HUE049460T2 - Heterociklusos vegyület és annak alkalmazása ampa receptor pozitív allosztérikus modulátorként - Google Patents

Heterociklusos vegyület és annak alkalmazása ampa receptor pozitív allosztérikus modulátorként

Info

Publication number
HUE049460T2
HUE049460T2 HUE11749944A HUE11749944A HUE049460T2 HU E049460 T2 HUE049460 T2 HU E049460T2 HU E11749944 A HUE11749944 A HU E11749944A HU E11749944 A HUE11749944 A HU E11749944A HU E049460 T2 HUE049460 T2 HU E049460T2
Authority
HU
Hungary
Prior art keywords
heterocyclic compound
positive allosteric
receptor positive
ampa receptor
allosteric modulator
Prior art date
Application number
HUE11749944A
Other languages
English (en)
Hungarian (hu)
Inventor
Masakuni Kori
Toshihiro Imaeda
Shinji Nakamura
Masashi Toyofuku
Eiji Honda
Yasutomi Asano
Osamu Ujikawa
Michiyo Mochizuki
Original Assignee
Takeda Pharmaceuticals Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceuticals Co filed Critical Takeda Pharmaceuticals Co
Publication of HUE049460T2 publication Critical patent/HUE049460T2/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biomedical Technology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
HUE11749944A 2010-08-10 2011-08-09 Heterociklusos vegyület és annak alkalmazása ampa receptor pozitív allosztérikus modulátorként HUE049460T2 (hu)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2010179577 2010-08-10

Publications (1)

Publication Number Publication Date
HUE049460T2 true HUE049460T2 (hu) 2020-09-28

Family

ID=44534564

Family Applications (1)

Application Number Title Priority Date Filing Date
HUE11749944A HUE049460T2 (hu) 2010-08-10 2011-08-09 Heterociklusos vegyület és annak alkalmazása ampa receptor pozitív allosztérikus modulátorként

Country Status (39)

Country Link
US (11) US8575154B2 (enExample)
EP (1) EP2603513B1 (enExample)
JP (2) JP5788496B2 (enExample)
KR (1) KR101852215B1 (enExample)
CN (2) CN103180326B (enExample)
AR (1) AR082618A1 (enExample)
AU (1) AU2011290126B2 (enExample)
BR (1) BR112013002250B1 (enExample)
CA (1) CA2807460C (enExample)
CL (1) CL2013000380A1 (enExample)
CO (1) CO6680700A2 (enExample)
CR (1) CR20130066A (enExample)
CY (1) CY1123507T1 (enExample)
DK (1) DK2603513T3 (enExample)
DO (1) DOP2013000030A (enExample)
EA (1) EA022078B1 (enExample)
EC (1) ECSP13012478A (enExample)
ES (1) ES2793723T3 (enExample)
GE (1) GEP20156216B (enExample)
HR (1) HRP20200844T1 (enExample)
HU (1) HUE049460T2 (enExample)
IL (1) IL224452A (enExample)
LT (1) LT2603513T (enExample)
MA (1) MA34509B1 (enExample)
MX (1) MX349470B (enExample)
MY (1) MY165908A (enExample)
NZ (1) NZ607593A (enExample)
PE (1) PE20131116A1 (enExample)
PH (1) PH12013500247A1 (enExample)
PL (1) PL2603513T3 (enExample)
PT (1) PT2603513T (enExample)
RS (1) RS60311B1 (enExample)
SG (1) SG187656A1 (enExample)
SI (1) SI2603513T1 (enExample)
TW (1) TWI504604B (enExample)
UA (1) UA111594C2 (enExample)
UY (1) UY33551A (enExample)
WO (1) WO2012020848A1 (enExample)
ZA (1) ZA201301120B (enExample)

