IL139865A0 - A liver selective glucocorticoid antagonist and pharmaceutical compositions containing the same - Google Patents
A liver selective glucocorticoid antagonist and pharmaceutical compositions containing the sameInfo
- Publication number
- IL139865A0 IL139865A0 IL13986599A IL13986599A IL139865A0 IL 139865 A0 IL139865 A0 IL 139865A0 IL 13986599 A IL13986599 A IL 13986599A IL 13986599 A IL13986599 A IL 13986599A IL 139865 A0 IL139865 A0 IL 139865A0
- Authority
- IL
- Israel
- Prior art keywords
- same
- pharmaceutical compositions
- compositions containing
- selective glucocorticoid
- glucocorticoid antagonist
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB9812314.4A GB9812314D0 (en) | 1998-06-08 | 1998-06-08 | Treatment of diabetes |
GBGB9815149.1A GB9815149D0 (en) | 1998-07-13 | 1998-07-13 | Treatment of diabetes |
PCT/IB1999/001175 WO1999063976A2 (en) | 1998-06-08 | 1999-06-07 | Liver-selective glucocorticoid antagonist for treating diabetes |
Publications (1)
Publication Number | Publication Date |
---|---|
IL139865A0 true IL139865A0 (en) | 2002-02-10 |
Family
ID=26313822
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL13986599A IL139865A0 (en) | 1998-06-08 | 1999-06-07 | A liver selective glucocorticoid antagonist and pharmaceutical compositions containing the same |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP1143948A3 (en) |
JP (1) | JP2002527355A (en) |
KR (1) | KR20010052431A (en) |
AU (1) | AU751569B2 (en) |
CA (1) | CA2334116A1 (en) |
IL (1) | IL139865A0 (en) |
WO (1) | WO1999063976A2 (en) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9816935D0 (en) * | 1998-08-05 | 1998-09-30 | Karobio Ab | Novel glucocortoid and thyroid receptor ligands for the treatment of metabolic disorders |
GB9907048D0 (en) | 1999-03-27 | 1999-05-19 | Karobio Ab | Novel glucocorticoid receptor ligands for the treatment of meta bolic disorders |
GB9928805D0 (en) * | 1999-12-07 | 2000-02-02 | Karobio Ab | Compounds active at the Glucocorticoid and Thyroid Hormone Receptors |
DE60113032T2 (en) | 2000-10-30 | 2006-07-06 | Pfizer Products Inc., Groton | Glucocorticoid receptor modulators |
GB0029100D0 (en) * | 2000-11-29 | 2001-01-10 | Karobio Ab | Compounds active at the glucocorticoid receptor |
GB0029102D0 (en) | 2000-11-29 | 2001-01-10 | Karobio Ab | Compounds active at the glucocorticoid receptor |
AU2002219192A1 (en) * | 2000-12-20 | 2002-07-01 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Dissociated glucocorticoid receptor antagonists for the treatment of clucocorticoid associated side-effect |
ES2328795T3 (en) * | 2001-02-14 | 2009-11-18 | Karo Bio Ab | GLUCOCORTICOID RECEIVER MODULATORS. |
US6583180B2 (en) | 2001-02-14 | 2003-06-24 | Abbott Laboratories | Glucocorticoid receptor modulators |
EP1285927A3 (en) | 2001-08-16 | 2005-06-29 | Schering Aktiengesellschaft | Use of glucocorticoid antagonists for the prevention and treatment of diseases of the male reproductive system |
AU2002359730A1 (en) * | 2001-12-21 | 2003-07-30 | Smithkline Beecham Corporation | Compositions and methods for altering glucose production |
ATE381333T1 (en) | 2002-03-26 | 2008-01-15 | Boehringer Ingelheim Pharma | GLUCOCORTICOID MIMETICS, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS AND USE |
US7186864B2 (en) | 2002-05-29 | 2007-03-06 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
US7074806B2 (en) | 2002-06-06 | 2006-07-11 | Boehringer Ingelheim Pharmaceuticals, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
US8097606B2 (en) | 2003-07-23 | 2012-01-17 | Corcept Therapeutics, Inc. | Antiglucocorticoids for the treatment of catatonia |
US7527829B2 (en) | 2003-07-31 | 2009-05-05 | Soken Chemical & Engineering Co., Ltd. | Fluid colloid crystal and process for producing three-dimensional aligned particle mass therefrom |
UY28526A1 (en) | 2003-09-24 | 2005-04-29 | Boehringer Ingelheim Pharma | GLUCOCORTICOID MIMETICS, METHODS OF PREPARATION PHARMACEUTICAL COMPOSITIONS AND USES OF THE SAME |
US7795272B2 (en) | 2004-03-13 | 2010-09-14 | Boehringer Ingelheim Pharmaceutical, Inc. | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof |
PE20060776A1 (en) | 2004-12-27 | 2006-09-26 | Boehringer Ingelheim Pharma | MIMETICS OF GLUCOCORTICOIDES, METHODS TO PREPARE THEM AND PHARMACEUTICAL COMPOSITIONS |
RU2009125614A (en) | 2006-12-06 | 2011-01-20 | Бёрингер Ингельхайм Интернациональ Гмбх (De) | Glucocorticoid mimetics, methods for their preparation, pharmaceutical compositions and their application |
US8268859B2 (en) | 2008-06-06 | 2012-09-18 | Boehringer Ingelheim International Gmbh | Glucocorticoid mimetics, methods of making them, pharmaceutical compositions and uses thereof |
US8138189B2 (en) * | 2009-03-26 | 2012-03-20 | Hoffman-La Roche Inc. | Substituted benzene compounds as modulators of the glucocorticoid receptor |
AU2010280323A1 (en) | 2009-07-31 | 2012-03-08 | Cadila Healthcare Limited | Novel compounds as modulators of glucocorticoid receptors |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4374148A (en) * | 1980-10-21 | 1983-02-15 | Pfizer Inc. | Carboxylic acid therapeutic agents |
US5929058A (en) * | 1996-12-24 | 1999-07-27 | Zymogenetics, Inc. | Treatment agents and methods for treating type II diabetes and symptoms of type II diabetes |
-
1999
- 1999-06-07 JP JP2000553045A patent/JP2002527355A/en active Pending
- 1999-06-07 KR KR1020007013430A patent/KR20010052431A/en not_active Application Discontinuation
- 1999-06-07 CA CA002334116A patent/CA2334116A1/en not_active Abandoned
- 1999-06-07 AU AU41606/99A patent/AU751569B2/en not_active Ceased
- 1999-06-07 IL IL13986599A patent/IL139865A0/en unknown
- 1999-06-07 WO PCT/IB1999/001175 patent/WO1999063976A2/en not_active Application Discontinuation
- 1999-06-07 EP EP99925232A patent/EP1143948A3/en not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
JP2002527355A (en) | 2002-08-27 |
AU4160699A (en) | 1999-12-30 |
AU751569B2 (en) | 2002-08-22 |
KR20010052431A (en) | 2001-06-25 |
EP1143948A3 (en) | 2002-09-11 |
EP1143948A2 (en) | 2001-10-17 |
WO1999063976A2 (en) | 1999-12-16 |
CA2334116A1 (en) | 1999-12-16 |
WO1999063976A3 (en) | 2001-12-20 |
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