HK1134076A1 - - Google Patents
Info
- Publication number
- HK1134076A1 HK1134076A1 HK10100903.4A HK10100903A HK1134076A1 HK 1134076 A1 HK1134076 A1 HK 1134076A1 HK 10100903 A HK10100903 A HK 10100903A HK 1134076 A1 HK1134076 A1 HK 1134076A1
- Authority
- HK
- Hong Kong
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/02—Stomatological preparations, e.g. drugs for caries, aphtae, periodontitis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A—HUMAN NECESSITIES
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P15/16—Masculine contraceptives
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
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- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A—HUMAN NECESSITIES
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- A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
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- A61P9/12—Antihypertensives
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/02—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
- C07D473/04—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
- C07D473/06—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
- C07D473/12—Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1, 3, and 7, e.g. caffeine
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10238243A DE10238243A1 (de) | 2002-08-21 | 2002-08-21 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
DE10312353A DE10312353A1 (de) | 2003-03-20 | 2003-03-20 | 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und deren Verwendung als Arzneimittel |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1134076A1 true HK1134076A1 (sr) | 2010-04-16 |
Family
ID=31947613
Family Applications (6)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK06101985.9A HK1081552A1 (en) | 2002-08-21 | 2006-02-16 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
HK10100903.4A HK1134076A1 (sr) | 2002-08-21 | 2010-01-28 | |
HK10100904.3A HK1134077A1 (en) | 2002-08-21 | 2010-01-28 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]- |
HK13110418.8A HK1183028A1 (zh) | 2002-08-21 | 2013-09-09 | -氨基-哌啶- -基 -黃嘌呤化合物,其製備方法及作為藥物製劑的用途 |
HK16103474.1A HK1215439A1 (zh) | 2002-08-21 | 2016-03-24 | -氨基-哌啶- -基 -黃嘌呤化合物,其製備方法及作為藥物製劑的用途 |
HK18109982.1A HK1250708A1 (zh) | 2002-08-21 | 2018-08-02 | 8-[3-氨基-呱啶-1-基]-黃嘌呤化合物,其製備方法及作為藥物製劑的用途 |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK06101985.9A HK1081552A1 (en) | 2002-08-21 | 2006-02-16 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments |
Family Applications After (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK10100904.3A HK1134077A1 (en) | 2002-08-21 | 2010-01-28 | 8-[3-amino-piperidin-1-yl]-xanthines, the production thereof and the use of the same as medicaments 8-[3---1-]- |
HK13110418.8A HK1183028A1 (zh) | 2002-08-21 | 2013-09-09 | -氨基-哌啶- -基 -黃嘌呤化合物,其製備方法及作為藥物製劑的用途 |
HK16103474.1A HK1215439A1 (zh) | 2002-08-21 | 2016-03-24 | -氨基-哌啶- -基 -黃嘌呤化合物,其製備方法及作為藥物製劑的用途 |
HK18109982.1A HK1250708A1 (zh) | 2002-08-21 | 2018-08-02 | 8-[3-氨基-呱啶-1-基]-黃嘌呤化合物,其製備方法及作為藥物製劑的用途 |
Country Status (38)
Country | Link |
---|---|
EP (6) | EP2308878A3 (sr) |
JP (6) | JP4233524B2 (sr) |
KR (2) | KR101111101B1 (sr) |
CN (4) | CN100522962C (sr) |
AR (3) | AR041025A1 (sr) |
AT (1) | ATE453644T1 (sr) |
AU (2) | AU2003253418B2 (sr) |
BE (1) | BE2011C038I2 (sr) |
BR (2) | BR122012026540B8 (sr) |
CA (1) | CA2496249C (sr) |
CY (3) | CY1109928T1 (sr) |
DE (2) | DE50312295D1 (sr) |
DK (1) | DK1532149T3 (sr) |
EA (3) | EA024251B1 (sr) |
EC (2) | ECSP055617A (sr) |
EG (1) | EG25011A (sr) |
ES (1) | ES2339112T3 (sr) |
FR (1) | FR11C0052I2 (sr) |
HK (6) | HK1081552A1 (sr) |
HR (2) | HRP20050157B1 (sr) |
HU (1) | HUS1100028I1 (sr) |
IL (1) | IL166964A (sr) |
IN (2) | IN2015DN01133A (sr) |
LU (2) | LU91889I2 (sr) |
ME (1) | ME00396B (sr) |
MX (1) | MXPA05001684A (sr) |
MY (2) | MY165643A (sr) |
NO (4) | NO333970B1 (sr) |
PE (1) | PE20040897A1 (sr) |
PL (2) | PL216134B1 (sr) |
PT (1) | PT1532149E (sr) |
RS (2) | RS52142B (sr) |
SA (1) | SA03240448B1 (sr) |
SI (1) | SI1532149T1 (sr) |
TW (3) | TWI469783B (sr) |
UA (1) | UA84275C2 (sr) |
UY (1) | UY27946A1 (sr) |
WO (1) | WO2004018468A2 (sr) |
Families Citing this family (174)
Publication number | Priority date | Publication date | Assignee | Title |
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CN100497336C (zh) * | 2002-05-31 | 2009-06-10 | 先灵公司 | 制备黄嘌呤磷酸二酯酶v抑制剂及其前体的方法 |
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