HRP20040887A2 - Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof - Google Patents

Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof Download PDF

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Publication number
HRP20040887A2
HRP20040887A2 HR20040887A HRP20040887A HRP20040887A2 HR P20040887 A2 HRP20040887 A2 HR P20040887A2 HR 20040887 A HR20040887 A HR 20040887A HR P20040887 A HRP20040887 A HR P20040887A HR P20040887 A2 HRP20040887 A2 HR P20040887A2
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Croatia
Prior art keywords
methyl
trifluoro
ylmethyl
fluoro
methoxyphenyl
Prior art date
Application number
HR20040887A
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English (en)
Croatian (hr)
Inventor
Takahashi Hidenori
Bekkali Younes
Betageri Rajashekhar
G. Cardozo Mario
A. Gilmore Thomas
Hanke Justus Joachim Harcken Christian
M. Kirrane Thomas
Kuzmich Daniel
R. Proudfoot John
Razavi Hossein
Riether Doris
S. Thomson David
Wang Ji
Zindell Renee
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Boehringer Ingelheim Pharmaceuticals Inc.
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Application filed by Boehringer Ingelheim Pharmaceuticals Inc. filed Critical Boehringer Ingelheim Pharmaceuticals Inc.
Publication of HRP20040887A2 publication Critical patent/HRP20040887A2/hr

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    • C07D209/04Indoles; Hydrogenated indoles
    • C07D209/10Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/12Radicals substituted by oxygen atoms
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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HR20040887A 2002-03-26 2003-03-21 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof HRP20040887A2 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US36775802P 2002-03-26 2002-03-26
US43181702P 2002-12-09 2002-12-09
US44240403P 2003-01-24 2003-01-24
PCT/US2003/008901 WO2003082280A1 (en) 2002-03-26 2003-03-21 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof

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