PE20131116A1 - Compuestos heterociclicos potenciadores de ampa - Google Patents
Compuestos heterociclicos potenciadores de ampaInfo
- Publication number
- PE20131116A1 PE20131116A1 PE2013000244A PE2013000244A PE20131116A1 PE 20131116 A1 PE20131116 A1 PE 20131116A1 PE 2013000244 A PE2013000244 A PE 2013000244A PE 2013000244 A PE2013000244 A PE 2013000244A PE 20131116 A1 PE20131116 A1 PE 20131116A1
- Authority
- PE
- Peru
- Prior art keywords
- thadiazine
- dihydropyride
- ring
- ampa
- enhancing
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Peptides Or Proteins (AREA)
Abstract
REFERIDA A UN COMPUESTO HETEROCICLICO DE FORMULA (I), DONDE EL ANILLO A ES UN HETEROCICLO DE 5 A 7 MIEMBROS OPCIONALMENTE SUSTITUIDO; EL ANILLO B ES UN HETEROCICLO DE 5 A 8 MIEMBROS OPCIONALMENTE SUSTITUIDO; EL ANILLO D ES CICLOALCANO C3-C7, ARENO C6-C14, DIHIDRONAFTALENO, ENTRE OTROS; W ES ALQUILENO C1-C3 O ALQUENILENO C2-C3 OPCIONALMENTE SUSTITUIDOS; L ES UN ENLACE, O, O-CH2, CO-NH, ENTRE OTROS; n ES 0, 1 O 2. SON COMPUESTOS PREFERIDOS: 2,2-DIOXIDO DE 9-(4-FENOXIFENIL)-3,4-DIHIDROPIRIDO[2,1-c][1,2,4]TIADIAZINA, 2,2-DIOXIDO DE 9-[4-(4-METILFENOXI)FENIL]-3,4-DIHIDROPIRIDO[2,1-c][1,2,4]TIADIAZINA, 2,2-DIOXIDO DE 9-[4-(CICLOHEXILOXI)FENIL]-3,4-DIHIDROPIRIDO[2,1-c][1,2,4]TIADIAZINA, ENTRE OTROS. TAMBIEN ESTA REFERIDA A UNA COMPOSICION FARMACEUTICA. DICHOS COMPUESTOS TIENEN ACCION POTENCIADORA DEL RECEPTOR DE AMPA (ACIDO ALFA-AMINO-3-HIDROXI-5-METIL-4-ISOXAZOLPROPIONICO) Y SON UTILES EN EL TRATAMIENTO DE LA DEPRESION, ESQUIZOFRENIA, ENFERMEDAD DE ALZHEIMER, TRANSTORNO DE HIPERACTIVIDAD, ENTRE OTRAS
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2010179577 | 2010-08-10 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20131116A1 true PE20131116A1 (es) | 2013-10-24 |
Family
ID=44534564
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2013000244A PE20131116A1 (es) | 2010-08-10 | 2011-08-09 | Compuestos heterociclicos potenciadores de ampa |
Country Status (38)
Country | Link |
---|---|
US (10) | US8575154B2 (es) |
EP (1) | EP2603513B1 (es) |
JP (2) | JP5788496B2 (es) |
KR (1) | KR101852215B1 (es) |
CN (2) | CN103180326B (es) |
AR (1) | AR082618A1 (es) |
AU (1) | AU2011290126B2 (es) |
BR (1) | BR112013002250B1 (es) |
CA (1) | CA2807460C (es) |
CL (1) | CL2013000380A1 (es) |
CO (1) | CO6680700A2 (es) |
CR (1) | CR20130066A (es) |
CY (1) | CY1123507T1 (es) |
DK (1) | DK2603513T3 (es) |
DO (1) | DOP2013000030A (es) |
EA (1) | EA022078B1 (es) |
EC (1) | ECSP13012478A (es) |
ES (1) | ES2793723T3 (es) |
GE (1) | GEP20156216B (es) |
HR (1) | HRP20200844T1 (es) |
HU (1) | HUE049460T2 (es) |
IL (1) | IL224452A (es) |
LT (1) | LT2603513T (es) |
MA (1) | MA34509B1 (es) |
MX (1) | MX349470B (es) |
MY (1) | MY165908A (es) |
NZ (1) | NZ607593A (es) |
PE (1) | PE20131116A1 (es) |
PL (1) | PL2603513T3 (es) |
PT (1) | PT2603513T (es) |
RS (1) | RS60311B1 (es) |
SG (1) | SG187656A1 (es) |
SI (1) | SI2603513T1 (es) |
TW (1) | TWI504604B (es) |
UA (1) | UA111594C2 (es) |
UY (1) | UY33551A (es) |
WO (1) | WO2012020848A1 (es) |
ZA (1) | ZA201301120B (es) |
Families Citing this family (31)
