PL206255B1
(pl)
*
|
2000-07-21 |
2010-07-30 |
Dendreon Corporationdendreon Corporation |
Inhibitor proteazy wirusa zapalenia wątroby C, zawierająca go kompozycja farmaceutyczna i zastosowanie inhibitora do wytwarzania leku do leczenia chorób związanych z HCV oraz zastosowanie do wytwarzania kompozycji do stosowania w kombinowanej terapii
|
EP2399588B1
(fr)
|
2001-01-22 |
2020-04-29 |
Merck Sharp & Dohme Corp. |
Dérivés de nucléosides en tant qu'inhibiteurs de polymérase virale d'arn dépendante de l'arn
|
US6867185B2
(en)
*
|
2001-12-20 |
2005-03-15 |
Bristol-Myers Squibb Company |
Inhibitors of hepatitis C virus
|
CA2369711A1
(fr)
*
|
2002-01-30 |
2003-07-30 |
Boehringer Ingelheim (Canada) Ltd. |
Peptides macrocycliques qui agissent contre le virus de l'hepatite c
|
US7119072B2
(en)
|
2002-01-30 |
2006-10-10 |
Boehringer Ingelheim (Canada) Ltd. |
Macrocyclic peptides active against the hepatitis C virus
|
US6642204B2
(en)
|
2002-02-01 |
2003-11-04 |
Boehringer Ingelheim International Gmbh |
Hepatitis C inhibitor tri-peptides
|
CA2369970A1
(fr)
*
|
2002-02-01 |
2003-08-01 |
Boehringer Ingelheim (Canada) Ltd. |
Tri-peptides inhibiteur de l'hepatite c
|
US7091184B2
(en)
|
2002-02-01 |
2006-08-15 |
Boehringer Ingelheim International Gmbh |
Hepatitis C inhibitor tri-peptides
|
US6828301B2
(en)
|
2002-02-07 |
2004-12-07 |
Boehringer Ingelheim International Gmbh |
Pharmaceutical compositions for hepatitis C viral protease inhibitors
|
PL373399A1
(en)
|
2002-04-11 |
2005-08-22 |
Vertex Pharmaceuticals Incorporated |
Inhibitors of serine proteases, particularly hcv ns3-ns4a protease
|
AU2003301959A1
(en)
|
2002-05-20 |
2004-06-03 |
Bristol-Myers Squibb Company |
Substituted cycloalkyl p1' hepatitis c virus inhibitors
|
JP4312711B2
(ja)
|
2002-05-20 |
2009-08-12 |
ブリストル−マイヤーズ スクイブ カンパニー |
ヘテロ環式スルホンアミドc型肝炎ウイルス阻害剤
|
MY140680A
(en)
|
2002-05-20 |
2010-01-15 |
Bristol Myers Squibb Co |
Hepatitis c virus inhibitors
|
DE60336550D1
(de)
|
2002-05-20 |
2011-05-12 |
Bristol Myers Squibb Co |
Inhibitoren des hepatitis-c-virus
|
US20040138109A1
(en)
*
|
2002-09-30 |
2004-07-15 |
Boehringer Ingelheim Pharmaceuticals, Inc. |
Potent inhibitor of HCV serine protease
|
EP1408031A1
(fr)
*
|
2002-10-09 |
2004-04-14 |
3 D Gene Pharma |
Derivés de pyrolidine comme médicaments contre Hepatitis C
|
US20050075279A1
(en)
|
2002-10-25 |
2005-04-07 |
Boehringer Ingelheim International Gmbh |
Macrocyclic peptides active against the hepatitis C virus
|
US20050159345A1
(en)
*
|
2002-10-29 |
2005-07-21 |
Boehringer Ingelheim International Gmbh |
Composition for the treatment of infection by Flaviviridae viruses
|
DK1558730T3
(da)
*
|
2002-10-29 |
2008-05-26 |
Boehringer Ingelheim Int |
Inhibitorresistent HCV-NS3-protease
|
US7601709B2
(en)
|
2003-02-07 |
2009-10-13 |
Enanta Pharmaceuticals, Inc. |
Macrocyclic hepatitis C serine protease inhibitors
|
WO2004072243A2
(fr)
*
|
2003-02-07 |
2004-08-26 |
Enanta Pharmaceuticals, Inc. |
Inhibiteurs macrocycliques de la serine protease de l'hepatite c
|
UY28240A1
(es)
*
|
2003-03-27 |
2004-11-08 |
Boehringer Ingelheim Pharma |
Fases cristalinas de un potente inhibidor de la hcv
|
NZ543250A
(en)
*
|
2003-04-02 |
2008-12-24 |
Boehringer Ingelheim Int |
Pharmaceutical compositions for hepatitis C viral protease inhibitors
|
WO2004089974A1
(fr)
*
|
2003-04-10 |
2004-10-21 |
Boehringer Ingelheim International Gmbh |
Procede pour preparer des composes macrocycliques par reaction de metathese catalysee par complexe de ruthenium
|
EP1615947A2
(fr)
*
|
2003-04-10 |
2006-01-18 |
Boehringer Ingelheim International GmbH |
Procede de preparation de composes macrocycliques
|
WO2004094452A2
(fr)
|
2003-04-16 |
2004-11-04 |
Bristol-Myers Squibb Company |
Peptide d'isoquinoleine macrocyclique inhibiteurs du virus de l'hepatite c
|
US7176208B2
(en)
|
2003-04-18 |
2007-02-13 |
Enanta Pharmaceuticals, Inc. |
Quinoxalinyl macrocyclic hepatitis C serine protease inhibitors
|
WO2004093798A2
(fr)
|
2003-04-18 |
2004-11-04 |
Enanta Pharmaceuticals, Inc. |
Composes macrocycliques de quinoxalinyle inhibant les serine proteases de l'hepatite c
|
DE602004010137T2
(de)
|
2003-05-21 |
2008-09-11 |
Boehringer Ingelheim Pharma Gmbh & Co. Kg |
Verbindungen als hepatitis c inhibitoren
|
US7273851B2
(en)
|
2003-06-05 |
2007-09-25 |
Enanta Pharmaceuticals, Inc. |
Tri-peptide hepatitis C serine protease inhibitors
|
US7125845B2
(en)
*
|
2003-07-03 |
2006-10-24 |
Enanta Pharmaceuticals, Inc. |
Aza-peptide macrocyclic hepatitis C serine protease inhibitors
|
UY28500A1
(es)
|
2003-09-05 |
2005-04-29 |
Vertex Pharma |
Inhibidores de proteasas de serina, en particular proteasa ns3-ns4a del vhc.
