BR0116032A - imidazoquinolinas substituìdas com sulfonamido éster - Google Patents

imidazoquinolinas substituìdas com sulfonamido éster

Info

Publication number
BR0116032A
BR0116032A BRPI0116032-0A BR0116032A BR0116032A BR 0116032 A BR0116032 A BR 0116032A BR 0116032 A BR0116032 A BR 0116032A BR 0116032 A BR0116032 A BR 0116032A
Authority
BR
Brazil
Prior art keywords
sulfonamido
ester substituted
useful
substituted imidazoquinolines
diseases
Prior art date
Application number
BRPI0116032-0A
Other languages
English (en)
Inventor
Stephen L Crooks
George W Greisgraber
Philip D Heppner
Bryon A Merrill
Ralph R Roberts
Al-Ping Wei
Original Assignee
3M Innovative Properties Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 3M Innovative Properties Co filed Critical 3M Innovative Properties Co
Publication of BR0116032A publication Critical patent/BR0116032A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
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    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
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    • A61P31/22—Antivirals for DNA viruses for herpes viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
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    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/08—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis for Pneumocystis carinii
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P37/02—Immunomodulators
    • A61P37/04—Immunostimulants
    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/02—Immunomodulators
    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

"IMIDAZOQUINOLINAS SUBSTITUìDAS COM SULFONAMIDO éSTER". Compostos de imidazopiridina que contêm funcionalidade amina substituída na posição 1 são úteis como modificadores da resposta imune. Os compostos e composições da invenção podem induzir à biossíntese de várias citocinas e são úteis no tratamento de uma variedade de condições, incluindo doenças virais e doenças meoplásticas.
BRPI0116032-0A 2000-12-08 2001-12-06 imidazoquinolinas substituìdas com sulfonamido éster BR0116032A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US25421800P 2000-12-08 2000-12-08
PCT/US2001/046582 WO2002046190A2 (en) 2000-12-08 2001-12-06 Sulfonamido ether substituted imidazoquinolines

Publications (1)

Publication Number Publication Date
BR0116032A true BR0116032A (pt) 2006-02-21

Family

ID=22963391

Family Applications (6)

Application Number Title Priority Date Filing Date
BR0116470-8A BR0116470A (pt) 2000-12-08 2001-12-06 éteres de imidazoquinolina substituìdos com uréia
BRPI0116464-3A BR0116464A (pt) 2000-12-08 2001-12-06 imidazoquinolinas substituìdas com amido éter
BR0116026-5A BR0116026A (pt) 2000-12-08 2001-12-06 Imidazoquinolinas substituìdas por tioéter
BR0116047-8A BR0116047A (pt) 2000-12-08 2001-12-06 Imidazoquinolinas substituìdas de éter heterocìclico
BRPI0116032-0A BR0116032A (pt) 2000-12-08 2001-12-06 imidazoquinolinas substituìdas com sulfonamido éster
BRPI0116052-4A BR0116052A (pt) 2000-12-08 2001-12-06 imidazoquinolinas substituìdas por éter arìlico

Family Applications Before (4)

Application Number Title Priority Date Filing Date
BR0116470-8A BR0116470A (pt) 2000-12-08 2001-12-06 éteres de imidazoquinolina substituìdos com uréia
BRPI0116464-3A BR0116464A (pt) 2000-12-08 2001-12-06 imidazoquinolinas substituìdas com amido éter
BR0116026-5A BR0116026A (pt) 2000-12-08 2001-12-06 Imidazoquinolinas substituìdas por tioéter
BR0116047-8A BR0116047A (pt) 2000-12-08 2001-12-06 Imidazoquinolinas substituìdas de éter heterocìclico

Family Applications After (1)

Application Number Title Priority Date Filing Date
BRPI0116052-4A BR0116052A (pt) 2000-12-08 2001-12-06 imidazoquinolinas substituìdas por éter arìlico

Country Status (32)

Country Link
US (8) US6670372B2 (pt)
EP (6) EP1343784B1 (pt)
JP (7) JP2004515501A (pt)
KR (6) KR20040047733A (pt)
CN (6) CN1247575C (pt)
AR (6) AR035669A1 (pt)
AT (3) ATE296301T1 (pt)
AU (12) AU2002232482B2 (pt)
BR (6) BR0116470A (pt)
CA (6) CA2430844A1 (pt)
CY (2) CY1105586T1 (pt)
CZ (6) CZ20031562A3 (pt)
DE (3) DE60126645T2 (pt)
DK (3) DK1341791T3 (pt)
EE (6) EE200300271A (pt)
ES (3) ES2260323T3 (pt)
HK (3) HK1064383A1 (pt)
HR (6) HRP20030466A2 (pt)
HU (6) HUP0400710A2 (pt)
IL (6) IL155950A0 (pt)
MX (6) MXPA03005012A (pt)
NO (6) NO20032449D0 (pt)
NZ (6) NZ526106A (pt)
PL (7) PL392462A1 (pt)
PT (2) PT1341790E (pt)
RU (6) RU2315049C2 (pt)
SI (1) SI1341790T1 (pt)
SK (6) SK6842003A3 (pt)
TW (3) TWI222972B (pt)
UA (2) UA74852C2 (pt)
WO (6) WO2002046188A2 (pt)
ZA (6) ZA200305270B (pt)

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EP2572715A1 (en) 2002-12-30 2013-03-27 3M Innovative Properties Company Immunostimulatory Combinations
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