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DK2603513T3 (da) * | 2010-08-10 | 2020-06-15 | Takeda Pharmaceuticals Co | Heterocyklisk forbindelse og anvendelse deraf som AMPA-receptorpositiv allosterisk modulator |
EP2694472B1 (en) * | 2011-04-05 | 2020-03-11 | Takeda Pharmaceutical Company Limited | Sulfonamide derivative and use thereof |
US9493484B2 (en) | 2012-02-08 | 2016-11-15 | Takeda Pharmaceutical Company Limited | Heterocyclic compound and use thereof |
EP3008167A4 (en) * | 2013-06-13 | 2017-06-07 | VeroScience LLC | Compositions and methods for treating metabolic disorders |
PT3013813T (pt) | 2013-06-27 | 2019-06-14 | Pfizer | Compostos heteroaromáticos e a sua utilização como ligandos de d1 de dopamina |
KR102395827B1 (ko) | 2013-12-03 | 2022-05-10 | 에프엠씨 코포레이션 | 제초제로서의 피롤리디논 |
US11589583B2 (en) | 2013-12-03 | 2023-02-28 | Fmc Corporation | Pyrrolidinones herbicides |
UA125012C2 (uk) | 2014-07-02 | 2021-12-29 | ЕфЕмСі КОРПОРЕЙШН | Піперидинонові гербіциди |
KR102542215B1 (ko) | 2014-12-08 | 2023-06-12 | 에프엠씨 코포레이션 | 3-옥소-3-(아릴아미노)프로파노에이트, 이의 제조방법 및 피롤리디논 제조에 있어서 이의 용도 |
CA2978014A1 (en) | 2015-04-10 | 2016-10-13 | E I Du Pont De Nemours And Company | Substituted cyclic amides as herbicides |
US10582709B2 (en) | 2015-04-27 | 2020-03-10 | Fmc Corporation | Butyrolactones as herbicides |
MY194104A (en) * | 2015-04-29 | 2022-11-11 | Janssen Pharmaceutica Nv | Azabenzimidazoles and their use as ampa receptor modulators |
MX2017013874A (es) * | 2015-04-29 | 2018-06-22 | Janssen Pharmaceutica Nv | Imidazopirazinas y pirazolopirimidinas y su uso como moduladores del receptor de ampa. |
EP3650430A1 (en) | 2015-05-12 | 2020-05-13 | FMC Corporation | Intermediates and processes for the synthesis of herbicides |
US10906873B2 (en) | 2015-05-29 | 2021-02-02 | Fmc Corporation | Substituted cyclic amides as herbicides |
WO2016196593A1 (en) | 2015-06-02 | 2016-12-08 | E I Du Pont De Nemours And Company | Substituted cyclic amides and their use as herbicides |
WO2017023515A1 (en) | 2015-07-31 | 2017-02-09 | E. I. Du Pont De Nemours And Company | Cyclic n-carboxamide compounds useful as herbicides |
AU2016302697B2 (en) * | 2015-08-06 | 2020-10-29 | F. Hoffmann-La Roche Ag | Processes for the preparation of GalNAc acid derivatives |
TW201713774A (zh) | 2015-08-06 | 2017-04-16 | Kohjin Life Sciences Co Ltd | 含有β-菸鹼醯胺單核苷酸的酵母萃取物及其製造方法 |
US20170181292A1 (en) * | 2015-12-16 | 2017-06-22 | Rohm And Haas Electronic Materials Llc | Method for forming organic coating on nickel surface |
CN105669731B (zh) * | 2016-01-10 | 2017-06-30 | 沧州普瑞东方科技有限公司 | 一种4‑(4‑烷基环己氧基)苯硼酸的合成方法 |
CN110312712B (zh) | 2016-12-21 | 2023-06-23 | Fmc公司 | 硝酮除草剂 |
CN107892697B (zh) | 2016-12-26 | 2020-11-03 | 郑州泰基鸿诺医药股份有限公司 | 一种[1,3]噻嗪-2-胺类化合物及应用,药物组合物 |
CN110691516B (zh) | 2017-03-21 | 2022-10-28 | Fmc公司 | 吡咯烷酮及其制备方法 |
EP3599868A4 (en) | 2017-03-21 | 2020-12-02 | FMC Corporation | HERBICIDE MIXTURE, COMPOSITION AND PROCEDURE |
AR111839A1 (es) | 2017-05-30 | 2019-08-21 | Fmc Corp | Lactamas 3-sustituidas herbicidas |
AR111967A1 (es) | 2017-05-30 | 2019-09-04 | Fmc Corp | Amidas herbicidas |
US11407748B2 (en) | 2017-10-06 | 2022-08-09 | Takeda Pharmaceutical Company Limited | Substituted pyrido[1,2-a]pyrimidines and pyrazino[1,2-a]pyrimidines for enhancing AMPA receptor function |