|
MXPA06003141A
(es)
|
2003-09-22 |
2006-06-05 |
Boehringer Ingelheim Int |
Peptidos macrociclicos activos contra el virus de la hepatitis c.
|
DE602004031298D1
(de)
|
2003-09-26 |
2011-03-17 |
Schering Corp |
Makrocyclische inhibitoren der ns3-serinprotease des hepatitis-c-virus
|
EP1692157B1
(fr)
|
2003-10-10 |
2013-04-17 |
Vertex Pharmaceuticals Incorporated |
Inhibiteurs de serine proteases, en particulier la ns3-ns4a protease du hcv
|
AP2287A
(en)
|
2003-10-14 |
2011-10-31 |
Intermune Inc |
Macrocyclic carboxylic acids and acylsulfonamides as inhibitors of HCV replication.
|
CN1894276B
(zh)
|
2003-10-27 |
2010-06-16 |
威特克斯医药股份有限公司 |
Hcv ns3-ns4a蛋白酶抗药性突变体
|
EP1944042A1
(fr)
|
2003-10-27 |
2008-07-16 |
Vertex Pharmceuticals Incorporated |
Combinaisons pour le traitement HCV
|
WO2005043118A2
(fr)
|
2003-10-27 |
2005-05-12 |
Vertex Pharmaceuticals Incorporated |
Methode de decouverte de medicament
|
US7132504B2
(en)
|
2003-11-12 |
2006-11-07 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US7135462B2
(en)
|
2003-11-20 |
2006-11-14 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
CA2546290A1
(fr)
*
|
2003-11-20 |
2005-06-09 |
Schering Corporation |
Inhibiteurs depourvus de liaisons peptidiques de la protease ns3 du virus de l'hepatite c
|
JP2007516239A
(ja)
*
|
2003-11-20 |
2007-06-21 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
特に複分解反応生成物からの、遷移金属の除去方法
|
US7309708B2
(en)
*
|
2003-11-20 |
2007-12-18 |
Birstol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
DE602004019973D1
(de)
*
|
2003-12-08 |
2009-04-23 |
Boehringer Ingelheim Int |
Abtrennung von ruthenium-nebenprodukten durch behandlung mit überkritischen flüssigkeiten
|
GB0500020D0
(en)
|
2005-01-04 |
2005-02-09 |
Novartis Ag |
Organic compounds
|
JP4682155B2
(ja)
|
2004-01-21 |
2011-05-11 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
C型肝炎ウイルスに対して活性な大環状ペプチド
|
WO2005075502A1
(fr)
*
|
2004-01-28 |
2005-08-18 |
Boehringer Ingelheim International Gmbh |
Procede d'elimination de metaux de transition a partir de solutions reactionnelles comportant des sous-produits de metaux de transition
|
NZ548740A
(en)
*
|
2004-01-30 |
2010-06-25 |
Medivir Ab |
HCV NS-3 Serine protease inhibitors
|
AU2011203349B2
(en)
*
|
2004-01-30 |
2012-05-24 |
Medivir Ab |
HCV NS-3 serine protease inhibitors
|
JP2008505849A
(ja)
|
2004-02-04 |
2008-02-28 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
セリンプロテアーゼ、特に、hcv、ns3−ns4aプロテアーゼの阻害剤
|
US20050182252A1
(en)
|
2004-02-13 |
2005-08-18 |
Reddy K. R. |
Novel 2'-C-methyl nucleoside derivatives
|
DK1718608T3
(da)
|
2004-02-20 |
2013-10-14 |
Boehringer Ingelheim Int |
Virale polymeraseinhibitorer
|
US20070049593A1
(en)
|
2004-02-24 |
2007-03-01 |
Japan Tobacco Inc. |
Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor
|
WO2005085275A1
(fr)
|
2004-02-27 |
2005-09-15 |
Schering Corporation |
Inhibiteurs de la protease ns3 du virus de l'hepatite c
|
US7635694B2
(en)
|
2004-02-27 |
2009-12-22 |
Schering Corporation |
Cyclobutenedione-containing compounds as inhibitors of hepatitis C virus NS3 serine protease
|
US7342041B2
(en)
|
2004-02-27 |
2008-03-11 |
Schering Corporation |
3,4-(cyclopentyl)-fused proline compounds as inhibitors of hepatitis C virus NS3 serine protease
|
ES2349328T3
(es)
|
2004-02-27 |
2010-12-30 |
Schering Corporation |
Nuevos compuestos como inhibidores de la serina proteasa ns3 del virus de la hepatitis c.
