|
US4356170A
(en)
|
1981-05-27 |
1982-10-26 |
Canadian Patents & Development Ltd. |
Immunogenic polysaccharide-protein conjugates
|
|
IL93173A0
(en)
|
1989-02-01 |
1990-11-05 |
Shionogi & Co |
Production of glucagon
|
|
US5408037A
(en)
|
1991-01-17 |
1995-04-18 |
Zymogenetics, Inc. |
Methods for detecting glucagon antagonists
|
|
US5424286A
(en)
|
1993-05-24 |
1995-06-13 |
Eng; John |
Exendin-3 and exendin-4 polypeptides, and pharmaceutical compositions comprising same
|
|
US5480867A
(en)
|
1993-12-29 |
1996-01-02 |
The Rockefeller University |
Glucagon analogs with serine replacements
|
|
US5932462A
(en)
|
1995-01-10 |
1999-08-03 |
Shearwater Polymers, Inc. |
Multiarmed, monofunctional, polymer for coupling to molecules and surfaces
|
|
US5869602A
(en)
|
1995-03-17 |
1999-02-09 |
Novo Nordisk A/S |
Peptide derivatives
|
|
IL124109A
(en)
|
1995-09-08 |
2001-10-31 |
Novo Nordisk As |
Pharmaceutical composition of 2-alkylpyrrolidines for use in the manufacture of medicaments for the treatment of diabetes
|
|
EP0876379A1
(en)
|
1996-01-17 |
1998-11-11 |
Novo Nordisk A/S |
Fused 1,2,4-thiadiazine and fused 1,4-thiazine derivatives, their preparation and use
|
|
WO1997041120A1
(en)
|
1996-07-26 |
1997-11-06 |
Dr. Reddy's Research Foundation |
Thiazolidinedione compounds having antidiabetic, hypolipidaemic, antihypertensive properties, process for their preparation and pharmaceutical compositions thereof
|
|
IL128332A0
(en)
|
1996-08-30 |
2000-01-31 |
Novo Nordisk As |
GLP-1 derivatives
|
|
RU2200161C2
(ru)
|
1996-12-31 |
2003-03-10 |
Др. Редди'З Рисерч Фаундейшн |
Новые производные азолидиндиона, способ их получения (варианты), фармацевтические композиции на их основе, способ предупреждения или лечения, способ снижения глюкозы и промежуточное соединение
|
|
JP2001518069A
(ja)
|
1997-05-02 |
2001-10-09 |
ドクター・レディーズ・リサーチ・ファウンデーション |
低脂質性、抗高血圧性特性を有する新規な抗糖尿病化合物、それらの製造方法及びそれらを含有する薬学的組成物
|
|
WO1999001423A1
(en)
|
1997-07-01 |
1999-01-14 |
Novo Nordisk A/S |
Glucagon antagonists/inverse agonists
|
|
US6613942B1
(en)
|
1997-07-01 |
2003-09-02 |
Novo Nordisk A/S |
Glucagon antagonists/inverse agonists
|
|
JP2001510195A
(ja)
|
1997-07-16 |
2001-07-31 |
ノボ ノルディスク アクティーゼルスカブ |
縮合化1,2,4−チアジアジン誘導体、その調製及び使用
|
|
WO1999019313A1
(en)
|
1997-10-27 |
1999-04-22 |
Dr. Reddy's Research Foundation |
Novel tricyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them
|
|
US6440961B1
(en)
|
1997-10-27 |
2002-08-27 |
Dr. Reddy's Research Foundation |
Tricyclic compounds and their use in medicine: process for their preparation and pharmaceutical compositions containing them
|
|
AU6966498A
(en)
|
1997-12-02 |
1998-10-30 |
Dr. Reddy's Research Foundation |
Thiazolidinedione and oxazolidinedione derivatives having antidiabetic, hypol ipidaemic and antihypertensive properties
|
|
WO2000023415A1
(en)
|
1998-10-21 |
2000-04-27 |
Novo Nordisk A/S |
New compounds, their preparation and use
|
|
JP2002527502A
(ja)
|
1998-10-21 |
2002-08-27 |
ノボ ノルディスク アクティーゼルスカブ |
新規化合物、それらの調製及び使用
|
|
EP1123269A1
(en)
|
1998-10-21 |
2001-08-16 |
Novo Nordisk A/S |
New compounds, their preparation and use
|
|
AU6190299A
(en)
|
1998-10-21 |
2000-05-08 |
Dr. Reddy's Research Foundation |
New compounds, their preparation and use
|
|
AU6325599A
(en)
|
1998-10-21 |
2000-05-08 |
Dr. Reddy's Research Foundation |
New compounds, their preparation and use
|
|
WO2000023451A1
(en)
|
1998-10-21 |
2000-04-27 |
Novo Nordisk A/S |
New compounds, their preparation and use
|
|
ES2200575T3
(es)
|
1998-12-18 |
2004-03-01 |
Novo Nordisk A/S |
Derivados de 1,2,4-tiadiazina fusionados, su preparacion y uso.