JP7250687B2 (ja) * | 2017-10-06 | 2023-04-03 | 武田薬品工業株式会社 | 複素環化合物 |
EP4149478A1 (en) * | 2020-05-15 | 2023-03-22 | Takeda Pharmaceutical Company Limited | Treatment for depression |
CN113943294A (zh) * | 2020-07-15 | 2022-01-18 | 成都海博为药业有限公司 | 一种作为btk抑制剂的化合物及其制备方法与用途 |
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FR2801587B1 (fr) | 1999-11-30 | 2002-01-11 | Adir | Nouveaux derives de benzothiadiazines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
CA2458388A1 (en) | 2001-10-10 | 2003-04-17 | Neurosearch A/S | Novel benzothiazine derivatives, their preparation and use |
FR2833955B1 (fr) * | 2001-12-21 | 2004-01-30 | Servier Lab | Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
FR2854634B1 (fr) | 2003-05-05 | 2005-07-08 | Servier Lab | Nouveaux derives de thiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
FR2865474B1 (fr) | 2004-01-26 | 2008-06-13 | Servier Lab | Nouveaux derives de benzothiazines fluorees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
FR2879201B1 (fr) | 2004-12-10 | 2007-02-16 | Servier Lab | Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
ZA200810793B (en) | 2006-06-23 | 2010-03-31 | Nufarm Australia Ltd | Phenoxy alkanoate herbicidal composition and method of preparation and use |
CN101541741A (zh) * | 2006-12-11 | 2009-09-23 | 伊莱利利公司 | Ampa受体增强剂 |
US20080167374A1 (en) | 2007-01-09 | 2008-07-10 | Loveland Products, Inc. | Pesticide composition and method of use |
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JP2009248543A (ja) | 2008-04-11 | 2009-10-29 | Fujifilm Corp | 光情報記録媒体および情報記録方法 |
TW201012803A (en) | 2008-06-06 | 2010-04-01 | Organon Nv | Heterocyclic derivatives |
WO2010054067A1 (en) * | 2008-11-06 | 2010-05-14 | Schering Corporation | Gamma secretase modulators |
TW201030002A (en) | 2009-01-16 | 2010-08-16 | Bristol Myers Squibb Co | Bicyclic compounds for the reduction of beta-amyloid production |
JP2012051806A (ja) | 2009-02-26 | 2012-03-15 | Eisai R & D Management Co Ltd | イミダゾリルピラジン誘導体 |
FR2943342B1 (fr) | 2009-03-20 | 2011-03-04 | Servier Lab | Nouveaux derives de benzothiadiazepines,leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
WO2010140339A1 (ja) | 2009-06-01 | 2010-12-09 | 武田薬品工業株式会社 | 複素環化合物 |
WO2011007756A1 (ja) | 2009-07-13 | 2011-01-20 | 武田薬品工業株式会社 | 複素環化合物及びその用途 |
WO2011036885A1 (ja) | 2009-09-25 | 2011-03-31 | 武田薬品工業株式会社 | 複素環化合物 |
WO2011036889A1 (ja) | 2009-09-25 | 2011-03-31 | 武田薬品工業株式会社 | 複素環化合物 |
DK2603513T3 (da) * | 2010-08-10 | 2020-06-15 | Takeda Pharmaceuticals Co | Heterocyklisk forbindelse og anvendelse deraf som AMPA-receptorpositiv allosterisk modulator |
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2011
- 2011-08-09 DK DK11749944.2T patent/DK2603513T3/da active
- 2011-08-09 UY UY0001033551A patent/UY33551A/es not_active Application Discontinuation
- 2011-08-09 MX MX2013001614A patent/MX349470B/es active IP Right Grant
- 2011-08-09 LT LTEP11749944.2T patent/LT2603513T/lt unknown
- 2011-08-09 US US13/206,113 patent/US8575154B2/en active Active
- 2011-08-09 SG SG2013007463A patent/SG187656A1/en unknown
- 2011-08-09 WO PCT/JP2011/068497 patent/WO2012020848A1/en active Application Filing
