PT929563E - Cetolidos 6-0-substituidos possuindo actividade antibacteriana - Google Patents

Cetolidos 6-0-substituidos possuindo actividade antibacteriana

Info

Publication number
PT929563E
PT929563E PT97939765T PT97939765T PT929563E PT 929563 E PT929563 E PT 929563E PT 97939765 T PT97939765 T PT 97939765T PT 97939765 T PT97939765 T PT 97939765T PT 929563 E PT929563 E PT 929563E
Authority
PT
Portugal
Prior art keywords
alkyl
substituted
heteroaryl
aryl
optionally substituted
Prior art date
Application number
PT97939765T
Other languages
English (en)
Inventor
Yat Sun Or
Daniel T Chu
Jacob J Plattner
Richard F Clark
Zhenkun Ma
Original Assignee
Abbott Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27107953&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT929563(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/888,350 external-priority patent/US5866549A/en
Application filed by Abbott Lab filed Critical Abbott Lab
Publication of PT929563E publication Critical patent/PT929563E/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00Processes for the preparation of sugar derivatives
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Cephalosporin Compounds (AREA)
  • Food Preservation Except Freezing, Refrigeration, And Drying (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
PT97939765T 1996-09-04 1997-09-02 Cetolidos 6-0-substituidos possuindo actividade antibacteriana PT929563E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US70777696A 1996-09-04 1996-09-04
US08/888,350 US5866549A (en) 1996-09-04 1997-07-03 6-O-substituted ketolides having antibacterial activity

Publications (1)

Publication Number Publication Date
PT929563E true PT929563E (pt) 2005-10-31

Family

ID=27107953

Family Applications (5)

Application Number Title Priority Date Filing Date
PT97939765T PT929563E (pt) 1996-09-04 1997-09-02 Cetolidos 6-0-substituidos possuindo actividade antibacteriana
PT02024558T PT1291351E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos possuindo actividade antibacteriana
PT02024557T PT1291350E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos que possuem actividade antibacteriana
PT02024560T PT1291353E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos possuindo actividade antibacteriana
PT02024559T PT1291352E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos possuindo actividade antibacteriana

Family Applications After (4)

Application Number Title Priority Date Filing Date
PT02024558T PT1291351E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos possuindo actividade antibacteriana
PT02024557T PT1291350E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos que possuem actividade antibacteriana
PT02024560T PT1291353E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos possuindo actividade antibacteriana
PT02024559T PT1291352E (pt) 1996-09-04 1997-09-02 Cetolidos 6-o-substituidos possuindo actividade antibacteriana

Country Status (28)

Country Link
US (4) US6075133A (pt)
EP (5) EP1291353B1 (pt)
JP (1) JP4597274B2 (pt)
KR (5) KR20050044816A (pt)
CN (4) CN1680419A (pt)
AT (5) ATE296832T1 (pt)
BG (1) BG63547B1 (pt)
BR (1) BR9711661A (pt)
CA (1) CA2263972C (pt)
CZ (1) CZ300106B6 (pt)
DE (5) DE69733370T2 (pt)
DK (5) DK1291350T3 (pt)
ES (5) ES2242813T3 (pt)
HK (1) HK1021537A1 (pt)
HR (5) HRP970473B1 (pt)
HU (1) HU230166B1 (pt)
ID (1) ID19406A (pt)
IL (1) IL128681A0 (pt)
NO (1) NO314230B1 (pt)
NZ (1) NZ334274A (pt)
PL (1) PL188173B1 (pt)
PT (5) PT929563E (pt)
RO (1) RO121473B1 (pt)
RU (1) RU2192427C2 (pt)
SI (1) SI20023B (pt)
SK (5) SK286181B6 (pt)
TR (1) TR199901127T2 (pt)
WO (1) WO1998009978A1 (pt)

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US6265202B1 (en) 1998-06-26 2001-07-24 Regents Of The University Of Minnesota DNA encoding methymycin and pikromycin
FR2780977B1 (fr) * 1998-07-09 2000-09-01 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2792637B1 (fr) * 1999-04-26 2001-06-01 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
JP4573925B2 (ja) 1998-07-09 2010-11-04 アベンティス・ファーマ・ソシエテ・アノニム 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用
FR2785612A1 (fr) * 1998-11-10 2000-05-12 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
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CN109942653B (zh) * 2019-02-27 2021-06-25 北京理工大学 一种红霉素衍生物及其制备方法
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Also Published As

