AU2011290126B2 - Heterocyclic compound and use thereof - Google Patents

Heterocyclic compound and use thereof Download PDF

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Publication number
AU2011290126B2
AU2011290126B2 AU2011290126A AU2011290126A AU2011290126B2 AU 2011290126 B2 AU2011290126 B2 AU 2011290126B2 AU 2011290126 A AU2011290126 A AU 2011290126A AU 2011290126 A AU2011290126 A AU 2011290126A AU 2011290126 B2 AU2011290126 B2 AU 2011290126B2
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Australia
Prior art keywords
optionally substituted
halogen atom
alkyl
group
substituted
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AU2011290126A
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AU2011290126A1 (en
Inventor
Yasutomi Asano
Eiji Honda
Toshihiro Imaeda
Masakuni Kori
Michiyo Mochizuki
Shinji Nakamura
Masashi Toyofuku
Osamu Ujikawa
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Takeda Pharmaceutical Co Ltd
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Takeda Pharmaceutical Co Ltd
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Publication of AU2011290126A1 publication Critical patent/AU2011290126A1/en
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
AU2011290126A 2010-08-10 2011-08-09 Heterocyclic compound and use thereof Active AU2011290126B2 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2010-179577 2010-08-10
JP2010179577 2010-08-10
PCT/JP2011/068497 WO2012020848A1 (en) 2010-08-10 2011-08-09 Heterocyclic compound and use thereof

Publications (2)

Publication Number Publication Date
AU2011290126A1 AU2011290126A1 (en) 2013-03-07
AU2011290126B2 true AU2011290126B2 (en) 2016-01-07

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AU2011290126A Active AU2011290126B2 (en) 2010-08-10 2011-08-09 Heterocyclic compound and use thereof

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US (11) US8575154B2 (enExample)
EP (1) EP2603513B1 (enExample)
JP (2) JP5788496B2 (enExample)
KR (1) KR101852215B1 (enExample)
CN (2) CN103180326B (enExample)
AR (1) AR082618A1 (enExample)
AU (1) AU2011290126B2 (enExample)
BR (1) BR112013002250B1 (enExample)
CA (1) CA2807460C (enExample)
CL (1) CL2013000380A1 (enExample)
CO (1) CO6680700A2 (enExample)
CR (1) CR20130066A (enExample)
CY (1) CY1123507T1 (enExample)
DK (1) DK2603513T3 (enExample)
DO (1) DOP2013000030A (enExample)
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EC (1) ECSP13012478A (enExample)
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HU (1) HUE049460T2 (enExample)
IL (1) IL224452A (enExample)
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PE (1) PE20131116A1 (enExample)
PH (1) PH12013500247A1 (enExample)
PL (1) PL2603513T3 (enExample)
PT (1) PT2603513T (enExample)
RS (1) RS60311B1 (enExample)
SG (1) SG187656A1 (enExample)
SI (1) SI2603513T1 (enExample)
TW (1) TWI504604B (enExample)
UA (1) UA111594C2 (enExample)
UY (1) UY33551A (enExample)
WO (1) WO2012020848A1 (enExample)
ZA (1) ZA201301120B (enExample)

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AU2014357342B2 (en) 2013-12-03 2019-01-17 Fmc Corporation Pyrrolidinones as herbicides
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AU2015361018B2 (en) 2014-12-08 2020-01-16 Fmc Corporation 3-oxo-3-(arylamino)propanoates, a process for their preparation, and their use in preparing pyrrolidinones
JP6956637B2 (ja) 2015-04-10 2021-11-02 エフ エム シー コーポレーションFmc Corporation 除草剤としての置換環状アミド
BR112017020094B1 (pt) 2015-04-27 2022-01-11 Fmc Corporation Composto, composições herbicidas, mistura de herbicida e método para controlar o crescimento de vegetação indesejada
CA2984307A1 (en) * 2015-04-29 2016-11-03 Janssen Pharmaceutica Nv Imidazopyrazines and pyrazolopyrimidines and their use as ampa receptor modulators
CA2983826A1 (en) * 2015-04-29 2016-11-03 Janssen Pharmaceutica Nv Azabenzimidazoles and their use as ampa receptor modulators
CA2980643C (en) 2015-05-12 2023-10-17 E I Du Pont De Nemours And Company Aryl substituted bicyclic compounds as herbicides
US10906873B2 (en) 2015-05-29 2021-02-02 Fmc Corporation Substituted cyclic amides as herbicides
CN107709310B (zh) 2015-06-02 2021-09-24 Fmc公司 取代的环酰胺及其作为除草剂的用途
RU2720994C2 (ru) 2015-07-31 2020-05-15 Е.И.Дюпон Де Немур Энд Компани Новые соединения циклического n-карбоксамида, применяемые в качестве гербицидов
HRP20191589T1 (hr) * 2015-08-06 2019-12-13 Hoffmann La Roche Postupci za pripravu derivata galnac kiseline
US20170181292A1 (en) * 2015-12-16 2017-06-22 Rohm And Haas Electronic Materials Llc Method for forming organic coating on nickel surface
CN105669731B (zh) * 2016-01-10 2017-06-30 沧州普瑞东方科技有限公司 一种4‑(4‑烷基环己氧基)苯硼酸的合成方法
EP3558962B1 (en) 2016-12-21 2023-07-12 FMC Corporation Nitrone herbicides
CN107892697B (zh) 2016-12-26 2020-11-03 郑州泰基鸿诺医药股份有限公司 一种[1,3]噻嗪-2-胺类化合物及应用,药物组合物
WO2018175231A1 (en) 2017-03-21 2018-09-27 Fmc Corporation Herbicidal mixture, composition and method
EP3599854A4 (en) 2017-03-21 2020-12-23 FMC Corporation PYRROLIDINONES AND PROCESS FOR PREPARING THEM
AR111839A1 (es) 2017-05-30 2019-08-21 Fmc Corp Lactamas 3-sustituidas herbicidas
AR111967A1 (es) 2017-05-30 2019-09-04 Fmc Corp Amidas herbicidas
EP3693368B1 (en) * 2017-10-06 2023-12-06 Takeda Pharmaceutical Company Limited Heterocyclic compound
ES2971497T3 (es) 2017-10-06 2024-06-05 Takeda Pharmaceuticals Co Compuestos heterocíclicos
PH12022550597A1 (en) 2019-09-16 2024-03-04 Takeda Pharmaceuticals Co Azole-fused pyridazin-3(2h)-one derivatives
US20230338391A1 (en) * 2020-05-15 2023-10-26 Takeda Pharmaceutical Company Limited Treatment for depression
CN113943294A (zh) * 2020-07-15 2022-01-18 成都海博为药业有限公司 一种作为btk抑制剂的化合物及其制备方法与用途
WO2025224508A1 (en) 2024-04-22 2025-10-30 Takeda Pharmaceutical Company Limited Pharmaceutical composition for treating depressive disorders