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CN107892697B (zh) 2016-12-26 2020-11-03 郑州泰基鸿诺医药股份有限公司 一种[1,3]噻嗪-2-胺类化合物及应用,药物组合物
SG11201908640TA (en) 2017-03-21 2019-10-30 Fmc Corp Pyrrolidinones and a process to prepare them
BR112019019551A2 (pt) 2017-03-21 2020-04-22 Fmc Corp mistura, e, método para controlar o crescimento de vegetação indesejada
AR111967A1 (es) 2017-05-30 2019-09-04 Fmc Corp Amidas herbicidas
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JP7250686B2 (ja) * 2017-10-06 2023-04-03 武田薬品工業株式会社 複素環化合物
EP3693360B1 (en) * 2017-10-06 2023-12-13 Takeda Pharmaceutical Company Limited Heterocyclic compounds
PL4031552T3 (pl) 2019-09-16 2025-03-17 Takeda Pharmaceutical Company Limited Pochodne azolowo-skondensowanych pirydazyn-3(2h)-onów
TW202207944A (zh) * 2020-05-15 2022-03-01 日商武田藥品工業股份有限公司 抑鬱症之治療
CN113943294A (zh) * 2020-07-15 2022-01-18 成都海博为药业有限公司 一种作为btk抑制剂的化合物及其制备方法与用途
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Also Published As

Publication number Publication date
US20140080817A1 (en) 2014-03-20
CA2807460A1 (en) 2012-02-16
JP6113789B2 (ja) 2017-04-12
ZA201301120B (en) 2014-04-30
CN103180326A (zh) 2013-06-26
US9499568B2 (en) 2016-11-22
US20130190291A1 (en) 2013-07-25
UY33551A (es) 2012-03-30
AU2011290126A1 (en) 2013-03-07
BR112013002250B1 (pt) 2020-10-27
US8778934B2 (en) 2014-07-15
LT2603513T (lt) 2020-05-25
EP2603513B1 (en) 2020-03-11
KR20130138738A (ko) 2013-12-19
US9150591B2 (en) 2015-10-06
WO2012020848A8 (en) 2012-09-27
ECSP13012478A (es) 2013-04-30
CL2013000380A1 (es) 2013-05-31
US8916551B2 (en) 2014-12-23
PE20131116A1 (es) 2013-10-24
PL2603513T3 (pl) 2020-07-27
DK2603513T3 (da) 2020-06-15
MY165908A (en) 2018-05-18
AR082618A1 (es) 2012-12-19
IL224452A (en) 2017-11-30
TWI504604B (zh) 2015-10-21
US20200317692A1 (en) 2020-10-08
HRP20200844T1 (hr) 2020-08-21
CA2807460C (en) 2018-09-18
MX349470B (es) 2017-07-31
JP2016006080A (ja) 2016-01-14
US20170022222A1 (en) 2017-01-26
SI2603513T1 (sl) 2020-07-31
UA111594C2 (uk) 2016-05-25
CO6680700A2 (es) 2013-05-31
US20190263832A1 (en) 2019-08-29
PT2603513T (pt) 2020-06-08
US20240360156A1 (en) 2024-10-31
CN103180326B (zh) 2015-06-10
TW201217386A (en) 2012-05-01
NZ607593A (en) 2015-01-30
US20150353578A1 (en) 2015-12-10
US11279713B2 (en) 2022-03-22
US10654874B2 (en) 2020-05-19
EA022078B1 (ru) 2015-10-30
CN104926837A (zh) 2015-09-23
PH12013500247A1 (en) 2013-03-11
MA34509B1 (fr) 2013-09-02
US20130184266A1 (en) 2013-07-18
ES2793723T3 (es) 2020-11-16
US20180162875A1 (en) 2018-06-14
RS60311B1 (sr) 2020-07-31
SG187656A1 (en) 2013-03-28
BR112013002250A2 (pt) 2016-05-24
DOP2013000030A (es) 2013-03-15
CY1123507T1 (el) 2022-03-24
EP2603513A1 (en) 2013-06-19
JP5788496B2 (ja) 2015-09-30
GEP20156216B (en) 2015-01-12
US9884875B2 (en) 2018-02-06
EA201390222A1 (ru) 2013-08-30
WO2012020848A1 (en) 2012-02-16
CR20130066A (es) 2013-05-03
KR101852215B1 (ko) 2018-04-25
JP2013535408A (ja) 2013-09-12
US20120077799A1 (en) 2012-03-29
AU2011290126B2 (en) 2016-01-07
US8575154B2 (en) 2013-11-05
MX2013001614A (es) 2013-07-05
US20150073137A1 (en) 2015-03-12

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