NO331016B1 - Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat - Google Patents

Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat

Info

Publication number
NO331016B1
NO331016B1 NO20052755A NO20052755A NO331016B1 NO 331016 B1 NO331016 B1 NO 331016B1 NO 20052755 A NO20052755 A NO 20052755A NO 20052755 A NO20052755 A NO 20052755A NO 331016 B1 NO331016 B1 NO 331016B1
Authority
NO
Norway
Prior art keywords
phenyl
crystal modification
pyrimidinamine derivative
pyrimidinamine
derivative
Prior art date
Application number
NO20052755A
Other languages
English (en)
Other versions
NO20052755L (no
NO20052755D0 (no
Inventor
Jürg Zimmermann
Bertrand Sutter
Hans Michael Bürger
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=4218028&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO331016(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Publication of NO20052755L publication Critical patent/NO20052755L/no
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20052755D0 publication Critical patent/NO20052755D0/no
Publication of NO331016B1 publication Critical patent/NO331016B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C30CRYSTAL GROWTH
    • C30BSINGLE-CRYSTAL GROWTH; UNIDIRECTIONAL SOLIDIFICATION OF EUTECTIC MATERIAL OR UNIDIRECTIONAL DEMIXING OF EUTECTOID MATERIAL; REFINING BY ZONE-MELTING OF MATERIAL; PRODUCTION OF A HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; SINGLE CRYSTALS OR HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; AFTER-TREATMENT OF SINGLE CRYSTALS OR A HOMOGENEOUS POLYCRYSTALLINE MATERIAL WITH DEFINED STRUCTURE; APPARATUS THEREFOR
    • C30B7/00Single-crystal growth from solutions using solvents which are liquid at normal temperature, e.g. aqueous solutions

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Metallurgy (AREA)
  • Materials Engineering (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO20052755A 1997-07-18 2005-06-07 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat NO331016B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH176497 1997-07-18
PCT/EP1998/004427 WO1999003854A1 (en) 1997-07-18 1998-07-16 Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use

Publications (3)

Publication Number Publication Date
NO20052755L NO20052755L (no) 2000-01-17
NO20052755D0 NO20052755D0 (no) 2005-06-07
NO331016B1 true NO331016B1 (no) 2011-09-12

Family

ID=4218028

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20000227A NO319486B1 (no) 1997-07-18 2000-01-17 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat, farmasøytisk sammensetning innbefattende samme, fremgangsmåte for fremstilling av samme og anvendelse av samme for fremstilling av preparat
NO20052755A NO331016B1 (no) 1997-07-18 2005-06-07 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO20000227A NO319486B1 (no) 1997-07-18 2000-01-17 Krystallmodifikasjon av et N-fenyl-2-pyrimidinaminderivat, farmasøytisk sammensetning innbefattende samme, fremgangsmåte for fremstilling av samme og anvendelse av samme for fremstilling av preparat

Country Status (31)

Country Link
US (5) US6894051B1 (no)
EP (1) EP0998473B1 (no)
JP (1) JP3276359B2 (no)
KR (1) KR100450356B1 (no)
CN (1) CN1134430C (no)
AR (2) AR016351A1 (no)
AT (1) ATE251152T1 (no)
AU (1) AU740713B2 (no)
BR (1) BR9810920A (no)
CA (1) CA2296604C (no)
CO (1) CO4940418A1 (no)
CZ (1) CZ298531B6 (no)
DE (1) DE69818674T2 (no)
DK (1) DK0998473T3 (no)
ES (1) ES2209194T3 (no)
HK (1) HK1028599A1 (no)
HU (1) HU230185B1 (no)
ID (1) ID24093A (no)
IL (5) IL133906A0 (no)
MY (2) MY128664A (no)
NO (2) NO319486B1 (no)
NZ (1) NZ502295A (no)
PE (1) PE97899A1 (no)
PL (1) PL188348B1 (no)
PT (1) PT998473E (no)
RU (1) RU2208012C2 (no)
SK (2) SK287276B6 (no)
TR (1) TR200000060T2 (no)
TW (1) TW491845B (no)
WO (1) WO1999003854A1 (no)
ZA (1) ZA986362B (no)

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