|
EP1742914A1
(fr)
*
|
2004-02-27 |
2007-01-17 |
Schering Corporation |
Groupes cyclobutenedione contenant des composes servant d'inhibiteurs a la serine protease ns3 du virus de l'hepatite c
|
US7192957B2
(en)
|
2004-02-27 |
2007-03-20 |
Schering Corporation |
Compounds as inhibitors of hepatitis C virus NS3 serine protease
|
BRPI0508867A
(pt)
*
|
2004-03-15 |
2007-09-04 |
Boehringer Ingelheim Int |
processo para a preparação de compostos macrocìclicos
|
WO2005095403A2
(fr)
*
|
2004-03-30 |
2005-10-13 |
Intermune, Inc. |
Composes macrocycliques inhibiteurs de replication virale
|
JP2008502718A
(ja)
|
2004-05-20 |
2008-01-31 |
シェーリング コーポレイション |
C型肝炎ウイルスns3セリンプロテアーゼのインヒビターとしての置換型プロリン
|
WO2005123087A2
(fr)
|
2004-06-15 |
2005-12-29 |
Merck & Co., Inc. |
Analogues nucleosidiques de c-purine, servant d'inhibiteurs d'arn-polymerase virale arn-dependante
|
CA2571079A1
(fr)
|
2004-06-24 |
2006-02-02 |
Merck & Co., Inc. |
Phosphoramidates d'aryle nucleosidiques pour le traitement d'infection virale arn dependante de l'arn
|
JP5676839B2
(ja)
*
|
2004-07-16 |
2015-02-25 |
ギリアード サイエンシーズ, インコーポレイテッド |
抗ウイルス化合物
|
CA2573346C
(fr)
|
2004-07-20 |
2011-09-20 |
Boehringer Ingelheim International Gmbh |
Analogues peptidiques inhibiteurs de l'hepatite c
|
UY29016A1
(es)
|
2004-07-20 |
2006-02-24 |
Boehringer Ingelheim Int |
Analogos de dipeptidos inhibidores de la hepatitis c
|
ATE513844T1
(de)
|
2004-08-27 |
2011-07-15 |
Schering Corp |
Acylsulfonamidverbindungen als inhibitoren der ns3-serinprotease des hepatitis-c-virus
|
CA2577831A1
(fr)
*
|
2004-09-17 |
2006-03-30 |
Boehringer Ingelheim International Gmbh |
Procede de fabrication d'inhibiteurs de protease hcv macrocycliques
|
JP2008513452A
(ja)
*
|
2004-09-17 |
2008-05-01 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
超臨界流体中の閉環複分解方法
|
JP4977611B2
(ja)
*
|
2004-09-24 |
2012-07-18 |
ベーリンガー インゲルハイム ファーマシューティカルズ インコーポレイテッド |
新規な種類の界面活性剤様物質
|
BRPI0517463A
(pt)
*
|
2004-10-21 |
2008-10-07 |
Pfizer |
inibidores da protease do vìrus da hepatite c, composições e tratamentos usando os mesmos
|
US7659263B2
(en)
|
2004-11-12 |
2010-02-09 |
Japan Tobacco Inc. |
Thienopyrrole compound and use thereof as HCV polymerase inhibitor
|
CA2591572A1
(fr)
|
2004-12-20 |
2006-06-29 |
Tibotec Pharmaceuticals Ltd. |
Procede et systeme de traitement de l'hepatite c
|
DE102005002336A1
(de)
|
2005-01-17 |
2006-07-20 |
Boehringer Ingelheim Pharma Gmbh & Co. Kg |
Verfahren zur Durchführung von kontinuierlichen Olefin-Ringschluss-Metathesen in komprimiertem Kohlendioxid
|
US7323447B2
(en)
|
2005-02-08 |
2008-01-29 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
WO2006096652A2
(fr)
|
2005-03-08 |
2006-09-14 |
Boehringer Ingelheim International Gmbh |
Preparation de composes macrocycliques
|
EP1879607B1
(fr)
|
2005-05-02 |
2014-11-12 |
Merck Sharp & Dohme Corp. |
Inhibiteurs de la protease ns3 du vhc
|
US7592336B2
(en)
|
2005-05-10 |
2009-09-22 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
JP5030947B2
(ja)
|
2005-05-13 |
2012-09-19 |
ヴァイロケム・ファーマ・インコーポレーテッド |
フラビウイルス感染の治療及び予防のための化合物及び方法
|
AU2006252553B2
(en)
|
2005-06-02 |
2012-03-29 |
Merck Sharp & Dohme Corp. |
Combination of HCV protease inhibitors with a surfactant
|
WO2006130666A2
(fr)
*
|
2005-06-02 |
2006-12-07 |
Schering Corporation |
Medicaments et procedes destines a combiner un inhibiteur de protease hcv et un competiteur akr
|
PL1891089T3
(pl)
|
2005-06-02 |
2015-05-29 |
Merck Sharp & Dohme |
Inhibitory proteazy HCV w połączeniu z pokarmem
|
US7608592B2
(en)
|
2005-06-30 |
2009-10-27 |
Virobay, Inc. |
HCV inhibitors
|
US7601686B2
(en)
|
2005-07-11 |
2009-10-13 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US7470664B2
(en)
|
2005-07-20 |
2008-12-30 |
Merck & Co., Inc. |
HCV NS3 protease inhibitors
|
SG166791A1
(en)
*
|
2005-07-25 |
2010-12-29 |
Intermune Inc |
Novel macrocyclic inhibitors of hepatitis c virus replication
|
TWI393723B
(zh)
|
2005-07-29 |
2013-04-21 |
Tibotec Pharm Ltd |
C型肝炎病毒之大環抑制劑(九)
|
TWI383980B
(zh)
*
|
2005-07-29 |
2013-02-01 |
Tibotec Pharm Ltd |
C型肝炎病毒之大環抑制劑
|
JO2768B1
(en)
|
2005-07-29 |
2014-03-15 |
تيبوتيك فارماسيوتيكالز ليمتد |
Large cyclic inhibitors of hepatitis C virus
|
ES2360417T3
(es)
*
|
2005-07-29 |
2011-06-03 |
Tibotec Pharmaceuticals |
Inhibidores macrocíclicos del virus de la hepatitis c.
|
PE20070210A1
(es)
|
2005-07-29 |
2007-04-16 |
Tibotec Pharm Ltd |
Compuestos macrociclicos como inhibidores del virus de hepatitis c
|
PE20070211A1
(es)
|
2005-07-29 |
2007-05-12 |
Medivir Ab |
Compuestos macrociclicos como inhibidores del virus de hepatitis c
|
PE20070343A1
(es)
*
|
2005-07-29 |
2007-05-12 |
Medivir Ab |
Inhibidores macrociclicos del virus de la hepatitis c
|
CA2617096C
(fr)
|
2005-07-29 |
2013-12-24 |
Tibotec Pharmaceuticals Ltd. |
Inhibiteurs macrocycliques du virus de l'hepatite c
|
ES2373685T3
(es)
|
2005-07-29 |
2012-02-07 |
Tibotec Pharmaceuticals |
Inhibidores macrocíclicos del virus de la hepatitis c.
