IL164003A0 - Sulfonylamino-derivatives as novel inhibitors of histone deacetylase - Google Patents

Sulfonylamino-derivatives as novel inhibitors of histone deacetylase

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Publication number
IL164003A0
IL164003A0 IL16400303A IL16400303A IL164003A0 IL 164003 A0 IL164003 A0 IL 164003A0 IL 16400303 A IL16400303 A IL 16400303A IL 16400303 A IL16400303 A IL 16400303A IL 164003 A0 IL164003 A0 IL 164003A0
Authority
IL
Israel
Prior art keywords
sulfonylamino
derivatives
histone deacetylase
novel inhibitors
inhibitors
Prior art date
Application number
IL16400303A
Other languages
English (en)
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Priority claimed from PCT/EP2003/002517 external-priority patent/WO2003076401A1/en
Publication of IL164003A0 publication Critical patent/IL164003A0/xx

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    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/22—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with hetero atoms directly attached to ring nitrogen atoms
    • C07D295/26—Sulfur atoms
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PL213783B1 (pl) 2013-05-31
NZ534832A (en) 2005-09-30
AU2003218737B2 (en) 2008-04-10
AU2003212335A1 (en) 2003-09-22
ZA200407233B (en) 2005-10-06
BR0307624A (pt) 2005-01-11
IL164006A0 (en) 2005-12-18
EP1485364B1 (en) 2009-03-11
EP1485353B1 (en) 2011-08-24
ZA200407237B (en) 2005-09-28
CA2476065A1 (en) 2003-09-18
US20120108603A1 (en) 2012-05-03
NO20044113L (no) 2004-09-28
CN100519527C (zh) 2009-07-29
US8343988B2 (en) 2013-01-01
JP2005525379A (ja) 2005-08-25
AU2003218736B2 (en) 2009-01-08
US8697717B2 (en) 2014-04-15
US20090170881A1 (en) 2009-07-02
NO20044194L (no) 2004-10-01
HRP20040799A2 (en) 2005-04-30
AR039566A1 (es) 2005-02-23
AU2003212335B8 (en) 2009-04-23
BR0308081A (pt) 2004-12-21
CA2476065C (en) 2012-07-24
DK1485353T3 (da) 2011-11-28
IL164005A0 (en) 2005-12-18
IL164006A (en) 2010-11-30
ATE473005T1 (de) 2010-07-15
EA200401201A1 (ru) 2005-02-24
EP1485370B1 (en) 2009-03-04
US8455498B2 (en) 2013-06-04
UA77263C2 (en) 2006-11-15
ES2371632T3 (es) 2012-01-05
US9533979B2 (en) 2017-01-03
US20090227558A1 (en) 2009-09-10
US20100010004A1 (en) 2010-01-14
CA2475764A1 (en) 2003-09-18
KR20040090979A (ko) 2004-10-27
AU2003212335B2 (en) 2008-11-27
EA008245B1 (ru) 2007-04-27

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