|
|
WO2000041121A1
(en)
|
1999-01-07 |
2000-07-13 |
Ccrewards.Com |
Method and arrangement for issuance and management of digital coupons and sales offers
|
|
WO2000042026A1
(en)
|
1999-01-15 |
2000-07-20 |
Novo Nordisk A/S |
Non-peptide glp-1 agonists
|
|
WO2000042023A1
(en)
|
1999-01-18 |
2000-07-20 |
Novo Nordisk A/S |
Substituted imidazoles, their preparation and use
|
|
HRP20010748A2
(en)
|
1999-04-16 |
2003-02-28 |
Reddys Lab Ltd Dr |
Novel polymorphic forms of an antidiabetic agent: process for their preparation and pharmaceutical compositions containing them
|
|
JP2002542245A
(ja)
|
1999-04-16 |
2002-12-10 |
ノボ ノルディスク アクティーゼルスカブ |
置換イミダゾール、それらの製造および使用
|
|
AU2953699A
(en)
|
1999-04-16 |
2000-11-02 |
Dr. Reddy's Research Foundation |
Novel polymorphic forms of an antidiabetic agent: process for their preparation and a pharmaceutical composition containing them
|
|
WO2000063189A1
(en)
|
1999-04-16 |
2000-10-26 |
Novo Nordisk A/S |
Crystalline r- guanidines, arginine or (l) -arginine (2s) -2- ethoxy -3-{4- [2-(10h -phenoxazin -10-yl)ethoxy]phenyl}propanoate
|
|
WO2000063196A1
(en)
|
1999-04-20 |
2000-10-26 |
Novo Nordisk A/S |
New compounds, their preparation and use
|
|
EP1171438A1
(en)
|
1999-04-20 |
2002-01-16 |
Novo Nordisk A/S |
Compounds, their preparation and use
|
|
CN1348439A
(zh)
|
1999-04-20 |
2002-05-08 |
诺沃挪第克公司 |
新化合物及其制备和用途
|
|
EP1171431A1
(en)
|
1999-04-20 |
2002-01-16 |
Novo Nordisk A/S |
Compounds, their preparation and use
|
|
AU3957600A
(en)
|
1999-04-26 |
2000-11-10 |
Boehringer Ingelheim International Gmbh |
Piperidyl-imidazole derivatives, their preparations and therapeutic uses
|
|
EP1180121B9
(en)
|
1999-05-17 |
2004-09-08 |
Conjuchem, Inc. |
Long lasting insulinotropic peptides
|
|
SI1105409T1
(sl)
|
1999-05-17 |
2006-06-30 |
Conjuchem Inc |
Zascita endogenih peptidov pred peptidazno ucinkovitostjo s konjugacijo na krvne komponente
|
|
AU6479101A
(en)
|
2000-06-16 |
2002-01-02 |
Lilly Co Eli |
Glucagon-like peptide-1 analogs
|
|
AU2001287600B2
(en)
|
2000-07-20 |
2006-07-13 |
F. Hoffmann-La Roche Ag |
Alpha-acyl and alpha-heteroatom-substituted benzene acetamide glucokinase activators
|
|
GB0121709D0
(en)
|
2001-09-07 |
2001-10-31 |
Imp College Innovations Ltd |
Food inhibition agent
|
|
US7157277B2
(en)
|
2001-11-28 |
2007-01-02 |
Neose Technologies, Inc. |
Factor VIII remodeling and glycoconjugation of Factor VIII
|
|
EP2305312B1
(en)
|
2001-10-10 |
2015-03-04 |
ratiopharm GmbH |
Remodelling and glycoconjugation of follicle-stimulating hormone (FSH)
|
|
WO2003062290A1
(en)
|
2002-01-16 |
2003-07-31 |
Biocompatibles Uk Limited |
Polymer conjugates
|
|
US6953787B2
(en)
|
2002-04-12 |
2005-10-11 |
Arena Pharmaceuticals, Inc. |
5HT2C receptor modulators
|
|
WO2004060387A1
(en)
|
2002-12-27 |
2004-07-22 |
Diobex, Inc. |
Compositions and methods for the prevention and control of insulin-induced hypoglycemia
|
|
GB0300571D0
(en)
|
2003-01-10 |
2003-02-12 |
