IL133906A0 - Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use - Google Patents

Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use

Info

Publication number
IL133906A0
IL133906A0 IL13390698A IL13390698A IL133906A0 IL 133906 A0 IL133906 A0 IL 133906A0 IL 13390698 A IL13390698 A IL 13390698A IL 13390698 A IL13390698 A IL 13390698A IL 133906 A0 IL133906 A0 IL 133906A0
Authority
IL
Israel
Prior art keywords
phenyl
manufacture
processes
crystal modification
pyrimidineamine derivative
Prior art date
Application number
IL13390698A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4218028&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL133906(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of IL133906A0 publication Critical patent/IL133906A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C30—CRYSTAL GROWTH
    • C30B—SINGLE-CRYSTAL GROWTH; UNIDIRECTIONAL SOLIDIFICATION OF EUTECTIC MATERIAL OR UNIDIRECTIONAL DEMIXING OF EUTECTOID MATERIAL; REFINING BY ZONE-MELTING OF MATERIAL; PRODUCTION OF A HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; SINGLE CRYSTALS OR HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; AFTER-TREATMENT OF SINGLE CRYSTALS OR A HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; APPARATUS THEREFOR
    • C30B7/00—Single-crystal growth from solutions using solvents which are liquid at normal temperature, e.g. aqueous solutions

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Metallurgy (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Materials Engineering (AREA)
  • Pulmonology (AREA)
  • Vascular Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
IL13390698A 1997-07-18 1998-07-16 Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use IL133906A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH176497 1997-07-18
PCT/EP1998/004427 WO1999003854A1 (en) 1997-07-18 1998-07-16 Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use

Publications (1)

Publication Number Publication Date
IL133906A0 true IL133906A0 (en) 2001-04-30

Family

ID=4218028

Family Applications (5)

Application Number Title Priority Date Filing Date
IL13390698A IL133906A0 (en) 1997-07-18 1998-07-16 Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
IL133906A IL133906A (en) 1997-07-18 2000-01-06 Different crystalline form of a derivative of N - phenyl - 2 - pyrimidinamine, processes for their preparation and its uses in the preparation of a medical preparation
IL168972A IL168972A (en) 1997-07-18 2005-06-02 A different crystalline form of a derivative of N-phenyl-2-pyrimidinamine
IL174082A IL174082A (en) 1997-07-18 2006-03-02 Methanesulfonate salt of n - phenyl - 2 - pyrimidineamine derivative, process for its preparation and use thereof for the preparation of a tablet containing the same
IL174732A IL174732A0 (en) 1997-07-18 2006-04-03 Use of crystal modification of a n-phenyl-2-pyrimidineamine derivative in the preparation of a medicament for the treatment of restenosis

Family Applications After (4)

Application Number Title Priority Date Filing Date
IL133906A IL133906A (en) 1997-07-18 2000-01-06 Different crystalline form of a derivative of N - phenyl - 2 - pyrimidinamine, processes for their preparation and its uses in the preparation of a medical preparation
IL168972A IL168972A (en) 1997-07-18 2005-06-02 A different crystalline form of a derivative of N-phenyl-2-pyrimidinamine
IL174082A IL174082A (en) 1997-07-18 2006-03-02 Methanesulfonate salt of n - phenyl - 2 - pyrimidineamine derivative, process for its preparation and use thereof for the preparation of a tablet containing the same
IL174732A IL174732A0 (en) 1997-07-18 2006-04-03 Use of crystal modification of a n-phenyl-2-pyrimidineamine derivative in the preparation of a medicament for the treatment of restenosis

Country Status (31)

Country Link
US (5) US6894051B1 (de)
EP (1) EP0998473B1 (de)
JP (1) JP3276359B2 (de)
KR (1) KR100450356B1 (de)
CN (1) CN1134430C (de)
AR (2) AR016351A1 (de)
AT (1) ATE251152T1 (de)
AU (1) AU740713B2 (de)
BR (1) BR9810920A (de)
CA (1) CA2296604C (de)
CO (1) CO4940418A1 (de)
CZ (1) CZ298531B6 (de)
DE (1) DE69818674T2 (de)
DK (1) DK0998473T3 (de)
ES (1) ES2209194T3 (de)
HK (1) HK1028599A1 (de)
HU (1) HU230185B1 (de)
ID (1) ID24093A (de)
IL (5) IL133906A0 (de)
MY (2) MY128664A (de)
NO (2) NO319486B1 (de)
NZ (1) NZ502295A (de)
PE (1) PE97899A1 (de)
PL (1) PL188348B1 (de)
PT (1) PT998473E (de)
RU (1) RU2208012C2 (de)
SK (2) SK287276B6 (de)
TR (1) TR200000060T2 (de)
TW (1) TW491845B (de)
WO (1) WO1999003854A1 (de)
ZA (1) ZA986362B (de)

Families Citing this family (345)

* Cited by examiner, † Cited by third party
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