Pharma | amino piperidin il ksantini njihova priprava in njihova uporaba kot zdravila |
US7407955B2 (en) | 2002-08-21 | 2008-08-05 | Boehringer Ingelheim Pharma Gmbh & Co., Kg | 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions |
US7495005B2 (en) | 2002-08-22 | 2009-02-24 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Xanthine derivatives, their preparation and their use in pharmaceutical compositions |
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