PL378181A1 - Pochodne kwasu hydroksamidowego jako inhibitory deacetylazy histonowej (HDAC) - Google Patents
Pochodne kwasu hydroksamidowego jako inhibitory deacetylazy histonowej (HDAC)Info
- Publication number
- PL378181A1 PL378181A1 PL378181A PL37818104A PL378181A1 PL 378181 A1 PL378181 A1 PL 378181A1 PL 378181 A PL378181 A PL 378181A PL 37818104 A PL37818104 A PL 37818104A PL 378181 A1 PL378181 A1 PL 378181A1
- Authority
- PL
- Poland
- Prior art keywords
- hdac
- inhibitors
- acid derivatives
- histone deacetylase
- hydroxamid
- Prior art date
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
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- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
- C07D473/08—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
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AU2003900116A AU2003900116A0 (en) | 2003-01-13 | 2003-01-13 | Hdac inhibitor |
AU2003905406A AU2003905406A0 (en) | 2003-10-06 | HDAC Inhibitor |
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CA2479906C (en) | 2002-04-03 | 2011-02-08 | Topotarget Uk Limited | Carbamic acid compounds comprising a piperazine linkage as hdac inhibitors |
AU2003219595A1 (en) | 2002-04-11 | 2003-10-27 | In2Gen Co., Ltd. | Alpha,Beta-UNSATURATED HYDROXAMIC ACID DERIVATIVES AND THEIR USE AS HISTONE DEACETYLASE INHIBITORS |
-
2004
- 2004-01-12 TW TW093100678A patent/TW200418806A/zh unknown
- 2004-01-12 US US10/754,541 patent/US7135493B2/en not_active Expired - Fee Related
- 2004-01-13 AR ARP040100085A patent/AR042851A1/es unknown
- 2004-01-13 CA CA002513436A patent/CA2513436A1/en not_active Abandoned
- 2004-01-13 PL PL378181A patent/PL378181A1/pl not_active Application Discontinuation
- 2004-01-13 KR KR1020057012908A patent/KR20050093826A/ko not_active Application Discontinuation
- 2004-01-13 WO PCT/JP2004/000157 patent/WO2004063169A1/en active Application Filing
- 2004-01-13 MX MXPA05007561A patent/MXPA05007561A/es unknown
- 2004-01-13 EP EP04701698A patent/EP1585735A1/en not_active Withdrawn
- 2004-01-13 JP JP2006500390A patent/JP2006518341A/ja not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
AR042851A1 (es) | 2005-07-06 |
WO2004063169A1 (en) | 2004-07-29 |
EP1585735A1 (en) | 2005-10-19 |
MXPA05007561A (es) | 2006-02-08 |
JP2006518341A (ja) | 2006-08-10 |
CA2513436A1 (en) | 2004-07-29 |
KR20050093826A (ko) | 2005-09-23 |
TW200418806A (en) | 2004-10-01 |
US20040229889A1 (en) | 2004-11-18 |
US7135493B2 (en) | 2006-11-14 |
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