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US8778934B2 (en) 2014-07-15
US20200317692A1 (en) 2020-10-08
DOP2013000030A (es) 2013-03-15
CR20130066A (es) 2013-05-03
ES2793723T3 (es) 2020-11-16
MY165908A (en) 2018-05-18
UY33551A (es) 2012-03-30
US10654874B2 (en) 2020-05-19
TWI504604B (zh) 2015-10-21
BR112013002250A2 (pt) 2016-05-24
US20140080817A1 (en) 2014-03-20
US8575154B2 (en) 2013-11-05
HUE049460T2 (hu) 2020-09-28
JP6113789B2 (ja) 2017-04-12
CN103180326A (zh) 2013-06-26
JP2013535408A (ja) 2013-09-12
US20150353578A1 (en) 2015-12-10
US20130190291A1 (en) 2013-07-25
CN103180326B (zh) 2015-06-10
JP2016006080A (ja) 2016-01-14
CN104926837A (zh) 2015-09-23
IL224452A (en) 2017-11-30
PH12013500247A1 (en) 2013-03-11
US8916551B2 (en) 2014-12-23
DK2603513T3 (da) 2020-06-15
PE20131116A1 (es) 2013-10-24
SI2603513T1 (sl) 2020-07-31
UA111594C2 (uk) 2016-05-25
US20240360156A1 (en) 2024-10-31
LT2603513T (lt) 2020-05-25
EP2603513A1 (en) 2013-06-19
ECSP13012478A (es) 2013-04-30
PL2603513T3 (pl) 2020-07-27
ZA201301120B (en) 2014-04-30
JP5788496B2 (ja) 2015-09-30
WO2012020848A1 (en) 2012-02-16
CA2807460A1 (en) 2012-02-16
HRP20200844T1 (hr) 2020-08-21
GEP20156216B (en) 2015-01-12
CY1123507T1 (el) 2022-03-24
US9150591B2 (en) 2015-10-06
BR112013002250B1 (pt) 2020-10-27
RS60311B1 (sr) 2020-07-31
SG187656A1 (en) 2013-03-28
CO6680700A2 (es) 2013-05-31
EP2603513B1 (en) 2020-03-11
MX349470B (es) 2017-07-31
NZ607593A (en) 2015-01-30
CL2013000380A1 (es) 2013-05-31
US20150073137A1 (en) 2015-03-12
US9499568B2 (en) 2016-11-22
AR082618A1 (es) 2012-12-19
EA022078B1 (ru) 2015-10-30
KR101852215B1 (ko) 2018-04-25
US20130184266A1 (en) 2013-07-18
US20170022222A1 (en) 2017-01-26
AU2011290126A1 (en) 2013-03-07
WO2012020848A8 (en) 2012-09-27
US20190263832A1 (en) 2019-08-29
KR20130138738A (ko) 2013-12-19
EA201390222A1 (ru) 2013-08-30
US20180162875A1 (en) 2018-06-14
US20120077799A1 (en) 2012-03-29
CA2807460C (en) 2018-09-18
TW201217386A (en) 2012-05-01
PT2603513T (pt) 2020-06-08
MX2013001614A (es) 2013-07-05
US9884875B2 (en) 2018-02-06
MA34509B1 (fr) 2013-09-02
US11279713B2 (en) 2022-03-22

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