NO318203B1 - Imidazopyridinderivater som inhiberer magesyresekresjon - Google Patents

Imidazopyridinderivater som inhiberer magesyresekresjon Download PDF

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Publication number
NO318203B1
NO318203B1 NO20005451A NO20005451A NO318203B1 NO 318203 B1 NO318203 B1 NO 318203B1 NO 20005451 A NO20005451 A NO 20005451A NO 20005451 A NO20005451 A NO 20005451A NO 318203 B1 NO318203 B1 NO 318203B1
Authority
NO
Norway
Prior art keywords
compound
formula
alkyl
ethyl
methylbenzylamino
Prior art date
Application number
NO20005451A
Other languages
English (en)
Norwegian (no)
Other versions
NO20005451L (no
NO20005451D0 (no
Inventor
Ingemar Starke
Kosrat Amin
Mikael Dahlstrom
Peter Nordberg
Original Assignee
Astrazeneca Ab Global Ip
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab Global Ip filed Critical Astrazeneca Ab Global Ip
Publication of NO20005451D0 publication Critical patent/NO20005451D0/no
Publication of NO20005451L publication Critical patent/NO20005451L/no
Publication of NO318203B1 publication Critical patent/NO318203B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO20005451A 1998-04-29 2000-10-27 Imidazopyridinderivater som inhiberer magesyresekresjon NO318203B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE9801526A SE9801526D0 (sv) 1998-04-29 1998-04-29 New compounds
PCT/SE1999/000662 WO1999055705A1 (en) 1998-04-29 1999-04-23 Imidazo pyridine derivatives which inhibit gastric acid secretion

Publications (3)

Publication Number Publication Date
NO20005451D0 NO20005451D0 (no) 2000-10-27
NO20005451L NO20005451L (no) 2000-12-27
NO318203B1 true NO318203B1 (no) 2005-02-14

Family

ID=20411154

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20005450A NO317262B1 (no) 1998-04-29 2000-10-27 Imidazopyridinderivater som inhiberer magesyresekresjon, farmasoytisk formulering som inneholder slike derivater, fremgangsmate for deres fremstilling, anvendelse derav, og mellomprodukter.
NO20005451A NO318203B1 (no) 1998-04-29 2000-10-27 Imidazopyridinderivater som inhiberer magesyresekresjon

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO20005450A NO317262B1 (no) 1998-04-29 2000-10-27 Imidazopyridinderivater som inhiberer magesyresekresjon, farmasoytisk formulering som inneholder slike derivater, fremgangsmate for deres fremstilling, anvendelse derav, og mellomprodukter.

Country Status (33)

Country Link
US (2) US6313137B1 (cs)
EP (4) EP1491543B1 (cs)
JP (2) JP3692034B2 (cs)
KR (3) KR100595805B1 (cs)
CN (2) CN1174980C (cs)
AR (2) AR015769A1 (cs)
AT (4) ATE372340T1 (cs)
AU (2) AU769108B2 (cs)
BR (2) BR9909996B1 (cs)
CA (2) CA2329922C (cs)
CZ (2) CZ293977B6 (cs)
DE (4) DE69928792T2 (cs)
DK (2) DK1073657T3 (cs)
EE (2) EE04676B1 (cs)
ES (2) ES2252975T3 (cs)
HU (2) HUP0102313A3 (cs)
ID (2) ID26819A (cs)
IL (4) IL139200A0 (cs)
IS (2) IS5683A (cs)
MY (2) MY121379A (cs)
NO (2) NO317262B1 (cs)
NZ (2) NZ507639A (cs)
PL (2) PL195000B1 (cs)
RU (2) RU2238271C2 (cs)
SA (2) SA99200065B1 (cs)
SE (1) SE9801526D0 (cs)
SI (1) SI1073656T1 (cs)
SK (2) SK14912000A3 (cs)
TR (4) TR200003149T2 (cs)
TW (2) TW490466B (cs)
UA (2) UA66846C2 (cs)
WO (2) WO1999055706A1 (cs)
ZA (2) ZA200005797B (cs)

