SK282524B6 - Opticky čisté soli (-)-enantioméru pyridylmetylsulfinyl-1H- benzimidazolových zlúčenín, spôsob ich prípravy, farmaceutický prostriedok s ich obsahom, ich použitie a medziprodukty na ich prípravu - Google Patents

Opticky čisté soli (-)-enantioméru pyridylmetylsulfinyl-1H- benzimidazolových zlúčenín, spôsob ich prípravy, farmaceutický prostriedok s ich obsahom, ich použitie a medziprodukty na ich prípravu Download PDF

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Publication number
SK282524B6
SK282524B6 SK101-95A SK10195A SK282524B6 SK 282524 B6 SK282524 B6 SK 282524B6 SK 10195 A SK10195 A SK 10195A SK 282524 B6 SK282524 B6 SK 282524B6
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SK
Slovakia
Prior art keywords
methoxy
preparation
optically pure
methyl
pyridyl
Prior art date
Application number
SK101-95A
Other languages
English (en)
Slovak (sk)
Other versions
SK10195A3 (en
Inventor
Per Lennart Lindberg
Unge Sverker Von
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of SK10195A3 publication Critical patent/SK10195A3/sk
Publication of SK282524B6 publication Critical patent/SK282524B6/sk

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
SK101-95A 1993-05-28 1994-05-27 Opticky čisté soli (-)-enantioméru pyridylmetylsulfinyl-1H- benzimidazolových zlúčenín, spôsob ich prípravy, farmaceutický prostriedok s ich obsahom, ich použitie a medziprodukty na ich prípravu SK282524B6 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE19939301830A SE9301830D0 (sv) 1993-05-28 1993-05-28 New compounds
PCT/SE1994/000509 WO1994027988A1 (en) 1993-05-28 1994-05-27 Optically pure salts of pyridinylmethyl sulfinyl-ih-benzimidazole compounds

Publications (2)

Publication Number Publication Date
SK10195A3 SK10195A3 (en) 1995-09-13
SK282524B6 true SK282524B6 (sk) 2002-10-08

Family

ID=20390088

Family Applications (1)

Application Number Title Priority Date Filing Date
SK101-95A SK282524B6 (sk) 1993-05-28 1994-05-27 Opticky čisté soli (-)-enantioméru pyridylmetylsulfinyl-1H- benzimidazolových zlúčenín, spôsob ich prípravy, farmaceutický prostriedok s ich obsahom, ich použitie a medziprodukty na ich prípravu

Country Status (43)

Country Link
US (5) US5693818A (xx)
EP (3) EP1020460B1 (xx)
JP (3) JP3549111B2 (xx)
KR (1) KR100337274B1 (xx)
CN (2) CN1055469C (xx)
AT (1) ATE197452T1 (xx)
CA (2) CA2139653C (xx)
CL (1) CL2009000805A1 (xx)
CY (1) CY2224B1 (xx)
CZ (1) CZ287876B6 (xx)
DE (4) DE69435221D1 (xx)
DK (3) DK1020460T3 (xx)
DZ (1) DZ1785A1 (xx)
EE (1) EE03157B1 (xx)
ES (3) ES2099047T3 (xx)
FI (2) FI117755B (xx)
GR (2) GR970300012T1 (xx)
HK (3) HK1008330A1 (xx)
HR (1) HRP940307B1 (xx)
HU (1) HU226824B1 (xx)
IL (1) IL109684A (xx)
IS (1) IS1854B (xx)
LT (1) LT3287B (xx)
LU (1) LU91870I2 (xx)
LV (1) LV11034B (xx)
MA (1) MA23210A1 (xx)
MY (1) MY121192A (xx)
NO (2) NO307378B1 (xx)
NZ (1) NZ266915A (xx)
PL (1) PL178994B1 (xx)
PT (3) PT652872E (xx)
RU (1) RU2137766C1 (xx)
SA (2) SA05260103B1 (xx)
SE (1) SE9301830D0 (xx)
SG (1) SG49283A1 (xx)
SI (2) SI22752B (xx)
SK (1) SK282524B6 (xx)
TN (1) TNSN94058A1 (xx)
TW (1) TW389761B (xx)
UA (1) UA60289C2 (xx)
WO (1) WO1994027988A1 (xx)
YU (1) YU49065B (xx)
ZA (1) ZA943557B (xx)

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