JP4860474B2 - Pdgfrによって仲介される病気のためのジアリール尿素 - Google Patents
Pdgfrによって仲介される病気のためのジアリール尿素 Download PDFInfo
- Publication number
- JP4860474B2 JP4860474B2 JP2006533210A JP2006533210A JP4860474B2 JP 4860474 B2 JP4860474 B2 JP 4860474B2 JP 2006533210 A JP2006533210 A JP 2006533210A JP 2006533210 A JP2006533210 A JP 2006533210A JP 4860474 B2 JP4860474 B2 JP 4860474B2
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- Prior art keywords
- acid
- phenyl
- urea
- pyridyloxy
- trifluoromethyl
- Prior art date
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61L—METHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
- A61L2300/00—Biologically active materials used in bandages, wound dressings, absorbent pads or medical devices
- A61L2300/40—Biologically active materials used in bandages, wound dressings, absorbent pads or medical devices characterised by a specific therapeutic activity or mode of action
- A61L2300/416—Anti-neoplastic or anti-proliferative or anti-restenosis or anti-angiogenic agents, e.g. paclitaxel, sirolimus
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Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47173503P | 2003-05-20 | 2003-05-20 | |
| US60/471,735 | 2003-05-20 | ||
| US52039903P | 2003-11-17 | 2003-11-17 | |
| US60/520,399 | 2003-11-17 | ||
| US55606204P | 2004-03-25 | 2004-03-25 | |
| US60/556,062 | 2004-03-25 | ||
| PCT/US2004/015653 WO2005000284A2 (en) | 2003-05-20 | 2004-05-19 | Diaryl ureas for diseases mediated by pdgfr |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006528986A JP2006528986A (ja) | 2006-12-28 |
| JP2006528986A5 JP2006528986A5 (https=) | 2011-09-08 |
| JP4860474B2 true JP4860474B2 (ja) | 2012-01-25 |
Family
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
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| JP2006533210A Expired - Lifetime JP4860474B2 (ja) | 2003-05-20 | 2004-05-19 | Pdgfrによって仲介される病気のためのジアリール尿素 |
| JP2006533211A Pending JP2007511203A (ja) | 2003-05-20 | 2004-05-19 | キナーゼ阻害活性を有するジアリール尿素 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006533211A Pending JP2007511203A (ja) | 2003-05-20 | 2004-05-19 | キナーゼ阻害活性を有するジアリール尿素 |
Country Status (12)
| Country | Link |
|---|---|
| US (2) | US8796250B2 (https=) |
| EP (2) | EP1636585B2 (https=) |
| JP (2) | JP4860474B2 (https=) |
| AT (2) | ATE384264T1 (https=) |
| CA (2) | CA2526636C (https=) |
| DE (2) | DE602004007382T2 (https=) |
| DK (2) | DK1636585T3 (https=) |
| ES (2) | ES2305808T3 (https=) |
| MX (1) | MXPA05012486A (https=) |
| PL (2) | PL1626714T3 (https=) |
| PT (2) | PT1626714E (https=) |
| WO (2) | WO2004113274A2 (https=) |
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Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2000042012A1 (en) * | 1999-01-13 | 2000-07-20 | Bayer Corporation | φ-CARBOXYARYL SUBSTITUTED DIPHENYL UREAS AS RAF KINASE INHIBITORS |
| JP2006519264A (ja) * | 2003-02-28 | 2006-08-24 | バイエル、ファーマシューテイカルズ、コーポレイション | 癌および他の障害の処置に有用な新規シアノピリジン誘導体 |
| JP2006519265A (ja) * | 2003-02-28 | 2006-08-24 | バイエル ファーマシューティカルス コーポレーション | 癌その他の疾患の治療に有用な新規な二環尿素誘導体 |
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