JP2020503247A5 - - Google Patents

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JP2020503247A5
JP2020503247A5 JP2019519216A JP2019519216A JP2020503247A5 JP 2020503247 A5 JP2020503247 A5 JP 2020503247A5 JP 2019519216 A JP2019519216 A JP 2019519216A JP 2019519216 A JP2019519216 A JP 2019519216A JP 2020503247 A5 JP2020503247 A5 JP 2020503247A5
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JP2019519216A 2016-10-10 2017-10-10 Retキナーゼ阻害剤としての置換ピラゾロ[1,5−a]ピリジン化合物 Active JP6776446B2 (ja)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
US201662406252P 2016-10-10 2016-10-10
US62/406,252 2016-10-10
US201762447850P 2017-01-18 2017-01-18
US62/447,850 2017-01-18
US201762491164P 2017-04-27 2017-04-27
US62/491,164 2017-04-27
US201762554817P 2017-09-06 2017-09-06
US62/554,817 2017-09-06
US201762566093P 2017-09-29 2017-09-29
US62/566,093 2017-09-29
PCT/US2017/055983 WO2018071447A1 (en) 2016-10-10 2017-10-10 Substituted pyrazolo[1,5-a]pyridine compounds as ret kinase inhibitors

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JP2020503247A JP2020503247A (ja) 2020-01-30
JP2020503247A5 true JP2020503247A5 (enExample) 2020-07-09
JP6776446B2 JP6776446B2 (ja) 2020-10-28

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JP2019519216A Active JP6776446B2 (ja) 2016-10-10 2017-10-10 Retキナーゼ阻害剤としての置換ピラゾロ[1,5−a]ピリジン化合物
JP2020168202A Active JP7079303B2 (ja) 2016-10-10 2020-10-05 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2022015288A Active JP7311654B2 (ja) 2016-10-10 2022-02-03 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2022082682A Active JP7502365B2 (ja) 2016-10-10 2022-05-20 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2023111484A Active JP7634606B2 (ja) 2016-10-10 2023-07-06 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2024179747A Active JP7761732B2 (ja) 2016-10-10 2024-10-15 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物

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JP2020168202A Active JP7079303B2 (ja) 2016-10-10 2020-10-05 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2022015288A Active JP7311654B2 (ja) 2016-10-10 2022-02-03 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2022082682A Active JP7502365B2 (ja) 2016-10-10 2022-05-20 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2023111484A Active JP7634606B2 (ja) 2016-10-10 2023-07-06 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物
JP2024179747A Active JP7761732B2 (ja) 2016-10-10 2024-10-15 Retキナーゼ阻害剤としての置換ピラゾロ[1,5-a]ピリジン化合物

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US (8) US10112942B2 (enExample)
EP (2) EP3523301B1 (enExample)
JP (6) JP6776446B2 (enExample)
KR (1) KR102143899B1 (enExample)
CN (2) CN114163437B (enExample)
AU (1) AU2017342022B2 (enExample)
BR (1) BR112019007144B8 (enExample)
CA (1) CA3039760C (enExample)
CL (1) CL2019000941A1 (enExample)
CO (1) CO2019004650A2 (enExample)
CR (1) CR20190218A (enExample)
CY (1) CY1123201T1 (enExample)
DK (1) DK3523301T3 (enExample)
DO (1) DOP2019000090A (enExample)
EC (1) ECSP19032676A (enExample)
ES (1) ES2805087T3 (enExample)
HR (1) HRP20201008T1 (enExample)
HU (1) HUE051424T2 (enExample)
IL (2) IL265916B (enExample)
JO (1) JOP20190076B1 (enExample)
LT (1) LT3523301T (enExample)
MA (1) MA53675A (enExample)
MD (1) MD3523301T2 (enExample)
MX (2) MX376465B (enExample)
MY (1) MY195573A (enExample)
NZ (1) NZ752793A (enExample)
PE (1) PE20190918A1 (enExample)
PH (1) PH12019500775A1 (enExample)
PL (1) PL3523301T3 (enExample)
PT (1) PT3523301T (enExample)
RS (1) RS60536B1 (enExample)
SA (1) SA519401541B1 (enExample)
SG (1) SG11201903144PA (enExample)
SI (1) SI3523301T1 (enExample)
TN (1) TN2019000110A1 (enExample)
TW (1) TWI704148B (enExample)
UA (1) UA125030C2 (enExample)
WO (1) WO2018071447A1 (enExample)
ZA (1) ZA202004040B (enExample)

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