|
BRPI0614620A2
(pt)
|
2005-07-29 |
2011-04-12 |
Tibotec Pharm Ltd |
compostos inibidores macrocìclicos do vìrus da hepatite c, uso dos mesmos, processo para preparar os referidos compostos, combinação e composição farmacêutica
|
MY142972A
(en)
*
|
2005-07-29 |
2011-01-31 |
Tibotec Pharm Ltd |
Macrocyclic inhibitors of hepatitis c virus
|
RU2008107972A
(ru)
|
2005-08-01 |
2009-09-10 |
Мерк энд Ко., Инк. (US) |
Макроциклические пептиды в качестве ингибиторов ns3-протеазы hcv
|
CN101277950B
(zh)
|
2005-08-02 |
2013-03-27 |
弗特克斯药品有限公司 |
丝氨酸蛋白酶抑制剂
|
US7632821B2
(en)
|
2005-08-09 |
2009-12-15 |
Merck & Co., Inc. |
Ribonucleoside cyclic acetal derivatives for the treatment of RNA-dependent RNA viral infection
|
US8076365B2
(en)
|
2005-08-12 |
2011-12-13 |
Boehringer Ingelheim International Gmbh |
Viral polymerase inhibitors
|
PL1934179T4
(pl)
|
2005-08-19 |
2014-03-31 |
Vertex Pharma |
Sposoby i związki pośrednie
|
AR055395A1
(es)
|
2005-08-26 |
2007-08-22 |
Vertex Pharma |
Compuestos inhibidores de la actividad de la serina proteasa ns3-ns4a del virus de la hepatitis c
|
DE602006019323D1
(de)
|
2005-10-11 |
2011-02-10 |
Intermune Inc |
Verbindungen und verfahren zur inhibierung der replikation des hepatitis-c-virus
|
US7772183B2
(en)
|
2005-10-12 |
2010-08-10 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US7741281B2
(en)
|
2005-11-03 |
2010-06-22 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US7705138B2
(en)
|
2005-11-11 |
2010-04-27 |
Vertex Pharmaceuticals Incorporated |
Hepatitis C virus variants
|
EP2392590A3
(fr)
|
2005-11-11 |
2012-03-14 |
Vertex Pharmaceuticals Incorporated |
Variantes du virus de l'hépatite C
|
US7816348B2
(en)
|
2006-02-03 |
2010-10-19 |
Boehringer Ingelheim International Gmbh |
Viral polymerase inhibitors
|
GB0609492D0
(en)
|
2006-05-15 |
2006-06-21 |
Angeletti P Ist Richerche Bio |
Therapeutic agents
|
US8268776B2
(en)
|
2006-06-06 |
2012-09-18 |
Enanta Pharmaceuticals, Inc. |
Macrocylic oximyl hepatitis C protease inhibitors
|
US9526769B2
(en)
|
2006-06-06 |
2016-12-27 |
Enanta Pharmaceuticals, Inc. |
Macrocylic oximyl hepatitis C protease inhibitors
|
GB0612423D0
(en)
|
2006-06-23 |
2006-08-02 |
Angeletti P Ist Richerche Bio |
Therapeutic agents
|
PE20080992A1
(es)
|
2006-06-26 |
2008-08-06 |
Enanta Pharm Inc |
Quinoxalinil macrociclicos inhibidores de serina proteasa del virus de la hepatitis c
|
RU2008152171A
(ru)
|
2006-07-05 |
2010-08-10 |
Интермьюн, Инк. (Us) |
Новые ингибиторы вирусной репликации гепатита с
|
US7935670B2
(en)
|
2006-07-11 |
2011-05-03 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
KR101512477B1
(ko)
|
2006-07-13 |
2015-04-15 |
아칠리온 파르마세우티칼스 인코포레이티드 |
바이러스 복제 억제제로서 사용되는 4-아미노-4-옥소부타노일 펩티드
|
EP1886685A1
(fr)
|
2006-08-11 |
2008-02-13 |
INSERM (Institut National de la Santé et de la Recherche Médicale) |
Méthodes, utilisations et compositions pour la modulation de la réplication du HCV par activation ou inhibition du récepteur farnesoid X
|
JP2010500978A
(ja)
|
2006-08-17 |
2010-01-14 |
ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング |
ウイルスポリメラーゼインヒビター
|
AU2007309544B2
(en)
|
2006-10-24 |
2012-05-31 |
Msd Italia S.R.L. |
HCV NS3 protease inhibitors
|
CA2667266C
(fr)
|
2006-10-24 |
2015-11-24 |
Merck & Co., Inc. |
Inhibiteurs de la protease ns3 du hcv
|
US8377873B2
(en)
|
2006-10-24 |
2013-02-19 |
Merck Sharp & Dohme Corp. |
HCV NS3 protease inhibitors
|
CA2667032A1
(fr)
|
2006-10-27 |
2008-05-15 |
Merck & Co., Inc. |
Inhibiteurs de protease ns3 du vhc
|
BRPI0718161A2
(pt)
|
2006-10-27 |
2013-11-26 |
Merck & Co Inc |
Composto, composição farmacêutica, e, uso do composto.
