ECSP045315A - MIMÉTICOS DE GlucocorticoidES, PROCEDIMIENTOS PARA SU PREPARACIÓN, COMPOSICIONES FARMACÉUTICAS Y USOS DE LOS MISMOS - Google Patents
MIMÉTICOS DE GlucocorticoidES, PROCEDIMIENTOS PARA SU PREPARACIÓN, COMPOSICIONES FARMACÉUTICAS Y USOS DE LOS MISMOSInfo
- Publication number
- ECSP045315A ECSP045315A EC2004005315A ECSP045315A ECSP045315A EC SP045315 A ECSP045315 A EC SP045315A EC 2004005315 A EC2004005315 A EC 2004005315A EC SP045315 A ECSP045315 A EC SP045315A EC SP045315 A ECSP045315 A EC SP045315A
- Authority
- EC
- Ecuador
- Prior art keywords
- procedures
- pharmaceutical compositions
- formula
- glucocorticoids
- mimetics
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 4
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 239000003862 glucocorticoid Substances 0.000 title 1
- 229940037128 systemic glucocorticoids Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 102000003676 Glucocorticoid Receptors Human genes 0.000 abstract 2
- 108090000079 Glucocorticoid Receptors Proteins 0.000 abstract 2
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 2
- 230000000172 allergic effect Effects 0.000 abstract 1
- 208000010668 atopic eczema Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 230000002062 proliferating effect Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
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- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/12—Radicals substituted by oxygen atoms
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- Gastroenterology & Hepatology (AREA)
- Psychiatry (AREA)
Abstract
Compuestos de Fórmula (IA) y Fórmula (IB) en las que R1, R2, R3, R4, R5 y R6 son como se definen en la presente memoria para la Fórmula (IA) o la Fórmula (IB), o uno de sus tautómeros, profármacos, solvatos o sales; composiciones farmacéuticas que contienen dichos compuestos y procedimientos para modular la función del receptor de glucocorticoides y procedimientos para tratar estados de enfermedad o trastornos mediados por la función del receptor de glucocorticoides o caracterizados por procesos inflamatorios, alérgicos o proliferativos en un paciente usando estos compuestos.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US36775802P | 2002-03-26 | 2002-03-26 | |
| US43181702P | 2002-12-09 | 2002-12-09 | |
| US44240403P | 2003-01-24 | 2003-01-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP045315A true ECSP045315A (es) | 2004-10-26 |
Family
ID=28678922
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2004005315A ECSP045315A (es) | 2002-03-26 | 2004-09-24 | MIMÉTICOS DE GlucocorticoidES, PROCEDIMIENTOS PARA SU PREPARACIÓN, COMPOSICIONES FARMACÉUTICAS Y USOS DE LOS MISMOS |
Country Status (33)
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| AR (1) | AR039140A1 (es) |
| AT (1) | ATE381333T1 (es) |
| AU (1) | AU2003218342B8 (es) |
| BR (1) | BR0308784A (es) |
| CA (1) | CA2478156C (es) |
| CL (1) | CL2010000375A1 (es) |
| CO (1) | CO5611110A2 (es) |
| CY (1) | CY1107244T1 (es) |
| DE (1) | DE60318188T2 (es) |
| DK (1) | DK1490062T3 (es) |
| EA (1) | EA008830B1 (es) |
| EC (1) | ECSP045315A (es) |
| ES (1) | ES2298508T3 (es) |
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| IL (1) | IL163366A (es) |
| MX (1) | MXPA04009329A (es) |
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