Imp College Innovations Ltd |
Modification of feeding behaviour
|
|
EP1503283A1
(en)
|
2003-08-01 |
2005-02-02 |
Hewlett-Packard Development Company, L.P. |
Data processing system and method
|
|
KR101159559B1
(ko)
|
2003-08-05 |
2012-06-26 |
노보 노르디스크 에이/에스 |
신규의 인슐린 유도체
|
|
KR101113726B1
(ko)
|
2003-08-12 |
2012-02-27 |
리폭센 테크놀로지즈 리미티드 |
단백질 유도 및 컨쥬게이션용 시알산 유도체
|
|
CN101380476A
(zh)
|
2003-09-19 |
2009-03-11 |
诺沃挪第克公司 |
治疗肽的清蛋白结合型衍生物
|
|
CA2539253A1
(en)
|
2003-09-19 |
2005-03-31 |
Novo Nordisk A/S |
Albumin-binding derivatives of therapeutic peptides
|
|
RU2401276C2
(ru)
|
2003-09-19 |
2010-10-10 |
Ново Нордиск А/С |
Производные глюкагон-подобного пептида-1 (glp-1)
|
|
US7632921B2
(en)
|
2004-11-12 |
2009-12-15 |
Bayer Healthcare Llc |
Site-directed modification of FVIII
|
|
EP1853634B1
(en)
|
2005-02-23 |
2016-08-10 |
Lipoxen Technologies Limited |
Activated sialic acid derivatives for protein derivatisation and conjugation
|
|
EP1863537A2
(en)
|
2005-03-18 |
2007-12-12 |
Novo Nordisk A/S |
Dimeric peptide agonists of the glp-1 receptor
|
|
TWI372629B
(en)
*
|
2005-03-18 |
2012-09-21 |
Novo Nordisk As |
Acylated glp-1 compounds
|
|
WO2006103298A2
(en)
|
2005-04-01 |
2006-10-05 |
Novo Nordisk Health Care Ag |
Blood coagulation fviii analogues
|
|
DK1891105T3
(da)
|
2005-06-13 |
2012-07-16 |
Imp Innovations Ltd |
Hidtil ukendte forbindelser og deres påvirkninger på spiseadfærd
|
|
US20100197573A1
(en)
|
2005-06-15 |
2010-08-05 |
Novo Nordisk Health Care Ag |
Transglutaminase Mediated Conjugation of Growth Hormone
|
|
US20070105755A1
(en)
|
2005-10-26 |
2007-05-10 |
Neose Technologies, Inc. |
One pot desialylation and glycopegylation of therapeutic peptides
|
|
US8338368B2
(en)
|
2005-11-07 |
2012-12-25 |
Indiana University Research And Technology Corporation |
Glucagon analogs exhibiting physiological solubility and stability
|
|
EP1981977B1
(en)
|
2006-01-31 |
2015-12-23 |
National Research Council Of Canada |
Production of polysialic acid containing glyconjugates using a self-priming polysialyltransferase
|
|
WO2007100535A2
(en)
|
2006-02-22 |
2007-09-07 |
Merck & Co., Inc. |
Oxyntomodulin derivatives
|
|
US7645860B2
(en)
|
2006-03-31 |
2010-01-12 |
Baxter Healthcare S.A. |
Factor VIII polymer conjugates
|
|
EP2010222A1
(en)
|
2006-03-31 |
2009-01-07 |
Baxter International Inc. |
Pegylated factor viii
|
|
US9187532B2
(en)
|
2006-07-21 |
2015-11-17 |
Novo Nordisk A/S |
Glycosylation of peptides via O-linked glycosylation sequences
|
|
TWI428346B
(zh)
|
2006-12-13 |
2014-03-01 |
Imp Innovations Ltd |
新穎化合物及其等對進食行為影響
|
|
PT2101821E
(pt)
|
2006-12-15 |
2014-10-03 |
Baxter Int |
Fator conjugado viia-ácido (poli)siálico com prolongamento do tempo de meia vida in vivo
|
|
WO2008086086A2
(en)
|
2007-01-05 |
2008-07-17 |
Indiana University Research And Technology Corporation |
Glucagon analogs exhibiting enhanced solubility in physiological ph buffers
|
|
JP6017754B2
(ja)
|
2007-02-15 |
2016-11-02 |
インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションIndiana University Research And Technology Corporation |
グルカゴン/glp−1受容体コアゴニスト
|
|
CN101778937A
(zh)
|
2007-06-04 |
2010-07-14 |
诺和诺德公司 |
使用n-乙酰葡糖胺转移酶的o-联糖基化
|
|
DK2158214T3
(da)
|
2007-06-15 |
2011-12-05 |
Zealand Pharma As |
Glukagonanaloger
|
|
JP5356373B2
(ja)
|
2007-06-15 |
2013-12-04 |
ナショナル リサーチ カウンシル オブ カナダ |
酵素特性を向上させたポリシアリルトランスフェラーゼの操作されたバージョン
|
|
ES2672770T3
(es)
*
|
2007-09-05 |
2018-06-18 |
Novo Nordisk A/S |
Derivados del péptido-1 similar al glucagón y su uso farmacéutico
|
|
US20100261637A1
(en)
|
2007-09-05 |
2010-10-14 |
Novo Nordisk A/S |
Peptides derivatized with a-b-c-d- and their therapeutical use
|
|
WO2009033769A2
(en)
*
|
2007-09-11 |
2009-03-19 |
Mondobiotech Laboratories Ag |
Use of cortistatin 14 and others as a therapeutic agent
|
|
AU2008323768A1
(en)
|
2007-11-09 |
2009-05-14 |
Baxter Healthcare S.A. |
Modified recombinant Factor VIII and von Willebrand Factor and methods of use
|
|
US20100317057A1
(en)
|
2007-12-28 |
2010-12-16 |
Novo Nordisk A/S |
Semi-recombinant preparation of glp-1 analogues
|
|
WO2009089396A2
(en)
|
2008-01-08 |
2009-07-16 |
Neose Technologies, Inc. |
Glycoconjugation of polypeptides using oligosaccharyltransferases
|
|
EP2249853A4
(en)
|
2008-01-30 |
2012-12-26 |
Univ Indiana Res & Tech Corp |
ESTER BASED PEPTIDE PRODRUGS
|
|
CN103497247A
(zh)
|
2008-02-27 |
2014-01-08 |
诺沃—诺迪斯克有限公司 |
缀合的因子viii分子
|
|
JP5753779B2
(ja)
*
|
2008-06-17 |
2015-07-22 |
インディアナ ユニバーシティー リサーチ アンド テクノロジー コーポレーションIndiana University Research And Technology Corporation |
生理学的pHの緩衝液中で向上した溶解性及び安定性を示すグルカゴン類縁体
|
|
BRPI0915282A2
(pt)
|
2008-06-17 |
2017-02-07 |
Univ Indiana Res & Tech Corp |
agonistas mistos baseados no gip para o tratamento de distúrbios metabólicos e obesidade
|
|
AU2009260302B2
(en)
|
2008-06-17 |
2014-10-23 |
Indiana University Research And Technology Corporation |
Glucagon/GLP-1 receptor co-agonists
|
|
EP2328922A4
(en)
*
|
2008-08-07 |
2013-01-02 |
Ipsen Pharma Sas |
ANALOGUE OF GLUCOSE-DEPENDING INSULINOTROPIC POLYPEPTIDE
|
|
PT2349342T
(pt)
|
2008-10-17 |
2018-10-26 |
Baxalta Inc |
Factores sanguíneos modificados que compreendem um baixo grau de polímero solúvel na água
|
|
WO2010070252A1
(en)
|
2008-12-15 |
2010-06-24 |
Zealand Pharma A/S |
Glucagon analogues
|
|
NZ593813A
(en)
*
|
2008-12-15 |
2013-02-22 |
Zealand Pharma As |
Glucagon analogues
|
|
JP5635531B2
(ja)
|
2008-12-15 |
2014-12-03 |
ジーランド ファーマ アクティーゼルスカブ |
グルカゴン類似体
|
|
JP5635529B2
(ja)
|
2008-12-15 |
2014-12-03 |
ジーランド ファーマ アクティーゼルスカブ |
グルカゴン類似体
|
|
JP2012518029A
(ja)
|
2009-02-19 |
2012-08-09 |
ノヴォ・ノルディスク・アー/エス |
第viii因子の修飾
|
|
US9150632B2
(en)
|
2009-06-16 |
2015-10-06 |
Indiana University Research And Technology Corporation |
GIP receptor-active glucagon compounds
|
|
ME02220B
(me)
|
2009-07-13 |
2016-02-20 |
Zealand Pharma As |
Analozi acilovanog glukagona
|
|
GB0917072D0
(en)
|
2009-09-29 |
2009-11-11 |
Univ Ulster |
