EA201690357A1 - Лекарственные формы с замедленным высвобождением для ингибитора jak1 - Google Patents

Лекарственные формы с замедленным высвобождением для ингибитора jak1

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Publication number
EA201690357A1
EA201690357A1 EA201690357A EA201690357A EA201690357A1 EA 201690357 A1 EA201690357 A1 EA 201690357A1 EA 201690357 A EA201690357 A EA 201690357A EA 201690357 A EA201690357 A EA 201690357A EA 201690357 A1 EA201690357 A1 EA 201690357A1
Authority
EA
Eurasian Patent Office
Prior art keywords
dosage forms
slow release
jak1 inhibitor
jak1
inhibitor
Prior art date
Application number
EA201690357A
Other languages
English (en)
Russian (ru)
Inventor
Кришнасвами Елесварам
Бхавниш Парих
Дилип П. Моди
Трупти Шетх
Original Assignee
Инсайт Корпорейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Инсайт Корпорейшн filed Critical Инсайт Корпорейшн
Publication of EA201690357A1 publication Critical patent/EA201690357A1/ru

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2031—Organic macromolecular compounds obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyethylene glycol, polyethylene oxide, poloxamers
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    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
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    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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  • Health & Medical Sciences (AREA)
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  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Immunology (AREA)
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  • Rheumatology (AREA)
  • Neurology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Inorganic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Psychiatry (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
EA201690357A 2013-08-07 2014-08-06 Лекарственные формы с замедленным высвобождением для ингибитора jak1 EA201690357A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361863325P 2013-08-07 2013-08-07
US201361913066P 2013-12-06 2013-12-06
PCT/US2014/049940 WO2015021153A1 (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor

Publications (1)

Publication Number Publication Date
EA201690357A1 true EA201690357A1 (ru) 2016-07-29

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EA201690357A EA201690357A1 (ru) 2013-08-07 2014-08-06 Лекарственные формы с замедленным высвобождением для ингибитора jak1

Country Status (31)

Country Link
US (5) US9655854B2 (enExample)
EP (2) EP3030227B1 (enExample)
JP (6) JP6334700B2 (enExample)
KR (3) KR20160045081A (enExample)
CN (3) CN105579032A (enExample)
AU (3) AU2014305989B2 (enExample)
BR (1) BR122020001831A8 (enExample)
CA (2) CA3155500A1 (enExample)
CL (1) CL2016000292A1 (enExample)
CR (3) CR20230316A (enExample)
CY (1) CY1123314T1 (enExample)
DK (1) DK3030227T3 (enExample)
EA (1) EA201690357A1 (enExample)
ES (1) ES2792549T3 (enExample)
HR (1) HRP20200955T1 (enExample)
HU (1) HUE049345T2 (enExample)
IL (2) IL277554B2 (enExample)
LT (1) LT3030227T (enExample)
MX (2) MX394928B (enExample)
MY (2) MY203694A (enExample)
PE (2) PE20220579A1 (enExample)
PH (3) PH12019502074B1 (enExample)
PL (1) PL3030227T3 (enExample)
PT (1) PT3030227T (enExample)
RS (1) RS60469B1 (enExample)
SG (3) SG10201801069QA (enExample)
SI (1) SI3030227T1 (enExample)
SM (1) SMT202000315T1 (enExample)
TW (3) TWI822248B (enExample)
UA (1) UA120499C2 (enExample)
WO (1) WO2015021153A1 (enExample)

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