|
US8343477B2
(en)
|
2006-11-01 |
2013-01-01 |
Bristol-Myers Squibb Company |
Inhibitors of hepatitis C virus
|
US7772180B2
(en)
|
2006-11-09 |
2010-08-10 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
KR20090086081A
(ko)
|
2006-11-15 |
2009-08-10 |
바이로켐 파마 인코포레이티드 |
플라비바이러스 감염의 치료 또는 예방용 티오펜 유사체
|
US7763584B2
(en)
|
2006-11-16 |
2010-07-27 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US8003604B2
(en)
|
2006-11-16 |
2011-08-23 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US7888464B2
(en)
|
2006-11-16 |
2011-02-15 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
CA2661338C
(fr)
|
2006-11-17 |
2015-05-12 |
Tibotec Pharmaceuticals Ltd. |
Inhibiteurs macrocycliques du virus de l'hepatite c
|
US8101595B2
(en)
|
2006-12-20 |
2012-01-24 |
Istituto di Ricerche di Biologia Molecolare P. Angletti SpA |
Antiviral indoles
|
GB0625349D0
(en)
|
2006-12-20 |
2007-01-31 |
Angeletti P Ist Richerche Bio |
Therapeutic compounds
|
GB0625345D0
(en)
|
2006-12-20 |
2007-01-31 |
Angeletti P Ist Richerche Bio |
Therapeutic compounds
|
DE602008001251D1
(de)
|
2007-02-01 |
2010-06-24 |
Tibotec Pharm Ltd |
Verfahren und zwischenprodukte zur herstellung eines makrozyklischen proteasehemmers von hcv
|
CN101627020B
(zh)
*
|
2007-02-08 |
2015-06-17 |
泰博特克药品有限公司 |
抑制hcv的大环苯基氨基甲酸酯
|
WO2008095999A1
(fr)
*
|
2007-02-08 |
2008-08-14 |
Tibotec Pharmaceuticals Ltd. |
Inhibiteurs macrocycliques du virus de l'hépatite c (vhc) substitués par pyrimidine
|
WO2008106130A2
(fr)
*
|
2007-02-26 |
2008-09-04 |
Achillion Pharmaceuticals, Inc. |
Peptides substitués par une amine tertiaire utiles comme inhibiteurs de la réplication du virus de l'hépatite c
|
ATE548044T1
(de)
|
2007-05-04 |
2012-03-15 |
Vertex Pharma |
Kombinationstherapie zur behandlung von hiv- infektionen
|
BRPI0811447A2
(pt)
|
2007-05-10 |
2014-10-29 |
Intermune Inc |
Compostos, composição farmacêutica e métodos de inibição da atividade da protease ns3/ns4, de tratamento da fibrose hepática e de intensificação da função hepática num indivíduo tendo infecção de vírus da hepatite c.
|
JP5465666B2
(ja)
|
2007-06-29 |
2014-04-09 |
ギリアード サイエンシーズ, インコーポレイテッド |
抗ウイルス化合物
|
KR20100038417A
(ko)
|
2007-06-29 |
2010-04-14 |
길리애드 사이언시즈, 인코포레이티드 |
항바이러스 화합물
|
AU2008277440A1
(en)
|
2007-07-17 |
2009-01-22 |
Istituto Di Ricerche Di Biologia Molecolare P. Angeletti Spa |
Macrocyclic indole derivatives for the treatment of hepatitis C infections
|
CA2699891C
(fr)
|
2007-07-19 |
2013-10-22 |
Nigel Liverton |
Composes macrocycliques servant d'agents antiviraux
|
US8242140B2
(en)
|
2007-08-03 |
2012-08-14 |
Boehringer Ingelheim International Gmbh |
Viral polymerase inhibitors
|
GB0718575D0
(en)
|
2007-09-24 |
2007-10-31 |
Angeletti P Ist Richerche Bio |
Nucleoside derivatives as inhibitors of viral polymerases
|
US8383583B2
(en)
|
2007-10-26 |
2013-02-26 |
Enanta Pharmaceuticals, Inc. |
Macrocyclic, pyridazinone-containing hepatitis C serine protease inhibitors
|
JP5529036B2
(ja)
|
2007-12-05 |
2014-06-25 |
エナンタ ファーマシューティカルズ インコーポレイテッド |
フッ素化トリペプチドhcvセリンプロテアーゼ阻害剤
|
WO2009073780A1
(fr)
|
2007-12-06 |
2009-06-11 |
Enanta Pharmaceuticals, Inc. |
Procédé de préparation d'inhibiteurs de protéase de l'hépatite c oximyle macrocycliques
|
AU2008338273B2
(en)
|
2007-12-19 |
2014-10-02 |
Boehringer Ingelheim International Gmbh |
Viral polymerase inhibitors
|
US8202996B2
(en)
|
2007-12-21 |
2012-06-19 |
Bristol-Myers Squibb Company |
Crystalline forms of N-(tert-butoxycarbonyl)-3-methyl-L-valyl-(4R)-4-((7-chloro-4-methoxy-1-isoquinolinyl)oxy)-N- ((1R,2S)-1-((cyclopropylsulfonyl)carbamoyl)-2-vinylcyclopropyl)-L-prolinamide
|
AR070413A1
(es)
|
2008-02-04 |
2010-04-07 |
Idenix Pharmaceuticals Inc |
Inhibidores macrociclicos de proteasa de serina
|
JP5490778B2
(ja)
|
2008-03-20 |
2014-05-14 |
エナンタ ファーマシューティカルズ インコーポレイテッド |
C型肝炎ウイルス阻害剤としてのフッ素化大環状化合物
|
EP2282762A2
(fr)
|
2008-04-15 |
2011-02-16 |
Intermune, Inc. |
Nouveaux inhibiteurs macrocycliques de la réplication du virus de l hépatite c
|
US8163921B2
(en)
|
2008-04-16 |
2012-04-24 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
CN102014911A
(zh)
|
2008-04-28 |
2011-04-13 |
默沙东公司 |
Hcv ns3蛋白酶抑制剂
|