Publication number Publication date
DK0929563T3 (da) 2005-10-03
HRP20060278B1 (hr) 2014-04-11
CN100441591C (zh) 2008-12-10
RU2192427C2 (ru) 2002-11-10
KR20050043993A (ko) 2005-05-11
HUP9902869A3 (en) 2001-04-28
PT1291352E (pt) 2005-09-30
ATE296831T1 (de) 2005-06-15
NO991022L (no) 1999-05-03
DK1291350T3 (da) 2005-09-26
SK286181B6 (sk) 2008-04-07
HRP20060275B1 (hr) 2014-04-11
KR100610043B1 (ko) 2006-08-08
DE69733723T2 (de) 2006-04-20
HRP20060276A2 (en) 2007-10-31
HRP20060277B1 (hr) 2014-04-11
HK1021537A1 (en) 2000-06-16
DE69733369D1 (de) 2005-06-30
SK285535B6 (sk) 2007-03-01
ES2242983T3 (es) 2005-11-16
PL332009A1 (en) 1999-08-16
EP1291352A1 (en) 2003-03-12
DE69733369T2 (de) 2006-01-26
RO121473B1 (ro) 2007-06-29
HRP20060276B1 (hr) 2014-04-25
KR100568455B1 (ko) 2006-04-07
DK1291351T3 (da) 2005-10-24
TR199901127T2 (xx) 1999-07-21
HRP20060275A2 (en) 2007-10-31
CZ300106B6 (cs) 2009-02-11
KR20000068435A (ko) 2000-11-25
US6147197A (en) 2000-11-14
JP4597274B2 (ja) 2010-12-15
CN1680420A (zh) 2005-10-12
US6075133A (en) 2000-06-13
HUP9902869A2 (hu) 2000-02-28
EP0929563B1 (en) 2005-06-01
SK28699A3 (en) 2000-03-13
IL128681A0 (en) 2000-01-31
CN1273475C (zh) 2006-09-06
BG63547B1 (bg) 2002-04-30
KR20050044816A (ko) 2005-05-12
DK1291352T3 (da) 2005-09-19
CN100460415C (zh) 2009-02-11
HRP20060277A2 (en) 2007-10-31
CA2263972A1 (en) 1998-03-12
DE69733422D1 (de) 2005-07-07
EP1291351A1 (en) 2003-03-12
DE69733422T2 (de) 2006-05-04
CZ68599A3 (cs) 1999-08-11
CN1680418A (zh) 2005-10-12
DE69733370T2 (de) 2006-02-02
EP1291351B1 (en) 2005-07-13
KR100576988B1 (ko) 2006-05-10
HRP970473A2 (en) 1998-08-31
SK285533B6 (sk) 2007-03-01
JP2001500855A (ja) 2001-01-23
ATE299508T1 (de) 2005-07-15
AU729348B2 (en) 2001-02-01
ATE296832T1 (de) 2005-06-15
PT1291350E (pt) 2005-09-30
ATE296308T1 (de) 2005-06-15
ATE296307T1 (de) 2005-06-15
EP1291353B1 (en) 2005-06-01
HRP970473B1 (en) 2007-02-28
KR100523679B1 (ko) 2005-10-26
DE69733439D1 (de) 2005-07-07
NZ334274A (en) 2001-02-23
USRE39591E1 (en) 2007-04-24
DE69733370D1 (de) 2005-06-30
PT1291353E (pt) 2005-10-31
PL188173B1 (pl) 2004-12-31
DE69733723D1 (de) 2005-08-18
EP1291352B1 (en) 2005-05-25
CN1680419A (zh) 2005-10-12
SK285536B6 (sk) 2007-03-01
EP0929563A1 (en) 1999-07-21
EP1291350A1 (en) 2003-03-12
EP1291350B1 (en) 2005-05-25
SK285534B6 (sk) 2007-03-01
EP1291353A1 (en) 2003-03-12
KR20050043994A (ko) 2005-05-11
BR9711661A (pt) 1999-08-24
HU230166B1 (hu) 2015-09-28
ES2242812T3 (es) 2005-11-16
NO314230B1 (no) 2003-02-17
ES2242813T3 (es) 2005-11-16
ID19406A (id) 1998-07-09
ES2244716T3 (es) 2005-12-16
KR20050044815A (ko) 2005-05-12
WO1998009978A1 (en) 1998-03-12
CA2263972C (en) 2008-01-29
NO991022D0 (no) 1999-03-02
ES2242811T3 (es) 2005-11-16
CN1237183A (zh) 1999-12-01
PT1291351E (pt) 2005-11-30
DK1291353T3 (da) 2005-10-03
SI20023A (sl) 2000-02-29
US6028181A (en) 2000-02-22
HRP20060278A2 (en) 2007-10-31
SI20023B (en) 2001-02-28
AU4178097A (en) 1998-03-26
DE69733439T2 (de) 2006-05-04
BG103292A (en) 1999-12-30

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