HK1058047A1 - Peptides as ns3-serine protease inhibitors of hepatitis c virus - Google Patents
Peptides as ns3-serine protease inhibitors of hepatitis c virusInfo
- Publication number
- HK1058047A1 HK1058047A1 HK04100762.2A HK04100762A HK1058047A1 HK 1058047 A1 HK1058047 A1 HK 1058047A1 HK 04100762 A HK04100762 A HK 04100762A HK 1058047 A1 HK1058047 A1 HK 1058047A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- hepatitis
- peptides
- virus
- protease inhibitors
- serine protease
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
- C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0802—Tripeptides with the first amino acid being neutral
- C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Crystallography & Structural Chemistry (AREA)
- Gastroenterology & Hepatology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22010800P | 2000-07-21 | 2000-07-21 | |
PCT/US2001/022678 WO2002008244A2 (en) | 2000-07-21 | 2001-07-19 | Peptides as ns3-serine protease inhibitors of hepatitis c virus |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1058047A1 true HK1058047A1 (en) | 2004-04-30 |
Family
ID=22822095
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK04100762.2A HK1058047A1 (en) | 2000-07-21 | 2004-02-06 | Peptides as ns3-serine protease inhibitors of hepatitis c virus |
Country Status (32)
Country | Link |
---|---|
US (4) | US7012066B2 (es) |
EP (1) | EP1385870B1 (es) |
JP (3) | JP4298289B2 (es) |
KR (2) | KR100904788B1 (es) |
CN (3) | CN102206247B (es) |
AR (2) | AR033985A1 (es) |
AT (1) | ATE461207T1 (es) |
AU (2) | AU2001276988B2 (es) |
BR (1) | BR0112540A (es) |
CA (1) | CA2410662C (es) |
CY (2) | CY1112267T1 (es) |
CZ (1) | CZ303213B6 (es) |
DE (2) | DE60141608D1 (es) |
DK (1) | DK1385870T3 (es) |
EC (1) | ECSP034438A (es) |
ES (1) | ES2341534T3 (es) |
HK (1) | HK1058047A1 (es) |
HU (1) | HU229997B1 (es) |
IL (2) | IL153670A0 (es) |
LU (1) | LU91910I2 (es) |
MX (1) | MXPA03000627A (es) |
MY (2) | MY143322A (es) |
NO (2) | NO332329B1 (es) |
NZ (1) | NZ523782A (es) |
PL (1) | PL206255B1 (es) |
PT (1) | PT1385870E (es) |
RU (2) | RU2355700C9 (es) |
SI (1) | SI1385870T1 (es) |
SK (1) | SK288064B6 (es) |
TW (1) | TWI324611B (es) |
WO (1) | WO2002008244A2 (es) |
ZA (1) | ZA200210312B (es) |
Families Citing this family (262)
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EP1318997B1 (en) | 2000-09-15 | 2006-05-31 | Vertex Pharmaceuticals Incorporated | Pyrazole compounds useful as protein kinase inhibitors |
US6660731B2 (en) | 2000-09-15 | 2003-12-09 | Vertex Pharmaceuticals Incorporated | Pyrazole compounds useful as protein kinase inhibitors |
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CN100402549C (zh) | 2001-07-11 | 2008-07-16 | 沃泰克斯药物股份有限公司 | 桥连二环的丝氨酸蛋白酶抑制剂 |
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