HRP20090665A2 - 8-[3-amino-piperidin-1-il]-ksantini, njihovo dobivanje i upotreba kao lijekova - Google Patents
8-[3-amino-piperidin-1-il]-ksantini, njihovo dobivanje i upotreba kao lijekova Download PDFInfo
- Publication number
- HRP20090665A2 HRP20090665A2 HR20090665A HRP20090665A HRP20090665A2 HR P20090665 A2 HRP20090665 A2 HR P20090665A2 HR 20090665 A HR20090665 A HR 20090665A HR P20090665 A HRP20090665 A HR P20090665A HR P20090665 A2 HRP20090665 A2 HR P20090665A2
- Authority
- HR
- Croatia
- Prior art keywords
- methyl
- xanthine
- piperidin
- amino
- group
- Prior art date
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
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- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A61K9/4841—Filling excipients; Inactive ingredients
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
- C07D473/12—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1, 3, and 7, e.g. caffeine
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
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- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
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- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
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- Oncology (AREA)
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- Immunology (AREA)
- Reproductive Health (AREA)
- Pain & Pain Management (AREA)
- Virology (AREA)
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- Cardiology (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10238243A DE10238243A1 (de) | 2002-08-21 | 2002-08-21 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
| DE10312353A DE10312353A1 (de) | 2003-03-20 | 2003-03-20 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
| PCT/EP2003/009127 WO2004018468A2 (de) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-yl]-xanthine, deren herstellung und deren verwendung als arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HRP20090665A2 true HRP20090665A2 (hr) | 2010-07-31 |
Family
ID=31947613
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HR20050157 HRP20050157B1 (en) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-yl]-xanthines,the production thereof and the use of the same as medicaments |
| HR20090665A HRP20090665A2 (hr) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-il]-ksantini, njihovo dobivanje i upotreba kao lijekova |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HR20050157 HRP20050157B1 (en) | 2002-08-21 | 2003-08-18 | 8-[3-amino-piperidin-1-yl]-xanthines,the production thereof and the use of the same as medicaments |
Country Status (39)
| Country | Link |
|---|---|
| EP (6) | EP3424926A1 (cs) |
| JP (6) | JP4233524B2 (cs) |
| KR (2) | KR101150449B1 (cs) |
| CN (4) | CN100522962C (cs) |
| AR (3) | AR041025A1 (cs) |
| AT (1) | ATE453644T1 (cs) |
| AU (2) | AU2003253418B2 (cs) |
| BE (1) | BE2011C038I2 (cs) |
| BR (2) | BRPI0313648B8 (cs) |
| CA (1) | CA2496249C (cs) |
| CY (3) | CY1109928T1 (cs) |
| DE (2) | DE50312295D1 (cs) |
| DK (1) | DK1532149T3 (cs) |
| EA (3) | EA016166B1 (cs) |
| EC (2) | ECSP055617A (cs) |
| EG (1) | EG25011A (cs) |
| ES (1) | ES2339112T3 (cs) |
| FR (1) | FR11C0052I2 (cs) |
| HK (1) | HK1250708A1 (cs) |
| HR (2) | HRP20050157B1 (cs) |
| HU (1) | HUS1100028I1 (cs) |
| IL (1) | IL166964A (cs) |
| IN (2) | IN2015DN01132A (cs) |
| LT (1) | LTC1532149I2 (cs) |
| LU (2) | LU91889I2 (cs) |
| ME (1) | MEP59708A (cs) |
| MX (1) | MXPA05001684A (cs) |
| MY (2) | MY137619A (cs) |
| NO (4) | NO333970B1 (cs) |
| PE (1) | PE20040897A1 (cs) |
| PL (2) | PL403104A1 (cs) |
| PT (1) | PT1532149E (cs) |
| RS (2) | RS52142B (cs) |
| SA (1) | SA03240448B1 (cs) |
| SI (1) | SI1532149T1 (cs) |
| TW (3) | TWI319320B (cs) |
| UA (1) | UA84275C2 (cs) |
| UY (1) | UY27946A1 (cs) |
| WO (1) | WO2004018468A2 (cs) |
Families Citing this family (184)
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