HU229928B1 - Szulfonamid- és szulfamid-helyettesített imidazokinolinok - Google Patents

Szulfonamid- és szulfamid-helyettesített imidazokinolinok Download PDF

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Publication number
HU229928B1
HU229928B1 HU0201431A HUP0201431A HU229928B1 HU 229928 B1 HU229928 B1 HU 229928B1 HU 0201431 A HU0201431 A HU 0201431A HU P0201431 A HUP0201431 A HU P0201431A HU 229928 B1 HU229928 B1 HU 229928B1
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HU
Hungary
Prior art keywords
alkyl
substituted
aryl
heteroaryl
butyl
Prior art date
Application number
HU0201431A
Other languages
English (en)
Hungarian (hu)
Inventor
Stephen L Crooks
Kyle J Lindstrom
Bryon A Merrill
Michael J Rice
Original Assignee
3M Innovative Properties Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 3M Innovative Properties Co filed Critical 3M Innovative Properties Co
Publication of HUP0201431A2 publication Critical patent/HUP0201431A2/hu
Publication of HUP0201431A3 publication Critical patent/HUP0201431A3/hu
Publication of HU229928B1 publication Critical patent/HU229928B1/hu

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0063—Periodont
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Medicinal Preparation (AREA)
HU0201431A 1999-06-10 2000-06-08 Szulfonamid- és szulfamid-helyettesített imidazokinolinok HU229928B1 (hu)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US13836599P 1999-06-10 1999-06-10
US09/589,216 US6331539B1 (en) 1999-06-10 2000-06-07 Sulfonamide and sulfamide substituted imidazoquinolines
PCT/US2000/015722 WO2000076519A1 (en) 1999-06-10 2000-06-08 Sulfonamide and sulfamide substituted imidazoquinolines

Publications (3)

Publication Number Publication Date
HUP0201431A2 HUP0201431A2 (en) 2002-08-28
HUP0201431A3 HUP0201431A3 (en) 2002-12-28
HU229928B1 true HU229928B1 (hu) 2015-01-28

Family

ID=26836139

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0201431A HU229928B1 (hu) 1999-06-10 2000-06-08 Szulfonamid- és szulfamid-helyettesített imidazokinolinok

Country Status (28)

Country Link
US (5) US6331539B1 (enExample)
EP (1) EP1198233B1 (enExample)
JP (1) JP4833466B2 (enExample)
KR (1) KR100781428B1 (enExample)
CN (1) CN1249061C (enExample)
AT (1) ATE336249T1 (enExample)
AU (1) AU772179B2 (enExample)
BR (1) BR0011433B1 (enExample)
CA (1) CA2376305C (enExample)
CY (1) CY1108536T1 (enExample)
CZ (1) CZ303287B6 (enExample)
DE (1) DE60030126T2 (enExample)
DK (1) DK1198233T3 (enExample)
EE (1) EE05074B1 (enExample)
ES (1) ES2270840T3 (enExample)
HR (1) HRP20010890B1 (enExample)
HU (1) HU229928B1 (enExample)
IL (2) IL146486A0 (enExample)
MX (1) MXPA01012547A (enExample)
NO (1) NO320747B1 (enExample)
NZ (1) NZ515967A (enExample)
PL (1) PL211009B1 (enExample)
PT (1) PT1198233E (enExample)
RU (1) RU2248975C2 (enExample)
SK (1) SK286418B6 (enExample)
TR (1) TR200103575T2 (enExample)
UA (1) UA73503C2 (enExample)
WO (1) WO2000076519A1 (enExample)

Families Citing this family (254)

* Cited by examiner, † Cited by third party
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