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US6489346B1 (en) 1996-01-04 2002-12-03 The Curators Of The University Of Missouri Substituted benzimidazole dosage forms and method of using same
US5840737A (en) 1996-01-04 1998-11-24 The Curators Of The University Of Missouri Omeprazole solution and method for using same
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US6900324B2 (en) 2000-09-07 2005-05-31 Astrazeneca Ab Process for preparing a substituted imidazopyridine compound
SE0003186D0 (sv) 2000-09-07 2000-09-07 Astrazeneca Ab New process
UA80393C2 (uk) 2000-12-07 2007-09-25 Алтана Фарма Аг Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці
SE0100295D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
SE0100297D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
SE0100296D0 (sv) * 2001-02-01 2001-02-01 Astrazeneca Ab New compounds
AU2002228579B2 (en) * 2001-02-13 2006-07-27 Astrazeneca Ab Novel modified released formulation
WO2002069968A1 (en) * 2001-03-08 2002-09-12 Astrazeneca Ab New use
SE0102808D0 (sv) * 2001-08-22 2001-08-22 Astrazeneca Ab New compounds
MY140561A (en) * 2002-02-20 2009-12-31 Nycomed Gmbh Dosage form containing pde 4 inhibitor as active ingredient
SE0201940D0 (sv) * 2002-06-20 2002-06-20 Astrazeneca Ab New combination II
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MXPA05005117A (es) 2002-11-19 2005-07-01 Altana Pharma Ag Imidazopiridinas 8-sustituidas.
AR043002A1 (es) * 2003-02-18 2005-07-13 Altana Pharma Ag Imidazopirazinas 6-substituidos
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SE525349C2 (sv) * 2003-06-23 2005-02-08 Volvo Penta Ab Utombordsdrev för båtar
SE0301903D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound III with therapeutic effect
SE0301904D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound II with therapeutic effect
SE0301905D0 (sv) * 2003-06-26 2003-06-26 Astrazeneca Ab Novel imidazopyridine compound I with therapeutic effect
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EP1974730A1 (en) 2003-11-03 2008-10-01 AstraZeneca AB Imidazo[1,2-a]pyridine derivatives for use in the treatment of sleep disturbance due to silent gastro-esophageal reflux
SE0303451D0 (sv) * 2003-12-18 2003-12-18 Astrazeneca Ab New compounds
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ES2421916T3 (es) 2005-03-16 2013-09-06 Nycomed Gmbh Forma farmacéutica de sabor enmascarado que contiene roflumilast
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KR101777971B1 (ko) * 2016-07-05 2017-09-12 제일약품주식회사 이미다조[1,2-a]피리딘 유도체, 이의 제조방법 및 이의 용도
KR20190057569A (ko) * 2017-11-20 2019-05-29 제일약품주식회사 7-아미노-1h-인돌-5-카르복사미드 유도체 및 이의 용도
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Also Published As

