KR100398944B1 - 보론산에스테르및보론산화합물,이의합성방법및용도 - Google Patents

보론산에스테르및보론산화합물,이의합성방법및용도 Download PDF

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KR100398944B1
KR100398944B1 KR1019970702789A KR19970702789A KR100398944B1 KR 100398944 B1 KR100398944 B1 KR 100398944B1 KR 1019970702789 A KR1019970702789 A KR 1019970702789A KR 19970702789 A KR19970702789 A KR 19970702789A KR 100398944 B1 KR100398944 B1 KR 100398944B1
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aryl
compound
formula
aralkyl
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KR970706824A (ko
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줄리안 아담스
유팅 마
로스 스테인
매튜 베브스키
루이스 그레니어
루이스 플라몬돈
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밀레니엄 파머슈티컬스 인코퍼레이티드
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    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
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  • AIDS & HIV (AREA)
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  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pyridine Compounds (AREA)
KR1019970702789A 1994-10-28 1995-10-27 보론산에스테르및보론산화합물,이의합성방법및용도 Expired - Lifetime KR100398944B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US33052594A 1994-10-28 1994-10-28
US08/330526 1994-10-28
US08/442,581 US6083903A (en) 1994-10-28 1995-05-16 Boronic ester and acid compounds, synthesis and uses
US08/442581 1995-05-16

Publications (2)

Publication Number Publication Date
KR970706824A KR970706824A (ko) 1997-12-01
KR100398944B1 true KR100398944B1 (ko) 2004-06-04

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ID=26987313

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KR1019970702789A Expired - Lifetime KR100398944B1 (ko) 1994-10-28 1995-10-27 보론산에스테르및보론산화합물,이의합성방법및용도

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US (16) US6083903A (enExample)
EP (4) EP1997823A1 (enExample)
JP (1) JP3717934B2 (enExample)
KR (1) KR100398944B1 (enExample)
CN (2) CN101077875B (enExample)
AT (3) ATE411324T1 (enExample)
AU (1) AU710564B2 (enExample)
CA (2) CA2496538C (enExample)
CH (1) CH0788360H1 (enExample)
CY (1) CY2484B1 (enExample)
DE (5) DE122004000025I2 (enExample)
DK (3) DK0788360T5 (enExample)
ES (3) ES2314540T3 (enExample)
FI (2) FI114801B (enExample)
FR (1) FR04C0014I2 (enExample)
IL (5) IL133831A (enExample)
LU (1) LU91083I2 (enExample)
MX (1) MX9703063A (enExample)
NL (1) NL300151I2 (enExample)
NO (2) NO310558B1 (enExample)
NZ (2) NZ337211A (enExample)
PT (3) PT1627880E (enExample)
TW (1) TW318850B (enExample)
WO (1) WO1996013266A1 (enExample)

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NO2004004I2 (no) 2007-09-10
NZ296717A (en) 1999-11-29
KR970706824A (ko) 1997-12-01
CA2203936A1 (en) 1996-05-09
DE122004000025I2 (de) 2006-09-07
CA2496538C (en) 2011-08-02
FR04C0014I2 (enExample) 2005-05-21
CA2203936C (en) 2005-04-12
EP0788360A4 (en) 1998-05-06
CH0788360H1 (de) 2006-03-15
FI120974B (fi) 2010-05-31
CN1305475C (zh) 2007-03-21
US6617317B1 (en) 2003-09-09
US5780454A (en) 1998-07-14
NO971929D0 (no) 1997-04-25
US6066730A (en) 2000-05-23
US7119080B2 (en) 2006-10-10
WO1996013266A1 (en) 1996-05-09
US20080132678A1 (en) 2008-06-05
DK0788360T5 (da) 2017-09-18
ATE241631T1 (de) 2003-06-15
US20150072942A1 (en) 2015-03-12
US20070282100A1 (en) 2007-12-06
IL115790A0 (en) 1996-01-19
CN1168633A (zh) 1997-12-24
US20130310320A1 (en) 2013-11-21
LU91083I2 (fr) 2004-08-09
ES2314540T3 (es) 2009-03-16
JPH10510245A (ja) 1998-10-06
CN101077875A (zh) 2007-11-28
CN101077875B (zh) 2011-01-26
AU710564C (en) 1996-05-23
EP0788360A1 (en) 1997-08-13
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