- 2011-08-09 AU AU2011290126A patent/AU2011290126B2/en active Active
- 2011-08-09 EA EA201390222A patent/EA022078B1/ru not_active IP Right Cessation
- 2011-08-09 KR KR1020137006113A patent/KR101852215B1/ko active IP Right Grant
- 2011-08-09 AR ARP110102905A patent/AR082618A1/es active IP Right Grant
- 2011-08-09 PE PE2013000244A patent/PE20131116A1/es active IP Right Grant
- 2011-08-09 RS RS20200574A patent/RS60311B1/sr unknown
- 2011-08-09 CA CA2807460A patent/CA2807460C/en active Active
- 2011-08-09 JP JP2013506362A patent/JP5788496B2/ja active Active
- 2011-08-09 CN CN201180048970.3A patent/CN103180326B/zh active Active
- 2011-08-09 MY MYPI2013000428A patent/MY165908A/en unknown
- 2011-08-09 EP EP11749944.2A patent/EP2603513B1/en active Active
- 2011-08-09 TW TW100128311A patent/TWI504604B/zh active
- 2011-08-09 NZ NZ607593A patent/NZ607593A/en unknown
- 2011-08-09 PL PL11749944T patent/PL2603513T3/pl unknown
- 2011-08-09 BR BR112013002250-7A patent/BR112013002250B1/pt active IP Right Grant
- 2011-08-09 US US13/816,137 patent/US9150591B2/en active Active
- 2011-08-09 MA MA35708A patent/MA34509B1/fr unknown
- 2011-08-09 SI SI201131887T patent/SI2603513T1/sl unknown
- 2011-08-09 ES ES11749944T patent/ES2793723T3/es active Active
- 2011-08-09 GE GEAP201113021A patent/GEP20156216B/en unknown
- 2011-08-09 CN CN201510259936.0A patent/CN104926837A/zh active Pending
- 2011-08-09 PT PT117499442T patent/PT2603513T/pt unknown
- 2011-08-09 HU HUE11749944A patent/HUE049460T2/hu unknown
- 2011-09-08 UA UAA201302884A patent/UA111594C2/uk unknown
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2013
- 2013-01-28 IL IL224452A patent/IL224452A/en active IP Right Grant
- 2013-02-05 DO DO2013000030A patent/DOP2013000030A/es unknown
- 2013-02-07 CL CL2013000380A patent/CL2013000380A1/es unknown
- 2013-02-12 ZA ZA2013/01120A patent/ZA201301120B/en unknown
- 2013-02-18 CR CR20130066A patent/CR20130066A/es unknown
- 2013-02-22 US US13/774,635 patent/US8778934B2/en active Active
- 2013-02-22 US US13/774,707 patent/US8916551B2/en active Active
- 2013-03-06 EC ECSP13012478 patent/ECSP13012478A/es unknown
- 2013-03-07 CO CO13046020A patent/CO6680700A2/es active IP Right Grant
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2014
- 2014-11-13 US US14/540,699 patent/US20150073137A1/en not_active Abandoned
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2015
- 2015-07-21 US US14/804,935 patent/US9499568B2/en active Active
- 2015-07-29 JP JP2015149216A patent/JP6113789B2/ja active Active
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2016
- 2016-10-10 US US15/289,650 patent/US9884875B2/en active Active
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2017
- 2017-12-18 US US15/845,621 patent/US20180162875A1/en not_active Abandoned
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2019
- 2019-01-24 US US16/256,773 patent/US10654874B2/en active Active
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2020
- 2020-03-23 US US16/827,316 patent/US11279713B2/en active Active
- 2020-05-25 HR HRP20200844TT patent/HRP20200844T1/hr unknown
- 2020-05-25 CY CY20201100475T patent/CY1123507T1/el unknown
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