JP5918693B2 - Egfr阻害剤及び疾患の治療方法 - Google Patents

Egfr阻害剤及び疾患の治療方法 Download PDF

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JP5918693B2
JP5918693B2 JP2012509790A JP2012509790A JP5918693B2 JP 5918693 B2 JP5918693 B2 JP 5918693B2 JP 2012509790 A JP2012509790 A JP 2012509790A JP 2012509790 A JP2012509790 A JP 2012509790A JP 5918693 B2 JP5918693 B2 JP 5918693B2
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egfr
cancer
heterocycle
aryl
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JP2012526113A (ja
JP2012526113A5 (OSRAM
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エス. グレイ ナサニエル
エス. グレイ ナサニエル
ジャンネ パシ
ジャンネ パシ
ジェイ. エック マイケル
ジェイ. エック マイケル
チョウ ウェンジュン
チョウ ウェンジュン
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ダナ ファーバー キャンサー インスティテュート インコーポレイテッド
ダナ ファーバー キャンサー インスティテュート インコーポレイテッド
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
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    • C07D473/00Heterocyclic compounds containing purine ring systems
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    • C07D473/16Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two nitrogen atoms
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JP2012509790A 2009-05-05 2010-05-05 Egfr阻害剤及び疾患の治療方法 Active JP5918693B2 (ja)

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Application Number Priority Date Filing Date Title
US21541909P 2009-05-05 2009-05-05
US61/215,419 2009-05-05
PCT/US2010/001341 WO2010129053A2 (en) 2009-05-05 2010-05-05 Egfr inhibitors and methods of treating disorders

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JP2012526113A JP2012526113A (ja) 2012-10-25
JP2012526113A5 JP2012526113A5 (OSRAM) 2013-06-27
JP5918693B2 true JP5918693B2 (ja) 2016-05-18

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US (2) US9908884B2 (OSRAM)
EP (1) EP2440559B1 (OSRAM)
JP (1) JP5918693B2 (OSRAM)
KR (1) KR101705158B1 (OSRAM)
CN (1) CN102482277B (OSRAM)
CA (1) CA2760794C (OSRAM)
ES (1) ES2659725T3 (OSRAM)
IL (1) IL216140B (OSRAM)
WO (1) WO2010129053A2 (OSRAM)

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US9908884B2 (en) 2018-03-06
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US20190040065A1 (en) 2019-02-07
CA2760794C (en) 2017-07-25
US20120094999A1 (en) 2012-04-19
KR101705158B1 (ko) 2017-02-09
EP2440559A2 (en) 2012-04-18
EP2440559B1 (en) 2018-01-10
KR20120047208A (ko) 2012-05-11
IL216140A0 (en) 2012-01-31
IL216140B (en) 2018-03-29
CN102482277A (zh) 2012-05-30
EP2440559A4 (en) 2012-11-21
WO2010129053A8 (en) 2011-12-15
WO2010129053A2 (en) 2010-11-11
CA2760794A1 (en) 2010-11-11
JP2012526113A (ja) 2012-10-25
CN102482277B (zh) 2017-09-19

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