DE60326549D1 - Aminocarbonylderivate als histone-deacetylase-inhibitoren - Google Patents

Aminocarbonylderivate als histone-deacetylase-inhibitoren

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Publication number
DE60326549D1
DE60326549D1 DE60326549T DE60326549T DE60326549D1 DE 60326549 D1 DE60326549 D1 DE 60326549D1 DE 60326549 T DE60326549 T DE 60326549T DE 60326549 T DE60326549 T DE 60326549T DE 60326549 D1 DE60326549 D1 DE 60326549D1
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DE
Germany
Prior art keywords
aminocarbonylderivate
inhibitoren
deacetylase
histone
als
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
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DE60326549T
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English (en)
Inventor
Emelen Kristof Van
Winter Hans L J De
Springhouse Dyatkin
Marc G C Verdonck
Lieven Meerpoel
Heusden Jimmy Arnold Vivia Van
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Janssen Pharmaceutica NV
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Janssen Pharmaceutica NV
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Publication of DE60326549D1 publication Critical patent/DE60326549D1/de
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Expired - Lifetime legal-status Critical Current

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    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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EA008245B1 (ru) 2007-04-27
ATE473005T1 (de) 2010-07-15
WO2003075929A1 (en) 2003-09-18
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