US7964560B2
(en)
|
2008-05-29 |
2011-06-21 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
WO2009148923A1
(fr)
*
|
2008-05-29 |
2009-12-10 |
Bristol-Myers Squibb Company |
Inhibiteurs du virus de l’hépatite c
|
RS52534B
(en)
|
2008-07-22 |
2013-04-30 |
Merck Sharp & Dohme Corp. |
MACROCYCLIC COMPOUNDS OF HINOXALINE AS HCV NS3 PROTEASE INHIBITORS
|
US8207341B2
(en)
|
2008-09-04 |
2012-06-26 |
Bristol-Myers Squibb Company |
Process or synthesizing substituted isoquinolines
|
UY32099A
(es)
|
2008-09-11 |
2010-04-30 |
Enanta Pharm Inc |
Inhibidores macrocíclicos de serina proteasas de hepatitis c
|
AU2009293494B2
(en)
|
2008-09-16 |
2014-04-24 |
Boehringer Ingelheim International Gmbh |
Crystalline forms of a 2-thiazolyl- 4-quinolinyl-oxy derivative, a potent HCV inhibitor
|
US8563505B2
(en)
|
2008-09-29 |
2013-10-22 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US8044087B2
(en)
|
2008-09-29 |
2011-10-25 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
WO2010039801A2
(fr)
|
2008-10-02 |
2010-04-08 |
The J. David Gladstone Institutes |
Méthodes de traitement d’une infection par le virus de l’hépatite c
|
JP5600111B2
(ja)
|
2008-10-22 |
2014-10-01 |
アレイ バイオファーマ、インコーポレイテッド |
TRKキナーゼ阻害剤としての置換ピラゾロ[1,5−a]ピリミジン化合物
|
AU2009316472B2
(en)
*
|
2008-11-20 |
2015-07-09 |
Achillion Pharmaceuticals, Inc. |
Cyclic carboxamide compounds and analogues thereof as of Hepatitis C virus
|
CN102245599B
(zh)
|
2008-12-10 |
2014-05-14 |
艾其林医药公司 |
作为病毒复制抑制剂的新的4-氨基-4-氧代丁酰基肽
|
KR20110096557A
(ko)
*
|
2008-12-10 |
2011-08-30 |
아칠리온 파르마세우티칼스 인코포레이티드 |
바이러스 복제의 억제제로서 4-아미노-4-옥소부타노일 펩티드 사이클릭 유사체
|
US8283310B2
(en)
|
2008-12-15 |
2012-10-09 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
MX2011007195A
(es)
|
2009-01-07 |
2013-07-12 |
Scynexis Inc |
Derivado de ciclosporina para el uso en el tratamiento de infección de virus de hepatitis c (vhc) y virus de inmunodeficiencia humana (vih).
|
WO2010082050A1
(fr)
|
2009-01-16 |
2010-07-22 |
Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. |
Composés benzoxazocines substitués 7-aminoalkyle macrocycycliques destinés au traitement des infections par hépatite c
|
GB0900914D0
(en)
|
2009-01-20 |
2009-03-04 |
Angeletti P Ist Richerche Bio |
Antiviral agents
|
AR075584A1
(es)
|
2009-02-27 |
2011-04-20 |
Intermune Inc |
COMPOSICIONES TERAPEUTICAS QUE COMPRENDEN beta-D-2'-DESOXI-2'-FLUORO-2'-C-METILCITIDINA Y UN DERIVADO DE ACIDO ISOINDOL CARBOXILICO Y SUS USOS. COMPUESTO.
|
US8193372B2
(en)
|
2009-03-04 |
2012-06-05 |
Idenix Pharmaceuticals, Inc. |
Phosphothiophene and phosphothiazole HCV polymerase inhibitors
|
EP2408449A4
(fr)
|
2009-03-18 |
2012-08-08 |
Univ Leland Stanford Junior |
Méthodes et compositions pour traiter l'infection par un virus de la famille des flaviviridae
|
JP2012523419A
(ja)
|
2009-04-08 |
2012-10-04 |
イデニク プハルマセウティカルス,インコーポレイテッド |
大環状セリンプロテアーゼ阻害剤
|
JP5639155B2
(ja)
|
2009-05-13 |
2014-12-10 |
エナンタ ファーマシューティカルズ インコーポレイテッド |
C型肝炎ウイルスインヒビターとしての大環状化合物
|
US8232246B2
(en)
|
2009-06-30 |
2012-07-31 |
Abbott Laboratories |
Anti-viral compounds
|
AR077468A1
(es)
|
2009-07-09 |
2011-08-31 |
Array Biopharma Inc |
Compuestos de pirazolo (1,5 -a) pirimidina sustituidos como inhibidores de trk- quinasa
|
WO2011014487A1
(fr)
|
2009-07-30 |
2011-02-03 |
Merck Sharp & Dohme Corp. |
Inhibiteurs de protéase ns3 du virus de l'hépatite c
|
US9284307B2
(en)
|
2009-08-05 |
2016-03-15 |
Idenix Pharmaceuticals Llc |
Macrocyclic serine protease inhibitors
|
US20110117055A1
(en)
|
2009-11-19 |
2011-05-19 |
Macdonald James E |
Methods of Treating Hepatitis C Virus with Oxoacetamide Compounds
|
EP2504343A4
(fr)
*
|
2009-11-24 |
2013-04-17 |
Boehringer Ingelheim Int |
Composés inhibiteurs de l'hépatite c
|
EP2504344A4
(fr)
*
|
2009-11-24 |
2013-06-05 |
Boehringer Ingelheim Int |
Composés inhibiteurs de l'hépatite c
|
MX2012006026A
(es)
|
2009-11-25 |
2012-08-15 |
Vertex Pharma |
Derivados de acido 5-alquinil-tiofen-2-carboxilico y usos para tratamiento o prevencion de infecciones por flavivirus.
|
MX2012006877A
(es)
|
2009-12-18 |
2012-08-31 |
Idenix Pharmaceuticals Inc |
Inhibidores de virus de hepatitis c de arileno o heteroarileno 5, 5 - fusionado.