Publication number Publication date
IS5684A (is) 2000-10-25
EP1491542A3 (en) 2005-01-05
ID27530A (id) 2001-04-12
EP1491543A1 (en) 2004-12-29
DE69937076T2 (de) 2008-05-29
US6313136B1 (en) 2001-11-06
CN1165535C (zh) 2004-09-08
UA66846C2 (uk) 2004-06-15
RU2238271C2 (ru) 2004-10-20
SA99200065B1 (ar) 2006-11-07
IS5683A (is) 2000-10-25
SK14912000A3 (sk) 2001-06-11
KR20010043133A (ko) 2001-05-25
EE04916B1 (et) 2007-10-15
HUP0102425A2 (hu) 2001-11-28
DK1073657T3 (da) 2006-03-13
JP3692034B2 (ja) 2005-09-07
SA99200064B1 (ar) 2006-10-11
CA2329922A1 (en) 1999-11-04
UA67769C2 (uk) 2004-07-15
PL195000B1 (pl) 2007-07-31
KR100595805B1 (ko) 2006-07-03
SA99200065A (ar) 2005-12-03
DE69927803T2 (de) 2006-07-06
CN1174980C (zh) 2004-11-10
ATE372339T1 (de) 2007-09-15
NZ507639A (en) 2004-01-30
CN1307577A (zh) 2001-08-08
ZA200005797B (en) 2002-01-18
JP2002513025A (ja) 2002-05-08
JP2002513024A (ja) 2002-05-08
BR9909996B1 (pt) 2010-08-24
CZ292567B6 (cs) 2003-10-15
EP1073657B1 (en) 2005-12-07
EP1491542A2 (en) 2004-12-29
IL139200A0 (en) 2001-11-25
CA2329921A1 (en) 1999-11-04
HUP0102313A3 (en) 2002-10-28
BR9909995B1 (pt) 2010-07-13
WO1999055706A9 (en) 2000-03-16
DE69937077T2 (de) 2008-05-29
KR100595806B1 (ko) 2006-07-03
DE69937076D1 (de) 2007-10-18
TR200003176T2 (tr) 2001-03-21
HK1071139A1 (en) 2005-07-08
IL139200A (en) 2010-04-29
BR9909996A (pt) 2000-12-26
NO20005450D0 (no) 2000-10-27
KR100650472B1 (ko) 2006-11-28
HUP0102425A3 (en) 2002-12-28
IL139297A0 (en) 2001-11-25
MY121379A (en) 2006-01-28
DK1073656T3 (da) 2006-01-16
US6313137B1 (en) 2001-11-06
DE69937077D1 (de) 2007-10-18
EE200000626A (et) 2002-04-15
WO1999055705A1 (en) 1999-11-04
TR200003149T2 (tr) 2001-03-21
NZ507638A (en) 2003-10-31
JP3883383B2 (ja) 2007-02-21
DE69928792D1 (de) 2006-01-12
HK1036981A1 (en) 2002-01-25
EP1073656A1 (en) 2001-02-07
SE9801526D0 (sv) 1998-04-29
EP1073657A1 (en) 2001-02-07
PL343801A1 (en) 2001-09-10
ATE307130T1 (de) 2005-11-15
EE04676B1 (et) 2006-08-15
CZ293977B6 (cs) 2004-09-15
EE200000664A (et) 2002-04-15
EP1491542B1 (en) 2007-09-05
CZ20003982A3 (cs) 2001-02-14
ES2249913T3 (es) 2006-04-01
EP1073656B1 (en) 2005-10-19
HK1036984A1 (en) 2002-01-25
ATE312101T1 (de) 2005-12-15
EP1491543B1 (en) 2007-09-05
DE69927803D1 (de) 2006-03-02
HUP0102313A2 (hu) 2001-12-28
AU769190B2 (en) 2004-01-22
SK285768B6 (sk) 2007-07-06
SI1073656T1 (sl) 2006-02-28
WO1999055706A1 (en) 1999-11-04
TW490466B (en) 2002-06-11
CN1306533A (zh) 2001-08-01
TR200102728T2 (tr) 2002-06-21
MY121389A (en) 2006-01-28
ATE372340T1 (de) 2007-09-15
AU4300699A (en) 1999-11-16
NO20005451L (no) 2000-12-27
AR015769A1 (es) 2001-05-16
NO20005451D0 (no) 2000-10-27
SK14922000A3 (sk) 2001-06-11
KR20010043134A (ko) 2001-05-25
KR20050121760A (ko) 2005-12-27
AU4300799A (en) 1999-11-16
HK1033317A1 (en) 2001-08-24
IL139297A (en) 2007-06-03
TR200102612T2 (tr) 2002-06-21
NO317262B1 (no) 2004-09-27
CZ20003981A3 (cs) 2001-03-14
PL343797A1 (en) 2001-09-10
BR9909995A (pt) 2000-12-26
TWI250159B (en) 2006-03-01
ES2252975T3 (es) 2006-05-16
RU2235725C2 (ru) 2004-09-10
NO20005450L (no) 2000-12-22
AU769108B2 (en) 2004-01-15
CA2329922C (en) 2006-04-11
ID26819A (id) 2001-02-15
AR015768A1 (es) 2001-05-16
HK1033457A1 (en) 2001-08-31
ZA200005796B (en) 2002-01-18
DE69928792T2 (de) 2006-07-20

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