MX362275B - Co-agonista de peptido similar a glucagon tipo 1 (glp-1) receptor de glucagon de larga duracion, estables para uso medico. - Google Patents

Co-agonista de peptido similar a glucagon tipo 1 (glp-1) receptor de glucagon de larga duracion, estables para uso medico.

Info

Publication number
MX362275B
MX362275B MX2015014408A MX2015014408A MX362275B MX 362275 B MX362275 B MX 362275B MX 2015014408 A MX2015014408 A MX 2015014408A MX 2015014408 A MX2015014408 A MX 2015014408A MX 362275 B MX362275 B MX 362275B
Authority
MX
Mexico
Prior art keywords
agonists
stable
glucagon receptor
medical use
protracted glp
Prior art date
Application number
MX2015014408A
Other languages
English (en)
Other versions
MX2015014408A (es
Inventor
F Lau Jesper
Kruse Thomas
Sensfuss Ulrich
Original Assignee
Novo Nordisk As
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novo Nordisk As filed Critical Novo Nordisk As
Publication of MX2015014408A publication Critical patent/MX2015014408A/es
Publication of MX362275B publication Critical patent/MX362275B/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/28—Insulins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biophysics (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)

Abstract

La presente invención se refiere a co-agonistas novedosos de GLP-1 estable y de larga duración/receptor de glucagón, con el uso de estos péptidos en tratamiento, con métodos de tratamiento que comprenden la administración de los péptidos a los pacientes y con el uso de los péptidos en la elaboración de medicamentos.
MX2015014408A 2013-04-18 2014-04-22 Co-agonista de peptido similar a glucagon tipo 1 (glp-1) receptor de glucagon de larga duracion, estables para uso medico. MX362275B (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP13164272 2013-04-18
US201361814969P 2013-04-23 2013-04-23
EP13196656 2013-12-11
PCT/EP2014/058084 WO2014170496A1 (en) 2013-04-18 2014-04-22 Stable, protracted glp-1/glucagon receptor co-agonists for medical use

Publications (2)

Publication Number Publication Date
MX2015014408A MX2015014408A (es) 2017-07-28
MX362275B true MX362275B (es) 2019-01-10

Family

ID=51730843

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2015014408A MX362275B (es) 2013-04-18 2014-04-22 Co-agonista de peptido similar a glucagon tipo 1 (glp-1) receptor de glucagon de larga duracion, estables para uso medico.

Country Status (16)

Country Link
US (3) US9474790B2 (es)
EP (1) EP2986313B1 (es)
JP (1) JP6594856B2 (es)
KR (1) KR20160021758A (es)
CN (1) CN105307672B (es)
AU (1) AU2014255608B2 (es)
BR (1) BR112015025464A2 (es)
CA (1) CA2909581A1 (es)
MX (1) MX362275B (es)
MY (1) MY174727A (es)
PL (1) PL2986313T3 (es)
RS (1) RS59124B1 (es)
RU (1) RU2683039C2 (es)
SI (1) SI2986313T1 (es)
WO (1) WO2014170496A1 (es)
ZA (1) ZA201507010B (es)

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MX2015014408A (es) 2017-07-28
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