MX380147B - Formas de dosificacion de ruxolitinib de liberacion sostenida. - Google Patents

Formas de dosificacion de ruxolitinib de liberacion sostenida.

Info

Publication number
MX380147B
MX380147B MX2015005947A MX2015005947A MX380147B MX 380147 B MX380147 B MX 380147B MX 2015005947 A MX2015005947 A MX 2015005947A MX 2015005947 A MX2015005947 A MX 2015005947A MX 380147 B MX380147 B MX 380147B
Authority
MX
Mexico
Prior art keywords
ruxolitinib
sustained
dosage forms
release
useful
Prior art date
Application number
MX2015005947A
Other languages
English (en)
Other versions
MX2015005947A (es
Inventor
Bhavnish Parikh
Krishnaswamy Yeleswaram
Susan Erickson-Viitanen
William V Williams
Yong Ni
Original Assignee
Incyte Holdings Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49681181&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX380147(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Incyte Holdings Corp filed Critical Incyte Holdings Corp
Publication of MX2015005947A publication Critical patent/MX2015005947A/es
Publication of MX380147B publication Critical patent/MX380147B/es

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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Cardiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • AIDS & HIV (AREA)
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Abstract

La presente invención se refiere a formulaciones de liberación sostenida y formas de dosificación de ruxolitinib o su sal farmacéuticamente aceptable, que son útiles en el tratamiento de enfermedades relacionadas con las cinasa Janus como trastornos mieloproliferativos.
MX2015005947A 2012-11-15 2013-11-14 Formas de dosificacion de ruxolitinib de liberacion sostenida. MX380147B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261726893P 2012-11-15 2012-11-15
US201361769408P 2013-02-26 2013-02-26
PCT/US2013/070012 WO2014078486A1 (en) 2012-11-15 2013-11-14 Sustained-release dosage forms of ruxolitinib

Publications (2)

Publication Number Publication Date
MX2015005947A MX2015005947A (es) 2015-09-08
MX380147B true MX380147B (es) 2025-03-12

Family

ID=49681181

Family Applications (3)

Application Number Title Priority Date Filing Date
MX2020012676A MX2020012676A (es) 2012-11-15 2013-11-14 Formas de dosificación de ruxolitinib de liberación sostenida.
MX2015005947A MX380147B (es) 2012-11-15 2013-11-14 Formas de dosificacion de ruxolitinib de liberacion sostenida.
MX2023000255A MX2023000255A (es) 2012-11-15 2015-05-12 Formas de dosificacion de ruxolitinib de liberacion sostenida.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2020012676A MX2020012676A (es) 2012-11-15 2013-11-14 Formas de dosificación de ruxolitinib de liberación sostenida.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2023000255A MX2023000255A (es) 2012-11-15 2015-05-12 Formas de dosificacion de ruxolitinib de liberacion sostenida.

Country Status (34)

Country Link
US (9) US10166191B2 (es)
EP (2) EP2919766B1 (es)
JP (4) JP2015537030A (es)
KR (3) KR20210037012A (es)
CN (3) CN113384546A (es)
AR (1) AR093490A1 (es)
AU (4) AU2013344780B2 (es)
BR (1) BR112015010663B1 (es)
CA (2) CA3178452A1 (es)
CL (1) CL2015001286A1 (es)
CR (2) CR20190073A (es)
CY (1) CY1124446T1 (es)
DK (1) DK2919766T3 (es)
EA (1) EA201590930A1 (es)
ES (1) ES2880814T3 (es)
HR (1) HRP20211158T1 (es)
HU (1) HUE055894T2 (es)
IL (4) IL317061A (es)
LT (1) LT2919766T (es)
MX (3) MX2020012676A (es)
MY (1) MY191357A (es)
NZ (2) NZ748448A (es)
PE (2) PE20151157A1 (es)
PH (2) PH12020551186B1 (es)
PL (1) PL2919766T3 (es)
PT (1) PT2919766T (es)
RS (1) RS62329B1 (es)
SG (3) SG11201503695XA (es)
SI (1) SI2919766T1 (es)
SM (1) SMT202100436T1 (es)
TW (4) TW202228704A (es)
UA (1) UA120834C2 (es)
WO (1) WO2014078486A1 (es)
ZA (1) ZA202202711B (es)

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EP3070090B1 (en) 2007-06-13 2018-12-12 Incyte Holdings Corporation Use of salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h- pyrazol-1-yl)-3- cyclopentylpropanenitrile
AR076794A1 (es) 2009-05-22 2011-07-06 Incyte Corp Derivados de n-(hetero)aril-pirrolidina de pirazol-4-il-pirrolo [2,3-d]pirimidinas y pirrol-3-il-pirrolo [2,3-d ]pirimidinas como inhibidores de la quinasa janus y composiciones farmaceuticas que los contienen
EP3643312A1 (en) 2009-05-22 2020-04-29 Incyte Holdings Corporation 3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]octane- or heptane-nitrile as jak inhibitors
EP3050882B1 (en) 2010-03-10 2018-01-31 Incyte Holdings Corporation Piperidin-4-yl azetidine derivatives as jak1 inhibitors
SG10201503983QA (en) 2010-05-21 2015-06-29 Incyte Corp Topical Formulation for a JAK Inhibitor
CN103415515B (zh) 2010-11-19 2015-08-26 因塞特公司 作为jak抑制剂的环丁基取代的吡咯并吡啶和吡咯并嘧啶衍生物
PE20140832A1 (es) 2011-06-20 2014-07-14 Incyte Corp Derivados de azetidinil fenil, piridil o pirazinil carboxamida como inhibidores de jak
UA111854C2 (uk) 2011-09-07 2016-06-24 Інсайт Холдінгс Корпорейшн Способи і проміжні сполуки для отримання інгібіторів jak
ES2867048T3 (es) * 2012-06-15 2021-10-20 Concert Pharmaceuticals Inc Derivados deuterados de ruxolitinib
AU2013337824B2 (en) 2012-11-01 2018-03-08 Incyte Holdings Corporation Tricyclic fused thiophene derivatives as JAK inhibitors
PL2919766T3 (pl) 2012-11-15 2021-10-04 Incyte Holdings Corporation Postacie dawkowania ruksolitynibu o przedłużonym uwalnianiu
CN105189509B (zh) 2013-03-06 2017-12-19 因赛特公司 用于制备jak抑制剂的方法及中间体
SMT202100040T1 (it) 2013-05-17 2021-03-15 Incyte Corp Derivati di bipirazolo come inibitori di jak
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