|
WO2011079327A1
(fr)
|
2009-12-24 |
2011-06-30 |
Vertex Pharmaceuticals Incorporated |
Analogues destinés au traitement ou à la prévention d'infections à flavivirus
|
EP2550262A1
(fr)
|
2010-03-24 |
2013-01-30 |
Vertex Pharmaceuticals Incorporated |
Analogues destinés au traitement ou à la prévention d'infections à flavivirus
|
JP2013522375A
(ja)
|
2010-03-24 |
2013-06-13 |
バーテックス ファーマシューティカルズ インコーポレイテッド |
フラビウイルス感染を処置または予防するためのアナログ
|
AU2011232348A1
(en)
|
2010-03-24 |
2012-10-11 |
Vertex Pharmaceuticals Incorporated |
Analogues for the treatment or prevention of Flavivirus infections
|
EP2550268A1
(fr)
|
2010-03-24 |
2013-01-30 |
Vertex Pharmaceuticals Incorporated |
Analogues pour traiter ou prévenir les infections à flavivirus
|
KR101852169B1
(ko)
*
|
2010-05-20 |
2018-04-26 |
어레이 바이오파마 인크. |
Trk 키나제 저해제로서의 매크로시클릭 화합물
|
WO2011156545A1
(fr)
|
2010-06-09 |
2011-12-15 |
Vertex Pharmaceuticals Incorporated |
Modèle dynamique viral pour une polythérapie contre le vhc
|
EP2582717A2
(fr)
|
2010-06-15 |
2013-04-24 |
Vertex Pharmaceuticals Incorporated |
Mutants de la protéase ns5b du vhc
|
WO2012006070A1
(fr)
|
2010-06-28 |
2012-01-12 |
Vertex Pharmaceuticals Incorporated |
Composés et méthodes de traitement ou de prévention d'infections à flavivirus
|
EP2585447A2
(fr)
|
2010-06-28 |
2013-05-01 |
Vertex Pharmaceuticals Incorporated |
Composés et méthodes pour le traitement ou la prévention d'infections par flavivirus
|
WO2012006060A1
(fr)
|
2010-06-28 |
2012-01-12 |
Vertex Pharmaceuticals Incorporated |
Composés et méthodes de traitement ou de prévention d'infections à flavovirus
|
MX2013001869A
(es)
|
2010-08-17 |
2013-06-28 |
Vertex Pharma |
Compuestos y metodos para el tratamiento o prevencion de infecciones virales por flaviviridae.
|
RS54638B1
(en)
*
|
2010-09-21 |
2016-08-31 |
Enanta Pharmaceuticals, Inc. |
HCV SERIN PROTEASE INHIBITORS DERIVED FROM MACROCYCLIC PROLINE
|
WO2012092409A2
(fr)
|
2010-12-30 |
2012-07-05 |
Enanta Phararmaceuticals, Inc |
Inhibiteurs macrocycliques de sérine protéase d'hépatite c
|
CA2821340A1
(fr)
*
|
2010-12-30 |
2012-07-05 |
Enanta Pharmaceuticals, Inc. |
Inhibiteurs macrocycliques de phenanthridine de serine protease d'hepatite c
|
AR085352A1
(es)
|
2011-02-10 |
2013-09-25 |
Idenix Pharmaceuticals Inc |
Inhibidores macrociclicos de serina proteasa, sus composiciones farmaceuticas y su uso para tratar infecciones por hcv
|
WO2012107589A1
(fr)
|
2011-02-11 |
2012-08-16 |
INSERM (Institut National de la Santé et de la Recherche Médicale) |
Méthodes et compositions pharmaceutiques pour le traitement et la prévention des infections à vhc
|
US20120252721A1
(en)
|
2011-03-31 |
2012-10-04 |
Idenix Pharmaceuticals, Inc. |
Methods for treating drug-resistant hepatitis c virus infection with a 5,5-fused arylene or heteroarylene hepatitis c virus inhibitor
|
US8957203B2
(en)
|
2011-05-05 |
2015-02-17 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
US10201584B1
(en)
|
2011-05-17 |
2019-02-12 |
Abbvie Inc. |
Compositions and methods for treating HCV
|
US8691757B2
(en)
|
2011-06-15 |
2014-04-08 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
WO2013016501A1
(fr)
|
2011-07-26 |
2013-01-31 |
Vertex Pharmaceuticals Incorporated |
Formulations de composés de thiophène
|
WO2013016499A1
(fr)
|
2011-07-26 |
2013-01-31 |
Vertex Pharmaceuticals Incorporated |
Procédés de préparation de composés du thiophène
|
EP2780026B1
(fr)
|
2011-11-15 |
2019-10-23 |
Merck Sharp & Dohme Corp. |
Inhibiteurs de la protéase ns3 du vhc
|
AU2012347785B2
(en)
|
2011-12-06 |
2017-03-16 |
The Board Of Trustees Of The Leland Stanford Junior University |
Methods and compositions for treating viral diseases
|
RU2625796C2
(ru)
*
|
2012-01-11 |
2017-07-19 |
Ф. Хоффманн-Ля Рош Аг |
Макроциклические амиды в качестве ингибиторов протеазы
|
WO2013106344A1
(fr)
|
2012-01-12 |
2013-07-18 |
Ligand Pharmaceuticals, Inc. |
Nucléosides 2'-c-méthyl comprenant un diester de phosphate cyclique de 1,3-propanediol (2-oxo-[1,3,2]-dioxaphosphorinane à la position 5'
|
EP2827876A4
(fr)
|
2012-03-22 |
2015-10-28 |
Alios Biopharma Inc |
Combinaisons pharmaceutiques comprenant un analogue thionucléotidique
|
KR20150074051A
(ko)
*
|
2012-10-19 |
2015-07-01 |
브리스톨-마이어스 스큅 컴퍼니 |
C형 간염 바이러스 억제제
|
WO2014071007A1
(fr)
|
2012-11-02 |
2014-05-08 |
