BR9612465A - Compostos heterocíclicos - Google Patents

Compostos heterocíclicos

Info

Publication number
BR9612465A
BR9612465A BR9612465A BR9612465A BR9612465A BR 9612465 A BR9612465 A BR 9612465A BR 9612465 A BR9612465 A BR 9612465A BR 9612465 A BR9612465 A BR 9612465A BR 9612465 A BR9612465 A BR 9612465A
Authority
BR
Brazil
Prior art keywords
heterocyclic compounds
heterocyclic
compounds
Prior art date
Application number
BR9612465A
Other languages
English (en)
Other versions
BR9612465B1 (pt
Inventor
Philip A Carpino
Jardine Paul A Dasilva
Bruce A Lefker
John A Ragan
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=21737850&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9612465(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of BR9612465A publication Critical patent/BR9612465A/pt
Publication of BR9612465B1 publication Critical patent/BR9612465B1/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C07K5/06034—Dipeptides with the first amino acid being neutral and aliphatic the side chain containing 2 to 4 carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
BRPI9612465-2A 1995-12-28 1996-12-04 compostos dipeptìdicos secretagogos do hormÈnio do crescimento. BR9612465B1 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US946995P 1995-12-28 1995-12-28
PCT/IB1996/001353 WO1997024369A1 (en) 1995-12-28 1996-12-04 Growth-hormone secretagogues

Publications (2)

Publication Number Publication Date
BR9612465A true BR9612465A (pt) 1999-07-13
BR9612465B1 BR9612465B1 (pt) 2010-08-10

Family

ID=21737850

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9612465-2A BR9612465B1 (pt) 1995-12-28 1996-12-04 compostos dipeptìdicos secretagogos do hormÈnio do crescimento.

Country Status (43)

Country Link
US (7) US6124264A (pt)
EP (1) EP0869968B1 (pt)
JP (2) JP3511382B2 (pt)
KR (1) KR100320167B1 (pt)
CN (1) CN1113895C (pt)
AP (2) AP756A (pt)
AR (2) AR004367A1 (pt)
AT (1) ATE361314T1 (pt)
AU (1) AU716934B2 (pt)
BG (1) BG64055B1 (pt)
BR (1) BR9612465B1 (pt)
CA (1) CA2241725C (pt)
CO (1) CO4480108A1 (pt)
CZ (1) CZ293423B6 (pt)
DE (1) DE69637063T2 (pt)
DK (1) DK0869968T3 (pt)
EG (1) EG24195A (pt)
ES (1) ES2285715T3 (pt)
GT (1) GT199600100A (pt)
HN (1) HN1996000085A (pt)
HR (1) HRP960618B1 (pt)
HU (1) HUP9901246A3 (pt)
IL (4) IL138909A0 (pt)
IS (1) IS4758A (pt)
MA (1) MA26415A1 (pt)
MX (1) MX9805157A (pt)
MY (1) MY135727A (pt)
NO (1) NO325135B1 (pt)
NZ (1) NZ322172A (pt)
OA (1) OA10702A (pt)
PE (1) PE30398A1 (pt)
PL (1) PL186916B1 (pt)
PT (1) PT869968E (pt)
RS (1) RS49926B (pt)
SA (1) SA97170581B1 (pt)
SI (1) SI0869968T1 (pt)
SK (1) SK285678B6 (pt)
TN (1) TNSN96172A1 (pt)
TR (1) TR199801233T2 (pt)
TW (1) TW432073B (pt)
UA (1) UA66754C2 (pt)
WO (1) WO1997024369A1 (pt)
ZA (1) ZA9610858B (pt)

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