Peptide analogues of glucagon for diabetes therapy
|
|
WO2011075393A2
(en)
|
2009-12-18 |
2011-06-23 |
Indiana University Research And Technology Corporation |
Glucagon/glp-1 receptor co-agonists
|
|
JP2013517307A
(ja)
|
2010-01-20 |
2013-05-16 |
ジーランド ファーマ アクティーゼルスカブ |
心臓病の処置
|
|
WO2011117417A1
(en)
|
2010-03-26 |
2011-09-29 |
Novo Nordisk A/S |
Novel glucagon analogues
|
|
AR080592A1
(es)
*
|
2010-03-26 |
2012-04-18 |
Lilly Co Eli |
Peptido con actividad para el gip-r y glp-1-r, formulacion famaceutica que lo comprende, su uso para preparar un medicamento util para el tratamiento de diabetes mellitus y para inducir la perdida de peso
|
|
US20130143798A1
(en)
|
2010-03-26 |
2013-06-06 |
Novo Nordisk A/S |
Novel glucagon analogues
|
|
AR081975A1
(es)
|
2010-06-23 |
2012-10-31 |
Zealand Pharma As |
Analogos de glucagon
|
|
EP2585482B1
(en)
|
2010-06-24 |
2019-03-27 |
Zealand Pharma A/S |
Glucagon analogues
|
|
WO2011163473A1
(en)
|
2010-06-25 |
2011-12-29 |
Indiana University Research And Technology Corporation |
Glucagon analogs exhibiting enhanced solubility and stability in physiological ph buffers
|
|
CA2821766A1
(en)
*
|
2010-12-22 |
2012-06-28 |
Indiana University Research And Technology Corporation |
Glucagon analogs exhibiting gip receptor activity
|
|
SG191252A1
(en)
*
|
2010-12-22 |
2013-07-31 |
Marcadia Biotech Inc |
Methods for treating metabolic disorders and obesity with gip and glp-1 receptor-active glucagon-based peptides
|
|
MA34913B1
(fr)
|
2011-01-20 |
2014-02-01 |
Zealand Pharma As |
Combinaison d'analogues du glucagon acylé à des analogues d'insuline
|
|
KR20140020292A
(ko)
|
2011-03-28 |
2014-02-18 |
노보 노르디스크 에이/에스 |
신규 글루카곤 유사체
|
|
DK2694095T3
(en)
|
2011-04-05 |
2018-05-28 |
Longevity Biotech Inc |
COMPOSITIONS COMPREHENSIVE GLUCAGON ANALOGS AND METHODS FOR PREPARING AND USING THE SAME
|
|
WO2012150503A2
(en)
|
2011-05-03 |
2012-11-08 |
Zealand Pharma A/S |
Glu-glp-1 dual agonist signaling-selective compounds
|
|
KR102512178B1
(ko)
|
2011-05-18 |
2023-03-20 |
메더리스 다이어비티즈, 엘엘씨 |
개선된 펩티드 제약
|
|
EP2710031B9
(en)
|
2011-05-18 |
2018-02-28 |
Mederis Diabetes, LLC |
Improved peptide pharmaceuticals for insulin resistance
|
|
HRP20181591T1
(hr)
|
2011-06-10 |
2018-11-30 |
Hanmi Science Co., Ltd. |
Novi derivati oksintomodulina i farmaceutski pripravci za liječenje pretilosti koji ih sadrže
|
|
EA031230B1
(ru)
|
2011-06-22 |
2018-12-28 |
Индиана Юниверсити Рисерч Энд Текнолоджи Корпорейшн |
Агонисты глюкагонового рецептора/glp-1-рецептора
|
|
BR112013032717A2
(pt)
*
|
2011-06-22 |
2017-01-24 |
Univ Indiana Res & Tech Corp |
coagonistas do receptor de glucagon/glp-1
|
|
JP6352806B2
(ja)
*
|
2011-09-23 |
2018-07-04 |
ノヴォ ノルディスク アー/エス |
新規のグルカゴン類似体
|
|
PL2986313T3
(pl)
|
2013-04-18 |
2019-12-31 |
Novo Nordisk A/S |
Stabilni, dłużej działający współagoniści receptora glp-1/glukagonu do zastosowań medycznych
|
|
EP3080149A1
(en)
*
|
2013-12-13 |
2016-10-19 |
Sanofi |
Dual glp-1/glucagon receptor agonists
|