JPS6135986B2 - - Google Patents

Info

Publication number
JPS6135986B2
JPS6135986B2 JP52001997A JP199777A JPS6135986B2 JP S6135986 B2 JPS6135986 B2 JP S6135986B2 JP 52001997 A JP52001997 A JP 52001997A JP 199777 A JP199777 A JP 199777A JP S6135986 B2 JPS6135986 B2 JP S6135986B2
Authority
JP
Japan
Prior art keywords
group
formula
dimethylaminopropyl
acid
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP52001997A
Other languages
English (en)
Japanese (ja)
Other versions
JPS52105162A (en
Inventor
Peetaa Baagesa Kurausu
Sutausubaaru Tofuto Andaasu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
H Lundbeck AS
Original Assignee
Kefalas AS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=9722860&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JPS6135986(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Kefalas AS filed Critical Kefalas AS
Publication of JPS52105162A publication Critical patent/JPS52105162A/ja
Publication of JPS6135986B2 publication Critical patent/JPS6135986B2/ja
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP199777A 1976-01-14 1977-01-13 Phthleic derivatives and preparation thereof Granted JPS52105162A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB1486/76A GB1526331A (en) 1976-01-14 1976-01-14 Phthalanes

Publications (2)

Publication Number Publication Date
JPS52105162A JPS52105162A (en) 1977-09-03
JPS6135986B2 true JPS6135986B2 (https=) 1986-08-15

Family

ID=9722860

Family Applications (1)

Application Number Title Priority Date Filing Date
JP199777A Granted JPS52105162A (en) 1976-01-14 1977-01-13 Phthleic derivatives and preparation thereof

Country Status (19)

Country Link
US (1) US4136193A (https=)
JP (1) JPS52105162A (https=)
AT (1) AT359488B (https=)
AU (1) AU509445B2 (https=)
BE (1) BE850401A (https=)
CA (1) CA1094087A (https=)
CH (3) CH626886A5 (https=)
DE (1) DE2657013C2 (https=)
DK (1) DK143275C (https=)
ES (1) ES454980A1 (https=)
FI (1) FI63754C (https=)
FR (1) FR2338271A1 (https=)
GB (1) GB1526331A (https=)
IE (1) IE44055B1 (https=)
NL (2) NL192451C (https=)
NO (2) NO147243C (https=)
NZ (1) NZ183001A (https=)
SE (1) SE429551B (https=)
ZA (1) ZA7757B (https=)

Families Citing this family (162)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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GB8419963D0 (en) * 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) * 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
DK0759299T3 (da) * 1995-08-16 2000-08-07 Lilly Co Eli Potensering af serotoninrespons
ES2148120T3 (es) 1997-07-08 2002-01-16 Lundbeck & Co As H Metodo para la preparacion de citalopram.
UA62985C2 (en) * 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
EA002770B1 (ru) 1997-11-11 2002-08-29 Х.Лундбекк А/С Способ получения циталопрама
PL199423B1 (pl) 1998-10-20 2008-09-30 Lundbeck & Co As H Sposób wytwarzania citalopramu
KR20010081071A (ko) 1998-12-08 2001-08-25 피터슨 존 메이달 벤조푸란 유도체, 그것들의 제조 및 사용
AR021509A1 (es) * 1998-12-08 2002-07-24 Lundbeck & Co As H Derivados de benzofurano, su preparacion y uso
IL143422A0 (en) 1998-12-23 2002-04-21 Lundbeck & Co As H Method for the preparation of 5-cyanophthalide
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
DK1173431T4 (da) * 1999-04-14 2010-01-04 Lundbeck & Co As H Fremgangsmåde til fremstilling af citalopram
ITMI991581A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991486A1 (it) * 1999-07-06 2001-01-06 Vis Farmaceutici S P A Processo per la sintesi di citalopram
AR021155A1 (es) * 1999-07-08 2002-06-12 Lundbeck & Co As H Tratamiento de desordenes neuroticos
HRP20020344B1 (hr) 1999-10-25 2010-10-31 H. Lundbeck A/S Način priprave citaloprama
GB2360281B (en) 1999-10-25 2002-01-16 Lundbeck & Co As H Method for the preparation of citalopram
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AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
HUP0203635A3 (en) 1999-12-28 2005-02-28 Lundbeck & Co As H Method for the preparation of citalopram
PT1246813E (pt) * 1999-12-30 2004-02-27 Lundbeck & Co As H Metodo para a preparacao de citalopram
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IES20010143A2 (en) * 2000-02-24 2001-07-25 Lundbeck & Co As H Method for the preparation of citalopram
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KR100821912B1 (ko) * 2000-05-12 2008-04-16 하. 룬트벡 아크티에 셀스카브 시탈로프람의 제조 방법
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CA2383963A1 (en) * 2000-07-06 2002-01-17 Eva Bolzonella Method for the preparation of citalopram
AU8174001A (en) * 2000-07-21 2002-02-05 Lundbeck & Co As H Novel compounds and their use as glycine transport inhibitors
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US20030232881A1 (en) * 2000-10-27 2003-12-18 H. Lundbeck A/S Crystals of pharmaceutically acceptable salts of citalopram, methods of crystallization, and pharmaceutical compositions comprising them
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BE850401A (fr) 1977-07-14
DE2657013A1 (de) 1977-07-28
DK143275B (da) 1981-08-03
NO1996001I1 (no) 1996-01-05
CA1094087A (en) 1981-01-20
NL7700244A (nl) 1977-07-18
NO770109L (no) 1977-07-15
SE7614201L (sv) 1977-07-15
CH632259A5 (de) 1982-09-30
AU2107377A (en) 1978-07-13
FR2338271B1 (https=) 1982-11-05
SE429551B (sv) 1983-09-12
NL970031I2 (nl) 1997-10-01
AT359488B (de) 1980-11-10
NL192451C (nl) 1997-08-04
FI770073A7 (https=) 1977-07-15
IE44055B1 (en) 1981-07-29
US4136193A (en) 1979-01-23
NL192451B (nl) 1997-04-01
NL970031I1 (nl) 1997-10-01
DK143275C (da) 1982-01-18
GB1526331A (en) 1978-09-27
DK13177A (da) 1977-07-15
FI63754B (fi) 1983-04-29
AU509445B2 (en) 1980-05-15
FI63754C (fi) 1983-08-10
ATA947276A (de) 1980-04-15
FR2338271A1 (fr) 1977-08-12
NO147243C (no) 1983-03-02
DE2657013C2 (de) 1985-11-14
NZ183001A (en) 1978-06-02
JPS52105162A (en) 1977-09-03
CH626886A5 (https=) 1981-12-15
ZA7757B (en) 1977-11-30
IE44055L (en) 1977-07-14
ES454980A1 (es) 1978-04-01
CH632258A5 (de) 1982-09-30

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