Bristol-Myers Squibb Company |
Inhibiteurs du virus de l'hépatite c
|
US9643999B2
(en)
|
2012-11-02 |
2017-05-09 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
WO2014070964A1
(fr)
|
2012-11-02 |
2014-05-08 |
Bristol-Myers Squibb Company |
Inhibiteurs du virus de l'hépatite c
|
US9409943B2
(en)
|
2012-11-05 |
2016-08-09 |
Bristol-Myers Squibb Company |
Hepatitis C virus inhibitors
|
WO2014121418A1
(fr)
|
2013-02-07 |
2014-08-14 |
Merck Sharp & Dohme Corp. |
Composés hétérocycliques tétracycliques et leurs méthodes d'utilisation pour le traitement de l'hépatite c
|
WO2014121417A1
(fr)
|
2013-02-07 |
2014-08-14 |
Merck Sharp & Dohme Corp. |
Composés hétérocycliques tétracycliques et leurs procédés d'utilisation pour le traitement de l'hépatite c
|
TW201526899A
(zh)
|
2013-02-28 |
2015-07-16 |
Alios Biopharma Inc |
醫藥組成物
|
JP6342922B2
(ja)
|
2013-03-07 |
2018-06-13 |
ブリストル−マイヤーズ スクイブ カンパニーBristol−Myers Squibb Company |
C型肝炎ウイルス阻害剤
|
WO2014138374A1
(fr)
|
2013-03-08 |
2014-09-12 |
Boehringer Ingelheim International Gmbh |
Polythérapie par voie orale pour le traitement d'une infection par le vhc chez une sous-population spécifique de patients
|
WO2014145600A1
(fr)
|
2013-03-15 |
2014-09-18 |
Achillion Pharmaceuticals, Inc. |
Polymorphes de sel de sodium d'ach-0142684, composition les comprenant, et leur procédé de fabrication
|
US9006423B2
(en)
|
2013-03-15 |
2015-04-14 |
Achillion Pharmaceuticals Inc. |
Process for making a 4-amino-4-oxobutanoyl peptide cyclic analogue, an inhibitor of viral replication, and intermediates thereof
|
EP3046924A1
(fr)
|
2013-09-20 |
2016-07-27 |
IDENIX Pharmaceuticals, Inc. |
Inhibiteurs du virus de l'hépatite c
|
WO2015103490A1
(fr)
|
2014-01-03 |
2015-07-09 |
Abbvie, Inc. |
Formes galéniques antivirales solides
|
WO2015134560A1
(fr)
|
2014-03-05 |
2015-09-11 |
Idenix Pharmaceuticals, Inc. |
Formes solides d'un composé inhibiteur des virus de la famille des flaviviridae et sels de celui-ci
|
US20170135990A1
(en)
|
2014-03-05 |
2017-05-18 |
Idenix Pharmaceuticals Llc |
Pharmaceutical compositions comprising a 5,5-fused heteroarylene flaviviridae inhibitor and their use for treating or preventing flaviviridae infection
|
JP6914834B2
(ja)
|
2014-11-16 |
2021-08-04 |
アレイ バイオファーマ インコーポレイテッド |
(S)−N−(5−((R)−2−(2,5−ジフルオロフェニル)−ピロリジン−1−イル)−ピラゾロ[1,5−a]ピリミジン−3−イル)−3−ヒドロキシピロリジン−1−カルボキサミド硫酸水素塩の結晶形
|
AU2016344058A1
(en)
|
2015-10-26 |
2018-05-17 |
Array Biopharma Inc. |
Point mutations in Trk inhibitor-resistant cancer and methods relating to the same
|
US10045991B2
(en)
|
2016-04-04 |
2018-08-14 |
Loxo Oncology, Inc. |
Methods of treating pediatric cancers
|
TN2018000335A1
(en)
|
2016-04-04 |
2020-01-16 |
Loxo Oncology Inc |
Liquid formulations of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide
|
PL3800189T3
(pl)
|
2016-05-18 |
2023-10-23 |
Loxo Oncology, Inc. |
Wytwarzanie (s)-n-(5-((r)-2-(2,5-difluorofenylo)pirolidyn-1-ylo)pirazolo[1,5-a]pirymidyn-3-ylo)-3-hydroksypirolidyno-1-karboksyamidu
|
JOP20190092A1
(ar)
|
2016-10-26 |
2019-04-25 |
Array Biopharma Inc |
عملية لتحضير مركبات بيرازولو[1، 5-a]بيريميدين وأملاح منها
|
CN108059625A
(zh)
*
|
2016-11-09 |
2018-05-22 |
广东广康生化科技股份有限公司 |
一种由噻唑酸制备噻呋酰胺的新型工艺
|
JOP20190213A1
(ar)
|
2017-03-16 |
2019-09-16 |
Array Biopharma Inc |
مركبات حلقية ضخمة كمثبطات لكيناز ros1
|
US11091427B2
(en)
|
2017-03-24 |
2021-08-17 |
Agency For Science, Technology And Research |
Building blocks for stapled peptides
|
US11976084B2
(en)
|
2020-11-23 |
2024-05-07 |
Enanta Pharmaceuticals, Inc. |
Spiropyrrolidine derived antiviral agents
|
US11970502B2
(en)
|
2021-05-04 |
2024-04-30 |
Enanta Pharmaceuticals, Inc. |
Macrocyclic antiviral agents
|
WO2022240541A1
(fr)
*
|
2021-05-11 |
2022-11-17 |
Enanta Pharmaceuticals, Inc. |
Nouveaux agents antiviraux dérivés de spiropyrrolidine macrocycliques
|
US11919910B2
(en)
|
2021-11-12 |
2024-03-05 |
Enanta Pharmaceuticals, Inc. |
Spiropyrrolidine derived antiviral agents
|
WO2023086352A1
(fr)
|
2021-11-12 |
2023-05-19 |
Enanta Pharmaceuticals, Inc. |
Nouveaux agents antiviraux dérivés de spiropyrrolidine
|
WO2023086350A1
(fr)
|
2021-11-12 |
2023-05-19 |
Enanta Pharmaceuticals, Inc. |
Agents antiviraux contenant des alcynes
|
US11993600B2
(en)
|
2021-12-08 |
2024-05-28 |
Enanta Pharmaceuticals, Inc. |
Saturated spirocyclics as antiviral agents
|