KR20200083676A - 골수 섬유증을 치료하기 위한 조성물 및 방법 - Google Patents

골수 섬유증을 치료하기 위한 조성물 및 방법 Download PDF

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KR20200083676A
KR20200083676A KR1020207019018A KR20207019018A KR20200083676A KR 20200083676 A KR20200083676 A KR 20200083676A KR 1020207019018 A KR1020207019018 A KR 1020207019018A KR 20207019018 A KR20207019018 A KR 20207019018A KR 20200083676 A KR20200083676 A KR 20200083676A
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compound
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capsule
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Korean (ko)
Inventor
아빈드 자얀
제니스 카카스
아얄루 테페리
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임팩트 바이오메디신스, 인코포레이티드
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46024747&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR20200083676(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 임팩트 바이오메디신스, 인코포레이티드 filed Critical 임팩트 바이오메디신스, 인코포레이티드
Priority to KR1020247006181A priority Critical patent/KR20240029118A/ko
Publication of KR20200083676A publication Critical patent/KR20200083676A/ko
Ceased legal-status Critical Current

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4858—Organic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841—Filling excipients; Inactive ingredients
    • A61K9/4866—Organic macromolecular compounds

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
KR1020207019018A 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법 Ceased KR20200083676A (ko)

Priority Applications (1)

Application Number Priority Date Filing Date Title
KR1020247006181A KR20240029118A (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US41092410P 2010-11-07 2010-11-07
US61/410,924 2010-11-07
PCT/US2011/059643 WO2012061833A1 (en) 2010-11-07 2011-11-07 Compositions and methods for treating myelofibrosis

Related Parent Applications (1)

Application Number Title Priority Date Filing Date
KR1020187031287A Division KR102131241B1 (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020247006181A Division KR20240029118A (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법

Publications (1)

Publication Number Publication Date
KR20200083676A true KR20200083676A (ko) 2020-07-08

Family

ID=46024747

Family Applications (4)

Application Number Title Priority Date Filing Date
KR1020207019018A Ceased KR20200083676A (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법
KR1020247006181A Pending KR20240029118A (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법
KR1020137014479A Active KR101940979B1 (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법
KR1020187031287A Active KR102131241B1 (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법

Family Applications After (3)

Application Number Title Priority Date Filing Date
KR1020247006181A Pending KR20240029118A (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법
KR1020137014479A Active KR101940979B1 (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법
KR1020187031287A Active KR102131241B1 (ko) 2010-11-07 2011-11-07 골수 섬유증을 치료하기 위한 조성물 및 방법

Country Status (36)

Country Link
US (5) US10391094B2 (enExample)
EP (2) EP2635282B1 (enExample)
JP (1) JP6133211B2 (enExample)
KR (4) KR20200083676A (enExample)
CN (2) CN108125923A (enExample)
AU (2) AU2010363329A1 (enExample)
BR (1) BR112013011184A2 (enExample)
CA (2) CA2816957A1 (enExample)
CL (1) CL2013001252A1 (enExample)
CO (1) CO6801724A2 (enExample)
DK (1) DK2635282T3 (enExample)
DO (1) DOP2013000097A (enExample)
EC (1) ECSP13012658A (enExample)
ES (1) ES2930650T3 (enExample)
HR (1) HRP20221269T1 (enExample)
HU (1) HUE060254T2 (enExample)
IL (1) IL226101A (enExample)
LT (1) LT2635282T (enExample)
MA (1) MA34723B1 (enExample)
MX (2) MX360246B (enExample)
MY (1) MY161164A (enExample)
NI (1) NI201300038A (enExample)
NZ (1) NZ611363A (enExample)
PE (1) PE20140389A1 (enExample)
PH (1) PH12013500924A1 (enExample)
PL (1) PL2635282T3 (enExample)
PT (1) PT2635282T (enExample)
RS (1) RS63996B1 (enExample)
RU (1) RU2616262C2 (enExample)
SG (1) SG190134A1 (enExample)
SI (1) SI2635282T1 (enExample)
SM (1) SMT202200453T1 (enExample)
TW (1) TWI531389B (enExample)
UA (1) UA114076C2 (enExample)
WO (2) WO2012060847A1 (enExample)
ZA (1) ZA201303423B (enExample)

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WO2012060847A1 (en) 2010-11-07 2012-05-10 Targegen, Inc. Compositions and methods for treating myelofibrosis
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CN104771761A (zh) * 2015-03-19 2015-07-15 深圳国源国药有限公司 一种创新药用辅料硅化微晶纤维素及其制备方法
EP3327441B1 (en) * 2015-07-24 2021-02-17 Public University Corporation Nagoya City University Method for assisting diagnosis of conditions of myelofibrosis, method for monitoring therapeutic effect, and a device therefor
CN105919955A (zh) * 2016-06-13 2016-09-07 佛山市腾瑞医药科技有限公司 一种鲁索利替尼制剂及其应用
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WO2019140953A1 (zh) * 2018-01-16 2019-07-25 深圳市塔吉瑞生物医药有限公司 用于抑制激酶活性的二苯氨基嘧啶类化合物
US20220031699A1 (en) 2018-09-25 2022-02-03 Impact Biomedicines, Inc. Methods of treating myeloproliferative disorders
SG11202102982QA (en) * 2018-09-25 2021-04-29 Impact Biomedicines Inc Methods of treating myeloproliferative disorders
JP2022519885A (ja) * 2019-02-12 2022-03-25 インパクト バイオメディシンズ インコーポレイテッド Ｊａｋ２阻害剤の結晶形態
FR3092581A1 (fr) * 2019-02-12 2020-08-14 Impact Biomedicines, Inc Formes cristallines d'un inhibiteur de jak2
KR20220088699A (ko) 2019-09-27 2022-06-28 디스크 메디슨, 인크. 골수섬유증 및 관련 상태의 치료 방법
US11306062B2 (en) 2019-10-29 2022-04-19 Johnson Matthey Public Limited Forms of fedratinib dihydrochloride
CN114845702B (zh) * 2019-12-20 2024-03-15 英特维特国际股份有限公司 一种吡唑药物组合物
WO2021207051A1 (en) * 2020-04-06 2021-10-14 Bristol-Myers Squibb Company Methods of treating acute respiratory disorders
KR20230012539A (ko) 2020-05-13 2023-01-26 디스크 메디슨, 인크. 골수섬유증을 치료하기 위한 항-헤모주벨린 (hjv) 항체
CN116829136A (zh) 2020-12-16 2023-09-29 生物医学影响公司 菲卓替尼的给药
EP4297750A1 (en) 2021-02-25 2024-01-03 Impact Biomedicines, Inc. Use of a bet inhibitor alone or in combination with fedratinib or ruxolitinib for treating a hematological malignancy such as myelofibrosis
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