BR112015025464A2 - coagonistas do receptor de glp-1/glucagon estáveis, prolongados para uso médico - Google Patents

coagonistas do receptor de glp-1/glucagon estáveis, prolongados para uso médico

Info

Publication number
BR112015025464A2
BR112015025464A2 BR112015025464A BR112015025464A BR112015025464A2 BR 112015025464 A2 BR112015025464 A2 BR 112015025464A2 BR 112015025464 A BR112015025464 A BR 112015025464A BR 112015025464 A BR112015025464 A BR 112015025464A BR 112015025464 A2 BR112015025464 A2 BR 112015025464A2
Authority
BR
Brazil
Prior art keywords
stable
glucagon receptor
medical use
glp
prolonged
Prior art date
Application number
BR112015025464A
Other languages
English (en)
Portuguese (pt)
Inventor
F Lau Jesper
Kruse Thomas
Sensfuss Ulrich
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of BR112015025464A2 publication Critical patent/BR112015025464A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/28—Insulins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
BR112015025464A 2013-04-18 2014-04-22 coagonistas do receptor de glp-1/glucagon estáveis, prolongados para uso médico BR112015025464A2 (pt)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP13164272 2013-04-18
US201361814969P 2013-04-23 2013-04-23
EP13196656 2013-12-11
PCT/EP2014/058084 WO2014170496A1 (en) 2013-04-18 2014-04-22 Stable, protracted glp-1/glucagon receptor co-agonists for medical use

Publications (1)

Publication Number Publication Date
BR112015025464A2 true BR112015025464A2 (pt) 2017-10-10

Family

ID=51730843

Family Applications (1)

Application Number Title Priority Date Filing Date
BR112015025464A BR112015025464A2 (pt) 2013-04-18 2014-04-22 coagonistas do receptor de glp-1/glucagon estáveis, prolongados para uso médico

Country Status (16)

Country Link
US (3) US9474790B2 (https=)
EP (1) EP2986313B1 (https=)
JP (1) JP6594856B2 (https=)
KR (1) KR20160021758A (https=)
CN (1) CN105307672B (https=)
AU (1) AU2014255608B2 (https=)
BR (1) BR112015025464A2 (https=)
CA (1) CA2909581A1 (https=)
MX (1) MX362275B (https=)
MY (1) MY174727A (https=)
PL (1) PL2986313T3 (https=)
RS (1) RS59124B1 (https=)
RU (1) RU2683039C2 (https=)
SI (1) SI2986313T1 (https=)
WO (1) WO2014170496A1 (https=)
ZA (1) ZA201507010B (https=)

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US20160355562A1 (en) 2016-12-08
RS59124B1 (sr) 2019-09-30
US9751927B2 (en) 2017-09-05
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MY174727A (en) 2020-05-11
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